Target Details
| UniProt AC | P78536 |
|---|---|
| Gene Symbol | ADAM17 |
| Protein Name | Disintegrin and metalloproteinase domain-containing protein 17 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF16698 (ADAM17_MPD) PF00200 (Disintegrin) PF13574 (Reprolysin_2) |
Summary
- Multi-target molecules 785
- Clinical molecules 566
- Avg pChEMBL 7.43
KEGG Pathways (6)
Associated Diseases (2)
Active Molecules (785)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XMQNILGYVCROEB
|
7.1 | IC50 | 4 | Yes | |
YJZSNVXLDDRADS
|
7.1 | IC50 | 5 | Yes | |
YMQWZRPLMNNHEU
|
7.1 | IC50 | 6 | Yes | |
GTOFARSZXYDPTC
|
7.1 | IC50 | 5 | Yes | |
JVVFIHLIADCISB
|
7.1 | IC50 | 5 | Yes | |
PIHNCDLSZQOOPU
|
7.1 | Ki | 6 | Yes | |
BUUZULJJQMPZJK
|
7.1 | IC50 | 2 | — | |
CDVQKDXLTNVCDJ
|
7.1 | IC50 | 3 | — | |
CGAHNRKQXVGYMJ
|
7.1 | IC50 | 2 | — | |
CRJZQBWHTWJUPJ
|
7.1 | IC50 | 3 | — | |
DLWUUXWPNZKTFO
|
7.1 | IC50 | 3 | — | |
DVNZZKYEMTZGSP
|
7.1 | IC50 | 2 | — | |
FUVOMTJFSKUMQI
|
7.1 | IC50 | 3 | — | |
GSBJFDQGAVFCLJ
|
7.1 | IC50 | 3 | — | |
HPZRYZXQQVTWJN
|
7.1 | IC50 | 3 | — | |
IUOVINQVOHJYDU
|
7.1 | IC50 | 3 | — | |
JQSMTMOYUVJFIL
|
7.1 | IC50 | 2 | — | |
JSXIGTHUEBZKJY
|
7.1 | IC50 | 3 | — | |
LBEBGRPTXSMXMO
|
7.1 | IC50 | 3 | — | |
LPPROAMFDKZVIO
|
7.1 | IC50 | 2 | — | |
LRTSAWNNQKOXFU
|
7.1 | IC50 | 3 | — | |
LVIZNCUABWKXTG
|
7.1 | IC50 | 3 | — | |
MJMKBSLUNYUWCO
|
7.1 | IC50 | 3 | — | |
OTDAXJIWZBAIMD
|
7.1 | IC50 | 2 | — | |
PBIIXIBOBRDKAQ
|
7.1 | IC50 | 2 | — | |
PTZGCAFYBLXVGN
|
7.1 | IC50 | 3 | — | |
QFSLYLOLLOXSPR
|
7.1 | IC50 | 3 | — | |
QYERBIWZJAGVEU
|
7.1 | IC50 | 2 | — | |
RSYLDWPLCNLYJZ
|
7.1 | IC50 | 2 | — | |
SVLANDCYAZJNPV
|
7.1 | IC50 | 3 | — | |
SXKFYZOPGBFKLL
|
7.1 | IC50 | 2 | — | |
TXIMSNHHNJBLTN
|
7.1 | IC50 | 3 | Yes | |
URIKLEJPYMMEBH
|
7.1 | IC50 | 3 | — | |
VHLPSSCRYKMXMZ
|
7.1 | IC50 | 2 | — | |
WBCKZZUDBNRQQS
|
7.1 | IC50 | 2 | — | |
WIVGLBVPOCFAER
|
7.1 | IC50 | 2 | — | |
WIXQHARDFJRBSX
|
7.1 | IC50 | 2 | — | |
XPUGDXRRGXHBML
|
7.1 | IC50 | 3 | — | |
XRIFBRFEZLXEFP
|
7.1 | Ki | 5 | — | |
XXQLCMDLJMBMLB
|
7.1 | IC50 | 3 | — | |
YIJGRACDTOYEDJ
|
7.1 | IC50 | 2 | — | |
AENHIDVKFOYIJJ
|
7.1 | IC50 | 4 | Yes | |
QJCXYCVUFZIPQG
|
7.1 | Ki | 3 | — | |
RCOBSDNFRJAUBV
|
7.1 | IC50 | 4 | Yes | |
SBPPAFQZTZUQSW
|
7.1 | IC50 | 4 | Yes | |
VSZRGCMKCYLOIV
|
7.1 | IC50 | 4 | Yes | |
JUSNXCIZGYMOPC
|
7.1 | IC50 | 3 | Yes | |
LGVIBWRSRHZDQG
|
7.1 | IC50 | 6 | Yes | |
CBMKHOZXSARYNG
|
7.1 | IC50 | 6 | Yes | |
KZZUIFPIPUBRFP
|
7.1 | Ki | 2 | — |