Target Details
| UniProt AC | P78527 |
|---|---|
| Gene Symbol | PRKDC |
| Protein Name | DNA-dependent protein kinase catalytic subunit |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF20500 (DNA-PKcs_N) PF20502 (DNAPKcs_CC1-2) PF08163 (DNAPKcs_CC3) PF19704 (DNAPKcs_CC5) PF02259 (FAT) PF02260 (FATC) PF00454 (PI3_PI4_kinase) |
Summary
- Multi-target molecules 312
- Clinical molecules 140
- Avg pChEMBL 7.22
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (312)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LQUXOZIJMPWQAA
|
6.0 | IC50 | 2 | Yes | |
YZDHQXUAXYNXQS
|
6.0 | IC50 | 2 | — | |
ZNAZTNSMMJFJLP
|
6.0 | IC50 | 3 | Yes | |
FASPJDRKOSUHHS
|
6.0 | IC50 | 10 | Yes | |
IWGLXKVBQSBQMC
|
6.0 | IC50 | 13 | Yes | |
LXWKVQVKYRGEKE
|
6.0 | IC50 | 6 | Yes | |
JSXBAKOSLFZFQZ
|
6.0 | IC50 | 4 | Yes | |
HMKCVXALDWCZFL
|
6.0 | IC50 | 2 | Yes | |
ZRSCVKQQFCOUGY
|
6.0 | IC50 | 3 | — | |
JROFGZPOBKIAEW
|
6.0 | IC50 | 10 | — | |
MFZAHAAVYSHLCP
|
6.0 | IC50 | 7 | — | |
QILFSWGIDUVYFO
|
6.0 | IC50 | 2 | — |