Target Details
| UniProt AC | P78536 |
|---|---|
| Gene Symbol | ADAM17 |
| Protein Name | Disintegrin and metalloproteinase domain-containing protein 17 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF16698 (ADAM17_MPD) PF00200 (Disintegrin) PF13574 (Reprolysin_2) |
Summary
- Multi-target molecules 785
- Clinical molecules 566
- Avg pChEMBL 7.43
KEGG Pathways (6)
Associated Diseases (2)
Active Molecules (785)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LNPBBURQSUEIHO
|
8.8 | IC50 | 5 | Yes | |
SQWKFISUTRRKSE
|
8.8 | IC50 | 2 | Yes | |
MGIMQKIBRRRYRM
|
8.7 | IC50 | 4 | Yes | |
UBFGIEDUTRCMEQ
|
8.7 | IC50 | 3 | — | |
ZUMRSIZQUOZFGG
|
8.7 | IC50 | 3 | Yes | |
RFJSQAZBRWXDMS
|
8.7 | Ki | 4 | Yes | |
WZZROHGXDJBEMY
|
8.7 | Ki | 6 | Yes | |
UTAGRFZAWOLQHO
|
8.7 | IC50 | 4 | Yes | |
BKTXYTRQOBRSNS
|
8.7 | IC50 | 2 | — | |
CIPRRERRNXDHQR
|
8.7 | IC50 | 3 | Yes | |
DVAPUVGZYOTZOY
|
8.7 | IC50 | 4 | Yes | |
LJJFKNOMQHHBEW
|
8.7 | IC50 | 4 | Yes | |
LWFCUEQJXZSHMP
|
8.7 | IC50 | 7 | Yes | |
LYGIRBLDUCXHDY
|
8.7 | IC50 | 4 | Yes | |
RPWIXTPWMSUQKW
|
8.7 | IC50 | 4 | Yes | |
VMOSDDURWLNMNG
|
8.7 | IC50 | 8 | Yes | |
XOBSNYRLSVUYKY
|
8.7 | IC50 | 2 | — | |
XQTUJUSPSCMEOC
|
8.7 | IC50 | 4 | Yes | |
NPWNPFHGYNOBOO
|
8.7 | IC50 | 7 | Yes | |
BJIOETDXHXZDRQ
|
8.7 | IC50 | 2 | — | |
XIQNNSMTTLQUTR
|
8.7 | IC50 | 6 | Yes | |
BBCCMNOZBPHYAJ
|
8.7 | IC50 | 3 | Yes | |
BIGQJQKSDHOEOM
|
8.7 | IC50 | 3 | Yes | |
FYNYGUYHKZWCAU
|
8.7 | IC50 | 4 | Yes | |
KAWCOVYOZMDLKQ
|
8.7 | IC50 | 4 | Yes | |
MTSOZTJGECJILJ
|
8.7 | IC50 | 6 | Yes | |
MXMCYIBSFFNNTF
|
8.7 | IC50 | 3 | Yes | |
NILIMKWDWHKQOZ
|
8.7 | IC50 | 7 | Yes | |
DYUKSKSACQYNBM
|
8.6 | IC50 | 3 | Yes | |
OKHKINWJYOOKOF
|
8.6 | IC50 | 3 | — | |
RNHOXGSFKJUDNY
|
8.6 | IC50 | 2 | Yes | |
SFHMNFHDIRPFKM
|
8.6 | IC50 | 7 | Yes | |
WLWNRAWQDZRXMB
|
8.6 | Ki | 6 | Yes | |
YLRFPZVTHHHQAF
|
8.6 | IC50 | 4 | Yes | |
XFILPEOLDIKJHX
|
8.6 | IC50 | 12 | Yes | |
GQVOKPKZCNLEIK
|
8.6 | IC50 | 3 | Yes | |
IHSDOJRAORURAS
|
8.6 | IC50 | 5 | Yes | |
ZHCXOELPVFPGHI
|
8.6 | IC50 | 4 | Yes | |
KVLYVSHQXNTARE
|
8.6 | IC50 | 4 | Yes | |
SQYRXZTYDRVAMZ
|
8.5 | Ki | 5 | Yes | |
AXBBWELSCMNUPM
|
8.5 | IC50 | 3 | — | |
BVQJLICESKJIJB
|
8.5 | IC50 | 5 | Yes | |
FUYGKZYSHSZHFI
|
8.5 | IC50 | 4 | Yes | |
GKURRRNPHZGWQU
|
8.5 | IC50 | 4 | Yes | |
HZNCNAGYECABJB
|
8.5 | IC50 | 2 | — | |
KQEHQRICYJKJLB
|
8.5 | IC50 | 6 | Yes | |
OAXXNDPRBWJXOJ
|
8.5 | IC50 | 4 | Yes | |
XAISFEMYYICOMZ
|
8.5 | IC50 | 4 | Yes | |
XDSILIXRMZXTNX
|
8.5 | IC50 | 5 | Yes | |
DNFCKYUQJJTPGW
|
8.5 | IC50 | 2 | — |