Target Details
| UniProt AC | P78536 |
|---|---|
| Gene Symbol | ADAM17 |
| Protein Name | Disintegrin and metalloproteinase domain-containing protein 17 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF16698 (ADAM17_MPD) PF00200 (Disintegrin) PF13574 (Reprolysin_2) |
Summary
- Multi-target molecules 785
- Clinical molecules 566
- Avg pChEMBL 7.43
KEGG Pathways (6)
Associated Diseases (2)
Active Molecules (785)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QFAMXNMLWJDJPV
|
7.1 | IC50 | 5 | Yes | |
RRUNLAIBQVECGY
|
7.1 | IC50 | 5 | Yes | |
VVCQPDVATXLSSI
|
7.1 | IC50 | 5 | Yes | |
WVHOOIOSMOLBGZ
|
7.1 | IC50 | 4 | — | |
ZQORGANDVNQVJF
|
7.1 | IC50 | 6 | Yes | |
CLTINYAXRIROMY
|
7.1 | IC50 | 5 | Yes | |
FTFANCIOHXJKDG
|
7.1 | IC50 | 4 | Yes | |
NWEMVUGYMZFTLT
|
7.1 | IC50 | 2 | — | |
OCBYWAVDKLDIDI
|
7.1 | IC50 | 5 | Yes | |
SSQXFNKOLMHXPO
|
7.1 | IC50 | 6 | Yes | |
KQYGUXCNMQFLRN
|
7.1 | IC50 | 5 | Yes | |
MWMRJYLEVAWDDL
|
7.1 | IC50 | 7 | Yes | |
IGKZHEJCICMYIH
|
7.1 | IC50 | 3 | Yes | |
JIYWMQDJGOAJMD
|
7.1 | IC50 | 6 | Yes | |
KJGJYHSHMUFLOA
|
7.0 | Ki | 5 | Yes | |
KRJQQXQOPZJOSC
|
7.0 | IC50 | 5 | Yes | |
UCKDGXYIQSPPDL
|
7.0 | IC50 | 5 | Yes | |
PCAPSCAFNCUGDE
|
7.0 | Ki | 6 | Yes | |
XWQYRXPGPDOWAJ
|
7.0 | IC50 | 5 | Yes | |
DIIAIQCOHXBJHI
|
7.0 | IC50 | 6 | Yes | |
FEFNNGHDRQMMNY
|
7.0 | IC50 | 2 | — | |
GIGQELYOVAVUIF
|
7.0 | IC50 | 4 | Yes | |
PLYLMXDSDZFWLJ
|
7.0 | IC50 | 6 | Yes | |
SEFCVQRMTNTWJO
|
7.0 | IC50 | 6 | Yes | |
BMHWXBBJSOMNRF
|
7.0 | IC50 | 3 | Yes | |
ZRQWUQCXSKEXGA
|
7.0 | Ki | 6 | — | |
OOCSYABQMHKMLM
|
7.0 | IC50 | 6 | Yes | |
HIBWRSXXRMHOLM
|
7.0 | IC50 | 2 | Yes | |
ILUVAAMGYFXXGD
|
7.0 | IC50 | 2 | Yes | |
YGTYRNSBOZPWFY
|
7.0 | IC50 | 3 | — | |
ZMVFZGHWXXXQJL
|
7.0 | IC50 | 6 | Yes | |
JDBUKSMCZPXYJU
|
7.0 | IC50 | 4 | — | |
KSLUOGMHCJCRLQ
|
7.0 | IC50 | 6 | Yes | |
JUDXBTMVZVWJNP
|
7.0 | IC50 | 2 | Yes | |
WOGNSQDLIXXYFU
|
7.0 | IC50 | 3 | Yes | |
XXZNXULRAJJTRV
|
7.0 | IC50 | 5 | Yes | |
YAYGKNVDBLFWFW
|
7.0 | IC50 | 6 | Yes | |
HKAXLEJIOVCYCD
|
7.0 | IC50 | 5 | Yes | |
NPFGSGCFKYSLPI
|
6.9 | IC50 | 6 | Yes | |
CKZHFOKQZRZCPF
|
6.9 | IC50 | 9 | Yes | |
CXIDTYUJLXWEAY
|
6.9 | IC50 | 2 | — | |
DFRHCKHXGKQVLI
|
6.9 | IC50 | 3 | Yes | |
JRKVJTDYMGJJAK
|
6.9 | IC50 | 6 | Yes | |
LDMWZYZAAZFUTC
|
6.9 | IC50 | 2 | — | |
TZNUGSCRBFBAFR
|
6.9 | Ki | 7 | Yes | |
CSVWGAZPMRHMHB
|
6.9 | IC50 | 5 | Yes | |
DCZIFTAWIUHEEC
|
6.9 | IC50 | 4 | Yes | |
GKDAXRUOVHMLSA
|
6.9 | IC50 | 6 | Yes | |
MAVDNGWEBZTACC
|
6.9 | IC50 | 9 | Yes | |
RAOAFDPXSFVLJD
|
6.9 | IC50 | 6 | Yes |