Target Details
| UniProt AC | P78536 |
|---|---|
| Gene Symbol | ADAM17 |
| Protein Name | Disintegrin and metalloproteinase domain-containing protein 17 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF16698 (ADAM17_MPD) PF00200 (Disintegrin) PF13574 (Reprolysin_2) |
Summary
- Multi-target molecules 785
- Clinical molecules 566
- Avg pChEMBL 7.43
KEGG Pathways (6)
Associated Diseases (2)
Active Molecules (785)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AGMWQNDXCWDRDZ
|
8.5 | IC50 | 3 | Yes | |
LTVIJEFEZVFIST
|
8.5 | IC50 | 14 | Yes | |
OIJUXVJLPZUPIP
|
8.5 | IC50 | 3 | Yes | |
BNKOGVVBAYMLMZ
|
8.5 | IC50 | 6 | Yes | |
FTWOUUKMIDBQOJ
|
8.5 | IC50 | 2 | — | |
NMAKKNGSMZZSBP
|
8.5 | IC50 | 4 | Yes | |
CBEZXYHTYKUDTE
|
8.5 | IC50 | 3 | Yes | |
OCSMOTCMPXTDND
|
8.4 | IC50 | 14 | Yes | |
BQDVTMRZPWSYOT
|
8.4 | IC50 | 7 | — | |
BDLXCRNZHKNUCS
|
8.4 | IC50 | 3 | Yes | |
BXLWVAKSQMYQKF
|
8.4 | Ki | 5 | Yes | |
FNRFZJFDQHKMHF
|
8.4 | IC50 | 5 | Yes | |
RBRFAUFMZOIMMS
|
8.4 | IC50 | 2 | — | |
RBRFAUFMZOIMMS
|
8.4 | IC50 | 3 | — | |
RBRFAUFMZOIMMS
|
8.4 | IC50 | 3 | Yes | |
UFOCAFMHHPCHKN
|
8.4 | IC50 | 3 | Yes | |
VMMAOHBHWSKMLW
|
8.4 | IC50 | 4 | Yes | |
WICQDDCNCVTFDX
|
8.4 | Ki | 16 | Yes | |
ZXFJUXBYVRDBQU
|
8.4 | IC50 | 2 | Yes | |
MDENDLKFAFTBOF
|
8.4 | IC50 | 2 | — | |
YKVNFNGMIAJYOQ
|
8.4 | IC50 | 6 | Yes | |
SCRXVDGCFAHYTL
|
8.4 | IC50 | 2 | — | |
YFYQFPIGOKJLFD
|
8.3 | IC50 | 3 | Yes | |
YLPGDDBCDVVMDA
|
8.3 | IC50 | 4 | Yes | |
GKLAUAGSCYZMQP
|
8.3 | Ki | 7 | Yes | |
KSOLTKWEALJMDR
|
8.3 | IC50 | 5 | Yes | |
DNEUAPIVDBXPFN
|
8.3 | Ki | 2 | — | |
FAEZTVRCESNVJN
|
8.3 | IC50 | 6 | Yes | |
JLPMPXKOGZSSRK
|
8.3 | IC50 | 6 | Yes | |
KTCRMROJXXSPQJ
|
8.3 | Ki | 6 | Yes | |
MAVDNGWEBZTACC
|
8.3 | IC50 | 6 | — | |
RMUMGJZUGCOZOV
|
8.3 | IC50 | 6 | Yes | |
RXYVRCSDLULANF
|
8.3 | IC50 | 2 | — | |
RYUNWXPVOIGBCD
|
8.3 | IC50 | 4 | Yes | |
SEOIKBYFTLCBTF
|
8.3 | IC50 | 6 | Yes | |
LOMOBWUKCBVLNJ
|
8.3 | IC50 | 5 | Yes | |
WFARRRAQEGQWNJ
|
8.3 | IC50 | 4 | Yes | |
IOLRUMINDIUCLJ
|
8.3 | IC50 | 8 | Yes | |
YFKTVOCECCSHLJ
|
8.3 | IC50 | 3 | Yes | |
VRQPNJFSKYEBCN
|
8.2 | IC50 | 3 | Yes | |
JQJWNYAMOJOHCE
|
8.2 | IC50 | 4 | Yes | |
KLUBFNJJJWONQA
|
8.2 | IC50 | 4 | Yes | |
AYPPVQRNMZPQMU
|
8.2 | IC50 | 6 | Yes | |
FHAJCDXKKGQJQW
|
8.2 | IC50 | 5 | Yes | |
FUDBZSGMQCENEH
|
8.2 | IC50 | 6 | Yes | |
GRFJGGIFOFQTRL
|
8.2 | IC50 | 3 | Yes | |
JERYKMOBMXUTFQ
|
8.2 | IC50 | 6 | Yes | |
LIJQQAFTSYEDRO
|
8.2 | IC50 | 6 | Yes | |
QXSADLFWPARWTP
|
8.2 | IC50 | 6 | Yes | |
RSGVYIJLQVPSNJ
|
8.2 | IC50 | 4 | Yes |