Target Details
| UniProt AC | P78536 |
|---|---|
| Gene Symbol | ADAM17 |
| Protein Name | Disintegrin and metalloproteinase domain-containing protein 17 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF16698 (ADAM17_MPD) PF00200 (Disintegrin) PF13574 (Reprolysin_2) |
Summary
- Multi-target molecules 785
- Clinical molecules 566
- Avg pChEMBL 7.43
KEGG Pathways (6)
Associated Diseases (2)
Active Molecules (785)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UFJYSWCFYDZPKS
|
7.5 | IC50 | 4 | Yes | |
DKBDATWDEJHFQS
|
7.5 | IC50 | 2 | — | |
MQLHBSAEUUVJRX
|
7.5 | IC50 | 6 | Yes | |
ZYZUZMRFPDIWGW
|
7.5 | IC50 | 5 | Yes | |
AWDZLFOJMUGNPS
|
7.4 | IC50 | 6 | Yes | |
BODLESUVCQEUII
|
7.4 | IC50 | 7 | Yes | |
FSJPBIIVCZKHRS
|
7.4 | IC50 | 2 | — | |
RIYWMJMELHHCTR
|
7.4 | IC50 | 2 | — | |
DPQCHTZYBRQXQC
|
7.4 | Ki | 7 | Yes | |
HQUNVDQSUFWCJN
|
7.4 | IC50 | 2 | — | |
IAZFWEJODMHVIO
|
7.4 | Ki | 7 | Yes | |
JRFZSMAIBXKQOW
|
7.4 | IC50 | 3 | — | |
JTOKTYOQJGJDGG
|
7.4 | IC50 | 3 | — | |
KJFHTZIVTSKATM
|
7.4 | IC50 | 5 | Yes | |
RUAWTWDABHALSY
|
7.4 | IC50 | 3 | — | |
VUCZYOBGSLKTCS
|
7.4 | IC50 | 2 | — | |
RLUGMDBAWBLDJQ
|
7.4 | IC50 | 5 | Yes | |
WUQMFARMJJXJMN
|
7.4 | IC50 | 6 | Yes | |
KHORRYDPPCADSY
|
7.4 | IC50 | 5 | Yes | |
GHZXWVPNZMUKBT
|
7.4 | IC50 | 5 | Yes | |
LHUIUEQQDGBKCU
|
7.4 | IC50 | 5 | Yes | |
LWZOHIDILGLXGF
|
7.4 | IC50 | 5 | Yes | |
NRCQPJPKKZDRND
|
7.4 | IC50 | 6 | Yes | |
RBLCSCFFNCADJO
|
7.4 | IC50 | 5 | — | |
SMZPWUUYPYYHIV
|
7.4 | IC50 | 5 | Yes | |
WOZRCMBDSXXEAJ
|
7.4 | Ki | 6 | Yes | |
OUIRYNJKZCTIHG
|
7.4 | IC50 | 5 | Yes | |
RBLCSCFFNCADJO
|
7.4 | IC50 | 5 | — | |
AIBDPCDNFOFGFS
|
7.4 | Ki | 6 | Yes | |
AVQCFDJVRXAPJO
|
7.4 | IC50 | 5 | Yes | |
IXEFVZDHNHSUSD
|
7.4 | IC50 | 5 | Yes | |
QRXOZHSEEGNRFC
|
7.4 | IC50 | 8 | Yes | |
SHTYCRVVDNRZDY
|
7.4 | IC50 | 5 | Yes | |
WGPIMMRNIAYWBT
|
7.4 | IC50 | 5 | Yes | |
YBQLENDMILTZBB
|
7.4 | IC50 | 6 | Yes | |
CZYVJSTWDMVAFM
|
7.4 | IC50 | 6 | Yes | |
LMASIGSKSCEZDY
|
7.4 | IC50 | 5 | Yes | |
NUWGCPAPIJNAPL
|
7.4 | IC50 | 2 | — | |
GZISYEQJJGPWOA
|
7.3 | IC50 | 2 | Yes | |
WLWNRAWQDZRXMB
|
7.3 | IC50 | 6 | Yes | |
MDOGBVLWCBWUMC
|
7.3 | IC50 | 5 | Yes | |
UZCHBPQXZPPPNZ
|
7.3 | IC50 | 2 | — | |
YYOVZJXOBZVIQK
|
7.3 | IC50 | 3 | — | |
HDTMIVHMPQVMJD
|
7.3 | IC50 | 6 | Yes | |
MJYIMHGWKZRGTK
|
7.3 | IC50 | 2 | — | |
QAFRSDWNZLQCBN
|
7.3 | IC50 | 6 | Yes | |
PTSHMCCZVCAMNJ
|
7.3 | Ki | 6 | Yes | |
YINOLIYDTHQXKP
|
7.3 | IC50 | 2 | — | |
JQLHAXGMYALIFJ
|
7.3 | IC50 | 3 | — | |
ZWHIVWLHYJCFFA
|
7.3 | IC50 | 5 | Yes |