Target Details
| UniProt AC | P78536 |
|---|---|
| Gene Symbol | ADAM17 |
| Protein Name | Disintegrin and metalloproteinase domain-containing protein 17 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF16698 (ADAM17_MPD) PF00200 (Disintegrin) PF13574 (Reprolysin_2) |
Summary
- Multi-target molecules 785
- Clinical molecules 566
- Avg pChEMBL 7.43
KEGG Pathways (6)
Associated Diseases (2)
Active Molecules (785)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
TXTZEVLHPGQYAR
|
8.2 | IC50 | 6 | Yes | |
XQUSEXYSIGIEBX
|
8.2 | IC50 | 4 | Yes | |
KAJAADJOOYZIPJ
|
8.2 | IC50 | 4 | Yes | |
UVFPNZAMZZIJLE
|
8.2 | IC50 | 3 | Yes | |
CDUNTBSHRUTDFM
|
8.2 | Ki | 7 | Yes | |
CLSBMSGIRGYRMI
|
8.2 | IC50 | 3 | Yes | |
KHAOJBRQDUCAFK
|
8.2 | IC50 | 4 | Yes | |
LUOBAMXDTNOZAD
|
8.2 | IC50 | 2 | — | |
LBQUSUPCYKIDFL
|
8.2 | IC50 | 4 | Yes | |
ZMDMPUVIZFSSCM
|
8.2 | IC50 | 4 | Yes | |
DOOZILOLHOKUGO
|
8.2 | IC50 | 4 | Yes | |
HUBNMJYLBBXLHV
|
8.2 | IC50 | 6 | Yes | |
JOILTJHUYYDODY
|
8.2 | IC50 | 2 | — | |
LKFNHCFYLDRUTH
|
8.2 | IC50 | 4 | Yes | |
RBLCSCFFNCADJO
|
8.2 | Ki | 7 | Yes | |
VRUQYJXYEALKCT
|
8.2 | IC50 | 6 | Yes | |
ZEZNNQDUSMNIDE
|
8.2 | IC50 | 5 | Yes | |
ZOPDCQZNGWSOLM
|
8.2 | IC50 | 5 | Yes | |
BHRJTBRTTVQRNI
|
8.1 | IC50 | 5 | Yes | |
KPWHSOUKRWDBAT
|
8.1 | IC50 | 2 | — | |
MVPVFNYLHBJBHV
|
8.1 | IC50 | 5 | Yes | |
COUUBDFXGTZTPW
|
8.1 | Ki | 5 | Yes | |
CVZIHNYAZLXRRS
|
8.1 | IC50 | 10 | Yes | |
CVZIHNYAZLXRRS
|
8.1 | IC50 | 6 | Yes | |
FWJFNXPZKLJJSG
|
8.1 | IC50 | 6 | Yes | |
GYSTVJYXBPSVIF
|
8.1 | Ki | 4 | — | |
KIKBZIXCMWKZEI
|
8.1 | IC50 | 6 | Yes | |
LXKHXLQQHKRMFP
|
8.1 | Ki | 7 | Yes | |
PPNXUTAPILQZQN
|
8.1 | IC50 | 3 | Yes | |
QSFJZGINKPYVRC
|
8.1 | Ki | 7 | Yes | |
VNCIHKLPBWTDIP
|
8.1 | IC50 | 6 | Yes | |
XSFCSVRJCFLQJI
|
8.1 | IC50 | 3 | Yes | |
YTRMRJDVKQXSIU
|
8.1 | IC50 | 4 | Yes | |
ZLIOUDYFRDHHSM
|
8.1 | IC50 | 6 | Yes | |
NIBQFPHLKYOWJP
|
8.1 | IC50 | 4 | Yes | |
AHSZJHCTCQGTRY
|
8.1 | Ki | 4 | Yes | |
LEMMSOIQHPOJRA
|
8.1 | IC50 | 3 | Yes | |
HAKDXLDJTCFTIE
|
8.1 | IC50 | 3 | Yes | |
JEFVBTZAXMPPTH
|
8.1 | IC50 | 4 | Yes | |
LAQQWJARJKOYJJ
|
8.1 | IC50 | 6 | Yes | |
MKUAQMILBQCRIR
|
8.1 | IC50 | 2 | — | |
RTKNMWBYPISZDZ
|
8.1 | Ki | 7 | Yes | |
WRDNQNGMPREKKZ
|
8.1 | IC50 | 4 | Yes | |
XRGWUGBXRHDGDG
|
8.1 | IC50 | 6 | Yes | |
XRLMAIWPTHLVKY
|
8.0 | IC50 | 5 | Yes | |
AXPBXFSDSKBQDG
|
8.0 | IC50 | 5 | Yes | |
BLQAAMGUGMNRQN
|
8.0 | IC50 | 6 | Yes | |
CARKQNSZFCLNKM
|
8.0 | Ki | 3 | Yes | |
CCGWFLCBYDXLBZ
|
8.0 | IC50 | 5 | Yes | |
DQDPBMDGDOPPLK
|
8.0 | Ki | 7 | Yes |