Target Details
| UniProt AC | P78536 |
|---|---|
| Gene Symbol | ADAM17 |
| Protein Name | Disintegrin and metalloproteinase domain-containing protein 17 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF16698 (ADAM17_MPD) PF00200 (Disintegrin) PF13574 (Reprolysin_2) |
Summary
- Multi-target molecules 785
- Clinical molecules 566
- Avg pChEMBL 7.43
KEGG Pathways (6)
Associated Diseases (2)
Active Molecules (785)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PBCSMBZCRUWUMR
|
7.8 | IC50 | 2 | — | |
PBCSMBZCRUWUMR
|
7.8 | IC50 | 2 | — | |
ROSNVSQTEGHUKU
|
7.8 | IC50 | 12 | Yes | |
RZISBFWRHNXABZ
|
7.8 | IC50 | 3 | Yes | |
VOBFYBKSOTYYNL
|
7.8 | IC50 | 2 | — | |
ZAUSLRXPYLUTHB
|
7.8 | IC50 | 6 | Yes | |
ZAXFGRVMMQJZLL
|
7.8 | IC50 | 5 | Yes | |
OIGNJSKKLXVSLS
|
7.8 | IC50 | 7 | — | |
AOGWJSJATLXUOJ
|
7.8 | IC50 | 6 | Yes | |
BXQLLVHURXNRLY
|
7.8 | IC50 | 4 | Yes | |
IDKUTWZTCGVYET
|
7.8 | IC50 | 5 | Yes | |
MGQZHWBYKGXMDX
|
7.8 | IC50 | 5 | Yes | |
NYRVSWKULSLJMD
|
7.8 | IC50 | 3 | Yes | |
VAMKUUUJVOOTKN
|
7.8 | IC50 | 5 | Yes | |
KMYAHTGTYRRWEK
|
7.8 | Ki | 6 | Yes | |
BGNATPVKWHRROW
|
7.8 | Ki | 6 | Yes | |
PDBHRMUGMOPNOC
|
7.8 | IC50 | 5 | Yes | |
PRQWPDFKJBVNKQ
|
7.8 | IC50 | 6 | Yes | |
QPWBTJDQYIYLND
|
7.8 | IC50 | 4 | — | |
UBBKFTZMBAKVDC
|
7.8 | IC50 | 6 | Yes | |
DWBZTKJXPJGGSU
|
7.8 | IC50 | 6 | Yes | |
GHKVZKUXCOXDAW
|
7.8 | IC50 | 6 | Yes | |
KTMMYBDZBIJPLY
|
7.8 | IC50 | 4 | Yes | |
LOQCMKWGWBMVPA
|
7.8 | IC50 | 4 | Yes | |
NSLCGVDBXCHQFK
|
7.8 | Ki | 2 | — | |
QEWCDBOSGBDOOY
|
7.8 | IC50 | 5 | Yes | |
SMRKDKVRUIEVHG
|
7.8 | IC50 | 5 | Yes | |
BTZMVJPRQAIPRP
|
7.7 | IC50 | 5 | Yes | |
RZAVXBHMHDOVTM
|
7.7 | IC50 | 2 | — | |
XMKAMECIIHUBSZ
|
7.7 | IC50 | 5 | Yes | |
GBGAKFWYCGVPHY
|
7.7 | IC50 | 7 | Yes | |
GMNFREWQYNXZAF
|
7.7 | Ki | 7 | Yes | |
IJIWBJJLSPLOBZ
|
7.7 | IC50 | 2 | — | |
JGAIDLBSMBNOAG
|
7.7 | IC50 | 4 | Yes | |
JKWHUKMFJPDCMY
|
7.7 | IC50 | 5 | Yes | |
KLSLMSQYLRDFGN
|
7.7 | IC50 | 5 | Yes | |
ROWNCZWVCCMTQI
|
7.7 | IC50 | 5 | Yes | |
AHCJFAZGYUITPV
|
7.7 | Ki | 6 | Yes | |
DWAPKTBJQHYHER
|
7.7 | IC50 | 6 | Yes | |
QBIHWFSRXVWUDN
|
7.7 | IC50 | 3 | Yes | |
UFYJMKIWYONTIU
|
7.7 | IC50 | 5 | Yes | |
UWHDYIJAXRNLQS
|
7.7 | Ki | 6 | Yes | |
VDJRMQXPNKTLQA
|
7.7 | IC50 | 5 | Yes | |
LOTUNSOIIWVNBG
|
7.7 | IC50 | 2 | — | |
IISMJBOLNRKABL
|
7.7 | Ki | 6 | Yes | |
IXKRFERDVUXQLW
|
7.7 | IC50 | 6 | Yes | |
YFXAPTTTXDTWSV
|
7.7 | Ki | 6 | Yes | |
FABJTKDLHAAFNV
|
7.7 | Ki | 6 | Yes | |
HZRAYMWLJLWNAA
|
7.7 | IC50 | 5 | Yes | |
NYJKRUFCTNREQN
|
7.7 | IC50 | 3 | Yes |