Target Details
| UniProt AC | P80370 |
|---|---|
| Gene Symbol | DLK1 |
| Protein Name | Protein delta homolog 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00008 (EGF) |
Summary
- Multi-target molecules 211
- Clinical molecules 6
- Avg pChEMBL 7.55
Active Molecules (211)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LYWYGIOUJQXFNS
|
9.8 | Ki | 2 | — | |
MZUKCHWHYOQJRJ
|
9.4 | Ki | 2 | — | |
RHFIAUKMKYHHFA
|
9.0 | Kd | 9 | — | |
FSTMHVBLNXUGCA
|
8.9 | IC50 | 2 | — | |
GSZNVEWIZSZNJT
|
8.8 | IC50 | 2 | — | |
ITGNDUAJIYAXBQ
|
8.7 | IC50 | 2 | — | |
BURDQUKVCPYGRG
|
8.7 | IC50 | 3 | — | |
YZFKEUGDBXWILL
|
8.7 | Kd | 2 | — | |
CDLADWHUVKCMBZ
|
8.7 | IC50 | 2 | — | |
XZJAQIDXESVVQD
|
8.6 | IC50 | 2 | — | |
ABIXESJLYKUXCL
|
8.5 | IC50 | 2 | — | |
HHMAVLGGLJAODV
|
8.5 | IC50 | 2 | — | |
HCDVOAGDQONFDT
|
8.5 | Kd | 4 | — | |
OEWNOSRZQLNNAS
|
8.5 | IC50 | 2 | — | |
YGSNUGAPYIPPAS
|
8.5 | IC50 | 2 | — | |
SBJFXIVTSPDBLG
|
8.5 | IC50 | 2 | — | |
WEFXAEVNJQWAFZ
|
8.5 | IC50 | 2 | — | |
FYFUBZYNKUIYBM
|
8.5 | IC50 | 2 | — | |
MBVVLBMYGYYEIQ
|
8.4 | IC50 | 2 | — | |
CMXUWUGBGXEFFR
|
8.4 | IC50 | 3 | — | |
RVEPUEJNEZOKJM
|
8.4 | IC50 | 2 | — | |
JHEOSCUBGAKVIR
|
8.4 | IC50 | 2 | — | |
PYPUYISPPZTBSN
|
8.4 | IC50 | 2 | — | |
GQFXNVBXLWDSDI
|
8.4 | IC50 | 2 | — | |
PCPSRYQJUUUZDP
|
8.4 | IC50 | 2 | — | |
WLCGZUITPCUAHT
|
8.4 | Kd | 2 | — | |
OJEAHIAKOWKXKB
|
8.4 | IC50 | 2 | — | |
MTONHIAKMBYFEU
|
8.3 | Kd | 2 | — | |
NFNPYHGMNVWRTI
|
8.3 | IC50 | 2 | — | |
HYQKUJQMGQLFRV
|
8.3 | IC50 | 2 | — | |
ANXJEWGRRMFNLA
|
8.3 | IC50 | 2 | — | |
DHLYOTOZLPRAGO
|
8.3 | IC50 | 2 | — | |
SJGUZBLZMWKMLD
|
8.3 | IC50 | 2 | — | |
GJKOCNSRKFGAQL
|
8.3 | Kd | 2 | — | |
JCDUHLOBPFQKTC
|
8.3 | IC50 | 2 | — | |
QQWVKTNSZANSFF
|
8.3 | IC50 | 2 | — | |
UQGIRTPAHIWAPS
|
8.3 | IC50 | 2 | — | |
ARXOCNZUYXHLEU
|
8.2 | IC50 | 2 | — | |
NQHHNMZLRVDZHK
|
8.2 | Kd | 2 | — | |
XEKGZPBWPPGGBY
|
8.2 | IC50 | 2 | — | |
HOAYYWJFTLNUDU
|
8.2 | IC50 | 2 | — | |
KRFONFQVWHHIJW
|
8.2 | IC50 | 2 | — | |
KRSYURVMSJNSNJ
|
8.2 | Kd | 2 | — | |
WINHZLLDWRZWRT
|
8.2 | Ki | 201 | Yes | |
IFYGIDLAXXOLQM
|
8.2 | IC50 | 2 | — | |
LOGWNXFRIGDZFS
|
8.2 | IC50 | 2 | — | |
WMKWBCPSWSWXNF
|
8.2 | IC50 | 2 | — | |
KGGZQEBEACATEW
|
8.2 | IC50 | 2 | — | |
CSOUOHXVYQKYSZ
|
8.1 | IC50 | 2 | — | |
RSDXMMSONYPQFW
|
8.1 | Kd | 2 | — |