Target Details
| UniProt AC | P78527 |
|---|---|
| Gene Symbol | PRKDC |
| Protein Name | DNA-dependent protein kinase catalytic subunit |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF20500 (DNA-PKcs_N) PF20502 (DNAPKcs_CC1-2) PF08163 (DNAPKcs_CC3) PF19704 (DNAPKcs_CC5) PF02259 (FAT) PF02260 (FATC) PF00454 (PI3_PI4_kinase) |
Summary
- Multi-target molecules 312
- Clinical molecules 140
- Avg pChEMBL 7.22
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (312)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ULTBPCMFBBBUND
|
6.4 | IC50 | 3 | — | |
WXCKXLFOEBUZDO
|
6.4 | IC50 | 6 | Yes | |
ILKDWZKZLIHMFM
|
6.4 | IC50 | 8 | — | |
IRTDIKMSKMREGO
|
6.4 | IC50 | 6 | — | |
MZBVEJCJSWMSLU
|
6.4 | IC50 | 2 | — | |
PFRDPPRTLFHGLR
|
6.4 | IC50 | 10 | Yes | |
CJFWNLXLAAHQJY
|
6.4 | IC50 | 11 | Yes | |
BZYKWEQWEPHEQZ
|
6.3 | IC50 | 10 | Yes | |
ULLIAFSPUSWCIL
|
6.3 | IC50 | 10 | Yes | |
ZTWYTYUOHYGWSG
|
6.3 | IC50 | 9 | Yes | |
LMVAHLFZGWUGNF
|
6.3 | IC50 | 8 | Yes | |
ANYPGTJVYHIIEM
|
6.3 | IC50 | 2 | — | |
KLQFQJDEPBUNAK
|
6.3 | IC50 | 6 | Yes | |
RDALZZCKQFLGJP
|
6.3 | IC50 | 2 | — | |
ZTQOHJNXDAUMOA
|
6.3 | IC50 | 13 | Yes | |
FHNLPTRXVQOXQO
|
6.3 | IC50 | 11 | Yes | |
LNWUSIFVARIMOH
|
6.3 | IC50 | 6 | Yes | |
GGBQGMRDBYCCLW
|
6.2 | IC50 | 4 | Yes | |
NZELPIPZPVLYLT
|
6.2 | IC50 | 3 | Yes | |
QPZURRPXZSPBJE
|
6.2 | IC50 | 9 | Yes | |
YLDAIYDYJXZDGW
|
6.2 | IC50 | 15 | — | |
FHNLPTRXVQOXQO
|
6.2 | IC50 | 7 | Yes | |
KLQFKOVDEHUNHU
|
6.2 | IC50 | 10 | Yes | |
RNMJNHVCCXRKJE
|
6.2 | IC50 | 2 | — | |
CIRFQCDQKJVIFC
|
6.2 | IC50 | 7 | Yes | |
DISRGUXSEDBDDN
|
6.2 | IC50 | 2 | — | |
JDOVRLNHIYWZKZ
|
6.2 | IC50 | 7 | Yes | |
LKHMVKNMSWRHJH
|
6.2 | IC50 | 7 | — | |
ORVLOIUKTHUQPU
|
6.2 | IC50 | 4 | Yes | |
LBRPXBJBDBBMNZ
|
6.2 | IC50 | 6 | Yes | |
ZCBWPTBPKMKOLE
|
6.2 | IC50 | 5 | — | |
ZNRCBKKFSNMJEK
|
6.2 | IC50 | 2 | — | |
ORVLOIUKTHUQPU
|
6.2 | IC50 | 5 | Yes | |
WDMOOFMBMGLZGY
|
6.2 | IC50 | 5 | Yes | |
MPUATQFVQOUAJF
|
6.1 | IC50 | 6 | Yes | |
YFHBYQHMVTVHDA
|
6.1 | IC50 | 3 | — | |
CBHYTLBXAZHCMA
|
6.1 | IC50 | 3 | — | |
CBHYTLBXAZHCMA
|
6.1 | IC50 | 4 | — | |
CDJSZJDGHKEHCW
|
6.1 | IC50 | 5 | Yes | |
ISWAJEMQAQNLMY
|
6.1 | IC50 | 2 | — | |
MJALZBJFTIQSSR
|
6.1 | IC50 | 12 | Yes | |
BRGUQOISTYVOBM
|
6.1 | Ki | 3 | — | |
GTXKSDZLEOURPP
|
6.1 | IC50 | 4 | Yes | |
FXCRGRHHHOSJRE
|
6.1 | IC50 | 5 | Yes | |
MNJNKKYCZKBVRY
|
6.1 | IC50 | 10 | Yes | |
AMERZUAKIAGPBA
|
6.1 | IC50 | 7 | Yes | |
QIUHOMNRLMPPFS
|
6.1 | IC50 | 2 | — | |
ILBRKJBKDGCSCB
|
6.1 | IC50 | 2 | — | |
MWKYMZXCGYXLPL
|
6.1 | IC50 | 5 | — | |
OUQOXXMJLDQZQC
|
6.1 | IC50 | 6 | Yes |