Target Details
| UniProt AC | P78536 |
|---|---|
| Gene Symbol | ADAM17 |
| Protein Name | Disintegrin and metalloproteinase domain-containing protein 17 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF16698 (ADAM17_MPD) PF00200 (Disintegrin) PF13574 (Reprolysin_2) |
Summary
- Multi-target molecules 785
- Clinical molecules 566
- Avg pChEMBL 7.43
KEGG Pathways (6)
Associated Diseases (2)
Active Molecules (785)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DOFYUNJDVUXVMB
|
7.6 | IC50 | 5 | Yes | |
KADFIIKJGHEHDF
|
7.6 | Ki | 7 | Yes | |
KNCYWVRUUBOHGE
|
7.6 | IC50 | 7 | Yes | |
PYSVMZGECWVLOT
|
7.6 | IC50 | 4 | Yes | |
UNINFAIJOLFFHN
|
7.6 | IC50 | 5 | Yes | |
ZMAYDSCNOCAOHA
|
7.6 | IC50 | 5 | Yes | |
ZTVJLUOPMWIKSV
|
7.6 | IC50 | 6 | Yes | |
FYYONZZUDPFMJO
|
7.6 | IC50 | 5 | Yes | |
LJOOWNHZCTUDSG
|
7.6 | IC50 | 3 | — | |
MCYLJYADJGYSSU
|
7.6 | IC50 | 2 | — | |
JNFDCDGQVIEXPD
|
7.6 | IC50 | 5 | Yes | |
SHBOXSNAYNDDGN
|
7.6 | IC50 | 2 | — | |
UOLICGDBHYFWJG
|
7.6 | IC50 | 2 | — | |
DPCXVXNEMYTZOE
|
7.6 | IC50 | 6 | Yes | |
HEYGZWVOCCBCPY
|
7.6 | IC50 | 6 | Yes | |
JIZLXLHASQJXJD
|
7.6 | IC50 | 2 | — | |
MKEVHBFZBURDHJ
|
7.6 | IC50 | 2 | — | |
QCHHXEMLMRDLDA
|
7.6 | IC50 | 6 | Yes | |
ZLSOXSXSNCNKSX
|
7.6 | IC50 | 6 | Yes | |
NCKDXXIBASBEEV
|
7.6 | Ki | 6 | Yes | |
IPBVPRHDESNKFG
|
7.6 | Ki | 6 | Yes | |
BLIQFUCBRCDFAI
|
7.5 | Ki | 5 | Yes | |
CYIOQNVVHKTYRH
|
7.5 | IC50 | 5 | Yes | |
DCDJWNFOPNVBIM
|
7.5 | IC50 | 4 | Yes | |
FPHXOEUJYCDFQF
|
7.5 | IC50 | 4 | Yes | |
GHBQSNPRMVUGFE
|
7.5 | IC50 | 2 | — | |
IUPDLWWZWJCNBN
|
7.5 | IC50 | 2 | — | |
KEEWWGMUNANVLU
|
7.5 | IC50 | 5 | Yes | |
LCTLPROJUJRGOK
|
7.5 | IC50 | 3 | Yes | |
LCTLPROJUJRGOK
|
7.5 | IC50 | 3 | Yes | |
SQODILRODCBOCF
|
7.5 | IC50 | 5 | Yes | |
YCIYENASUWAOBH
|
7.5 | IC50 | 5 | Yes | |
YTTGWCXMRQNZJI
|
7.5 | IC50 | 5 | Yes | |
CVMOEYXHQALNTG
|
7.5 | Ki | 6 | Yes | |
XDKNQAWYSUZUDU
|
7.5 | IC50 | 3 | Yes | |
FROMXYGXLCSILK
|
7.5 | IC50 | 3 | — | |
LVVFBDASYOIWFN
|
7.5 | IC50 | 4 | Yes | |
UICCGUSKKDLVIN
|
7.5 | IC50 | 6 | Yes | |
TXFHRXOVMCSUEC
|
7.5 | Ki | 2 | — | |
YPFZRQMUNBCBEG
|
7.5 | Ki | 6 | Yes | |
YXMRNZNQTDDTSA
|
7.5 | IC50 | 5 | Yes | |
JXCARHJPSZBVFH
|
7.5 | IC50 | 6 | Yes | |
ZWHGUGYVAMXPJZ
|
7.5 | IC50 | 5 | Yes | |
FITSVZFOIGFQQI
|
7.5 | Ki | 6 | Yes | |
AHKGXKHDKHAJDE
|
7.5 | IC50 | 3 | — | |
DIHHYKCLOAQWIB
|
7.5 | IC50 | 4 | Yes | |
HFKQCTSECBMUHK
|
7.5 | IC50 | 4 | Yes | |
IVXFVTBAZBQGPK
|
7.5 | IC50 | 5 | Yes | |
NQUUIXIBNFFYTG
|
7.5 | Ki | 6 | Yes | |
GCDCQOTVUSLXRJ
|
7.5 | IC50 | 4 | Yes |