Target Details
| UniProt AC | P80192 |
|---|---|
| Gene Symbol | MAP3K9 |
| Protein Name | Mitogen-activated protein kinase kinase kinase 9 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF14604 (SH3_9) |
Summary
- Multi-target molecules 68
- Clinical molecules 14
- Avg pChEMBL 7.08
KEGG Pathways (1)
Active Molecules (68)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HVVKFYHINSILFO
|
6.5 | IC50 | 11 | Yes | |
DOZKSGRZZQMRCD
|
6.5 | IC50 | 2 | — | |
PXLLDBDHYSZSQP
|
6.4 | IC50 | 2 | — | |
ISXAVIPPPMJTPN
|
6.4 | IC50 | 2 | — | |
GCIKSSRWRFVXBI
|
6.4 | Kd | 109 | Yes | |
QQWUGDVOUVUTOY
|
6.4 | Kd | 231 | Yes | |
VAARYSWULJUGST
|
6.4 | Kd | 119 | Yes | |
IJICOKICFQCHBP
|
6.3 | IC50 | 2 | — | |
LEXMMFPAPDGYGZ
|
6.2 | IC50 | 7 | — | |
XCOSAQGGGZDYJN
|
6.2 | IC50 | 11 | — | |
GSHILQCUENBVBZ
|
6.2 | IC50 | 2 | — | |
YYLKKYCXAOBSRM
|
6.2 | Kd | 191 | — | |
HCBIATVCCJRSKR
|
6.0 | IC50 | 5 | — | |
CXQHYVUVSFXTMY
|
6.0 | Kd | 154 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
SEJGTFPOEJWEGG
|
6.0 | Kd | 149 | — |