Target Details
| UniProt AC | P78536 |
|---|---|
| Gene Symbol | ADAM17 |
| Protein Name | Disintegrin and metalloproteinase domain-containing protein 17 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF16698 (ADAM17_MPD) PF00200 (Disintegrin) PF13574 (Reprolysin_2) |
Summary
- Multi-target molecules 785
- Clinical molecules 566
- Avg pChEMBL 7.43
KEGG Pathways (6)
Associated Diseases (2)
Active Molecules (785)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HPBWNXRDTAWPAP
|
8.0 | IC50 | 3 | Yes | |
JRSOKCXTAIQJPK
|
8.0 | IC50 | 4 | Yes | |
LAGAITXTFHYXGS
|
8.0 | IC50 | 5 | Yes | |
UWPHCZNYIWQCKD
|
8.0 | IC50 | 5 | Yes | |
VMOSDDURWLNMNG
|
8.0 | IC50 | 5 | Yes | |
XVBKVNVPXQZYQF
|
8.0 | IC50 | 5 | Yes | |
YHQKAILNGYAYKF
|
8.0 | Ki | 3 | Yes | |
FODLAGUBVKDEIZ
|
8.0 | IC50 | 5 | Yes | |
IQHWFMFCBUDMAF
|
8.0 | Ki | 6 | Yes | |
JMJKKHVSMQBPSU
|
8.0 | IC50 | 6 | Yes | |
KQVRGIRNMDCIEB
|
8.0 | Ki | 3 | Yes | |
LFDHAXXLFUSQRL
|
8.0 | IC50 | 5 | Yes | |
LIKQSFURRNSUMR
|
8.0 | Ki | 2 | — | |
MRBPTYYVXXZQBB
|
8.0 | IC50 | 5 | Yes | |
NUDMVYOFBGJGMN
|
8.0 | IC50 | 5 | Yes | |
VUYBRUBUOZYSQS
|
8.0 | IC50 | 4 | Yes | |
YKPYIPVDTNNYCN
|
8.0 | IC50 | 11 | Yes | |
YSMSZPWEAVKTEN
|
8.0 | IC50 | 4 | Yes | |
ZXORTEVXPYNWIB
|
8.0 | IC50 | 5 | Yes | |
MXGYLPKHTGTZKG
|
8.0 | Ki | 7 | Yes | |
AYWKRESAZCSENH
|
7.9 | IC50 | 4 | Yes | |
BRHXKZALFBLRIF
|
7.9 | IC50 | 5 | Yes | |
BUDIJDXJWOVXRJ
|
7.9 | IC50 | 3 | Yes | |
DNUKGGCABDLAEO
|
7.9 | IC50 | 4 | Yes | |
JQGYJNKTRDAQCV
|
7.9 | IC50 | 5 | Yes | |
LQRPHHDGTPYXHT
|
7.9 | IC50 | 5 | Yes | |
LQZDEWIIFWHTLX
|
7.9 | IC50 | 4 | Yes | |
LZUHYMGQNXWOHQ
|
7.9 | IC50 | 6 | — | |
MCUUTMPQGFSADF
|
7.9 | IC50 | 3 | Yes | |
QFTWPDUNHCKGKX
|
7.9 | IC50 | 6 | Yes | |
QUEIBYWBRFSDLX
|
7.9 | IC50 | 6 | Yes | |
RBRFAUFMZOIMMS
|
7.9 | IC50 | 3 | — | |
SSQXFNKOLMHXPO
|
7.9 | Ki | 6 | Yes | |
XPKONFJMLMUKJB
|
7.9 | IC50 | 2 | — | |
YJPYNLASIFTSPY
|
7.9 | IC50 | 2 | — | |
GPENKXZRTRUYOG
|
7.9 | IC50 | 4 | Yes | |
KRUUUOUZTDKUCF
|
7.9 | IC50 | 5 | Yes | |
LRYRCUJGWNCKPO
|
7.9 | IC50 | 5 | Yes | |
MOODLLAARDEUNJ
|
7.9 | Ki | 6 | Yes | |
NITYDPDXAAFEIT
|
7.9 | IC50 | 20 | Yes | |
VCKCQHDSLLCTDH
|
7.9 | IC50 | 6 | Yes | |
VJCSPSPTFYXXJB
|
7.9 | IC50 | 6 | Yes | |
IBUXWZOBVVWCHD
|
7.9 | Ki | 7 | Yes | |
JFMSSTVXWKCAJH
|
7.9 | Ki | 7 | Yes | |
AXHCVGDTGFVLIU
|
7.8 | IC50 | 5 | Yes | |
BVVZNDQVRQLIPW
|
7.8 | IC50 | 4 | Yes | |
DWFUVVZGNJNHKO
|
7.8 | Ki | 7 | Yes | |
IKRKDUGQVRSGJX
|
7.8 | IC50 | 2 | — | |
ISBRGXFRKARDDV
|
7.8 | IC50 | 5 | Yes | |
NFUSRQFYPZGOLU
|
7.8 | IC50 | 3 | Yes |