Target Details
| UniProt AC | P78536 |
|---|---|
| Gene Symbol | ADAM17 |
| Protein Name | Disintegrin and metalloproteinase domain-containing protein 17 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF16698 (ADAM17_MPD) PF00200 (Disintegrin) PF13574 (Reprolysin_2) |
Summary
- Multi-target molecules 785
- Clinical molecules 566
- Avg pChEMBL 7.43
KEGG Pathways (6)
Associated Diseases (2)
Active Molecules (785)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AUWCRYUPRHMNCJ
|
10.2 | Ki | 2 | — | |
NSKDLLYTWJVRPJ
|
10.0 | Ki | 2 | — | |
SIICAQVADMFEDB
|
9.8 | IC50 | 8 | Yes | |
GKHRDWHFKKUYAX
|
9.7 | IC50 | 8 | Yes | |
QVNZBDLTUKCPGJ
|
9.7 | IC50 | 10 | — | |
DJQJEICJRBFEOV
|
9.6 | IC50 | 4 | Yes | |
SISZTYKGUNKWOD
|
9.5 | Ki | 2 | — | |
OBJBBLBMOOBABD
|
9.5 | IC50 | 8 | Yes | |
CNUCYIDHDPTDOD
|
9.4 | Ki | 5 | Yes | |
CIMXKGKYBNXAKQ
|
9.4 | Ki | 2 | — | |
ATUIUMZYBUFUGD
|
9.3 | Ki | 2 | — | |
CSQCYVHPHVXICP
|
9.3 | IC50 | 4 | Yes | |
WSWMIGCNSWBCNT
|
9.3 | Ki | 6 | Yes | |
CFNLVCZTXBNJGL
|
9.2 | Ki | 4 | Yes | |
FYZPCUXRTDXRBF
|
9.2 | Ki | 6 | Yes | |
PYTXPVHJIDYQEO
|
9.2 | Ki | 2 | — | |
RMMUGCXFUHIPQO
|
9.2 | IC50 | 2 | — | |
QOWBVKQSFCSJAK
|
9.2 | Ki | 5 | — | |
VOXBFNGVFFRNIE
|
9.1 | IC50 | 2 | — | |
YAWCEEHWRJZVNM
|
9.1 | IC50 | 2 | — | |
IIBLNMYMPDUKOQ
|
9.1 | Ki | 3 | Yes | |
NXWFYCXTAINJMY
|
9.1 | Ki | 6 | Yes | |
DDFFKEPNXVTRCY
|
9.0 | IC50 | 4 | Yes | |
DUPLEMOAJXTDKP
|
9.0 | IC50 | 4 | Yes | |
GGDBCZZATDMWMQ
|
9.0 | IC50 | 4 | Yes | |
HNEDFPGSHTUVKZ
|
9.0 | IC50 | 7 | Yes | |
JTCBZWXCQOLSNN
|
9.0 | IC50 | 2 | — | |
QXLMMZHXXOWCDY
|
9.0 | IC50 | 4 | Yes | |
VNIVLVJMMLQGNQ
|
9.0 | IC50 | 4 | Yes | |
VOYWXVODQDUTJD
|
9.0 | IC50 | 3 | Yes | |
YDMIPBHQKFOFQW
|
9.0 | IC50 | 7 | Yes | |
XWVXWDVYQZEQBA
|
9.0 | IC50 | 4 | Yes | |
HTEPICDCVMJOSJ
|
8.9 | IC50 | 3 | Yes | |
CXZHJWRHSTZNHB
|
8.9 | IC50 | 4 | Yes | |
RCCBHNFHHCGOQM
|
8.9 | IC50 | 4 | Yes | |
UFEAOVWYWYBIFX
|
8.9 | IC50 | 4 | Yes | |
VGMJDHAFWAQDDY
|
8.9 | IC50 | 4 | Yes | |
WHUGMPJJQOVPAC
|
8.9 | IC50 | 4 | Yes | |
IYSKDTAJMOMROJ
|
8.8 | IC50 | 4 | Yes | |
KRGBAILWDVNOCW
|
8.8 | IC50 | 6 | Yes | |
LOOGWNWWNBNMRC
|
8.8 | IC50 | 4 | Yes | |
RBTIHKNARDNLNU
|
8.8 | IC50 | 5 | Yes | |
CEVLUPQNDFOYSI
|
8.8 | IC50 | 5 | Yes | |
IASRCCATUJITDX
|
8.8 | IC50 | 4 | Yes | |
WUVJCBZUUQXYIT
|
8.8 | IC50 | 4 | Yes | |
HQGORWGMKQFFGB
|
8.8 | IC50 | 3 | Yes | |
LQZDEWIIFWHTLX
|
8.8 | Ki | 6 | Yes | |
NOBVVTLEQRHRBY
|
8.8 | IC50 | 3 | Yes | |
RXFCFGLSOUOCEA
|
8.8 | IC50 | 4 | Yes | |
IDHBZDJZPPEMGC
|
8.8 | IC50 | 4 | Yes |