Target Details
| UniProt AC | P80192 |
|---|---|
| Gene Symbol | MAP3K9 |
| Protein Name | Mitogen-activated protein kinase kinase kinase 9 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF14604 (SH3_9) |
Summary
- Multi-target molecules 68
- Clinical molecules 14
- Avg pChEMBL 7.08
KEGG Pathways (1)
Active Molecules (68)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NXSJMRCTGYTSTK
|
8.7 | Kd | 200 | — | |
OSVUGUHRKMMBSE
|
8.5 | Kd | 170 | — | |
UIARLYUEJFELEN
|
8.5 | Kd | 289 | Yes | |
NHHQJBCNYHBUSI
|
8.4 | Kd | 220 | — | |
HKSZLNNOFSGOKW
|
8.0 | IC50 | 408 | — | |
HKSZLNNOFSGOKW
|
8.0 | Kd | 213 | — | |
OCMCHCVNRKLMAQ
|
7.9 | IC50 | 4 | — | |
BMGQWWVMWDBQGC
|
7.8 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
7.8 | Kd | 91 | Yes | |
JZCWLJDSIRUGIN
|
7.8 | Ki | 16 | — | |
SIBOQVCECFIQAO
|
7.8 | IC50 | 2 | — | |
ZZSBPGIGIUFJRA
|
7.8 | Kd | 46 | — | |
MDAFGVXLBFQEJH
|
7.8 | IC50 | 4 | — | |
CVXZWDPKRAIHOI
|
7.7 | IC50 | 4 | — | |
QKKIWEILHCXECO
|
7.7 | IC50 | 24 | — | |
KOZFSFOOLUUIGY
|
7.7 | IC50 | 26 | — | |
KOZFSFOOLUUIGY
|
7.7 | IC50 | 88 | Yes | |
NHDDTLMPCVOXFH
|
7.7 | IC50 | 16 | Yes | |
HSWWFIPPMAFLPH
|
7.6 | IC50 | 2 | — | |
UFLRHQRKTYVKGB
|
7.5 | IC50 | 4 | — | |
WVXNSAVVKYZVOE
|
7.5 | IC50 | 92 | — | |
SCMLRESZJCKCTC
|
7.4 | IC50 | 7 | — | |
LYFDGRJCBMWOKJ
|
7.4 | IC50 | 3 | — | |
FZBVNCFBCNXULH
|
7.3 | IC50 | 18 | — | |
SIHPNVHZKXZMMW
|
7.3 | IC50 | 3 | — | |
VZJUKEQMHBEIKH
|
7.3 | IC50 | 2 | — | |
RAOJISQDGOOXTK
|
7.3 | IC50 | 14 | Yes | |
OHNNRNYUHNGDNO
|
7.3 | IC50 | 15 | — | |
APPXQUDJLJXULP
|
7.3 | IC50 | 47 | — | |
TXGKRVFSSHPBAJ
|
7.2 | IC50 | 11 | — | |
BFKOYMDZLSTZJN
|
7.2 | IC50 | 2 | — | |
JJQPROAZGIYDBL
|
7.2 | IC50 | 4 | — | |
RHFIAUKMKYHHFA
|
7.2 | IC50 | 9 | — | |
NBGYLHIDCLVBHE
|
7.2 | IC50 | 6 | Yes | |
FWLMVFUGMHIOAA
|
7.1 | IC50 | 26 | — | |
XIKCRRWSJXYZMA
|
7.0 | IC50 | 2 | — | |
SRZPGKHRQCVEAS
|
7.0 | IC50 | 2 | — | |
QMLALHXGVBGFIC
|
7.0 | IC50 | 2 | — | |
WENCWJUIDFEPSK
|
7.0 | IC50 | 3 | — | |
MEXUTNIFSHFQRG
|
6.9 | IC50 | 21 | Yes | |
ZTSOUDMNSOYCTG
|
6.8 | IC50 | 10 | — | |
FPXKTABMRKRDJN
|
6.8 | IC50 | 2 | — | |
ABMSAGZBJYEZGT
|
6.8 | IC50 | 4 | — | |
PKGQDPNUCJTZSZ
|
6.7 | IC50 | 2 | — | |
AILRADAXUVEEIR
|
6.7 | IC50 | 75 | — | |
XZXHXSATPCNXJR
|
6.7 | Kd | 165 | Yes | |
YOVVNQKCSKSHKT
|
6.6 | IC50 | 15 | — | |
CJQGLUJHMXCLQY
|
6.6 | IC50 | 11 | — | |
CUIHSIWYWATEQL
|
6.5 | Kd | 61 | Yes | |
CMAAJKFJPMUHEN
|
6.5 | IC50 | 3 | — |