Target Details
| UniProt AC | P80370 |
|---|---|
| Gene Symbol | DLK1 |
| Protein Name | Protein delta homolog 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00008 (EGF) |
Summary
- Multi-target molecules 211
- Clinical molecules 6
- Avg pChEMBL 7.55
Active Molecules (211)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SJZKCGAAKXNPOE
|
7.6 | IC50 | 2 | — | |
BEKZKKDPYXOBQB
|
7.6 | IC50 | 2 | — | |
VMLPMFIVJNUHLS
|
7.6 | Kd | 2 | — | |
FQRCKINZIWCFBW
|
7.5 | IC50 | 2 | — | |
IHMMZBVEKVDJAY
|
7.5 | IC50 | 2 | — | |
IUHHKZYWPMOFAH
|
7.5 | IC50 | 2 | — | |
UVDYXNFGTOKBLO
|
7.5 | Kd | 2 | — | |
RYJRIIUWHWEFRG
|
7.5 | IC50 | 2 | — | |
BCIDXHNJKHWJJL
|
7.5 | Kd | 2 | — | |
KIKARFDGXOXYJV
|
7.5 | IC50 | 2 | — | |
WBWAOSSZEUARHN
|
7.5 | IC50 | 2 | — | |
PYILNPDKSAJCQB
|
7.5 | IC50 | 2 | — | |
ZDPGILDKHLAGAW
|
7.5 | IC50 | 2 | — | |
IPSIEHCTZGXLQW
|
7.5 | IC50 | 2 | — | |
JAXBPMVTQNGQOE
|
7.5 | Ki | 2 | — | |
SJBKEBVXIUGVOZ
|
7.5 | IC50 | 2 | — | |
WVSYEVKDFSRHMH
|
7.5 | IC50 | 2 | — | |
YRVXIYRJTSIZFV
|
7.5 | IC50 | 2 | — | |
ZIHPELQWBDDGLM
|
7.5 | IC50 | 2 | — | |
GCIKSSRWRFVXBI
|
7.5 | Ki | 109 | Yes | |
MVIPEADYCBLILL
|
7.4 | IC50 | 2 | — | |
RVEPUEJNEZOKJM
|
7.4 | IC50 | 2 | — | |
LXBOBNTVWFNSKG
|
7.4 | IC50 | 2 | — | |
MHXWDVVRMXHYCD
|
7.4 | IC50 | 2 | — | |
YGSNUGAPYIPPAS
|
7.4 | IC50 | 2 | — | |
DGKUXDLHHLKSMP
|
7.4 | Kd | 2 | — | |
XYQFZKHCIZOACR
|
7.4 | IC50 | 2 | — | |
ZQBGYFILGRMBEE
|
7.4 | Kd | 2 | — | |
QQWUGDVOUVUTOY
|
7.4 | Kd | 231 | Yes | |
PFQNAFCKTCFGLS
|
7.4 | Kd | 2 | — | |
YZJXMZFIJMZAGN
|
7.4 | IC50 | 2 | — | |
MZZSOQZFENIENY
|
7.3 | Kd | 2 | — | |
WZFWHOVNHFFCHJ
|
7.3 | IC50 | 2 | — | |
DQMABCFMEBYHLF
|
7.3 | IC50 | 2 | — | |
ITAHIXXTUMBFLW
|
7.3 | Kd | 2 | — | |
GNWLHTMNFDUEGD
|
7.3 | IC50 | 2 | — | |
GVOOHMLKDGUNOS
|
7.2 | IC50 | 2 | — | |
CAGRBVWCHLFWPB
|
7.2 | IC50 | 2 | — | |
GLAAJDCGXKEMNM
|
7.2 | Kd | 2 | — | |
HBBBYGQTCMRVDY
|
7.2 | IC50 | 2 | — | |
NANPYAZEROEITB
|
7.2 | Kd | 2 | — | |
CQFUXFFJWXAJRC
|
7.2 | Kd | 2 | — | |
FHYMWFXNNDZTOE
|
7.2 | IC50 | 2 | — | |
LPMCTRBCMRCSRG
|
7.2 | Kd | 2 | — | |
YYLKKYCXAOBSRM
|
7.2 | Kd | 191 | — | |
HQZNAKDFOFNZRM
|
7.2 | IC50 | 2 | — | |
VOMOOSIWNGQCMM
|
7.2 | IC50 | 2 | — | |
ZZVBIQXZAHZKGS
|
7.1 | IC50 | 2 | — | |
VXERQKDPAMQZBK
|
7.1 | IC50 | 2 | — | |
RIPVLVJVLRJRKH
|
7.1 | Kd | 2 | — |