Target Details
| UniProt AC | P78527 |
|---|---|
| Gene Symbol | PRKDC |
| Protein Name | DNA-dependent protein kinase catalytic subunit |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF20500 (DNA-PKcs_N) PF20502 (DNAPKcs_CC1-2) PF08163 (DNAPKcs_CC3) PF19704 (DNAPKcs_CC5) PF02259 (FAT) PF02260 (FATC) PF00454 (PI3_PI4_kinase) |
Summary
- Multi-target molecules 312
- Clinical molecules 140
- Avg pChEMBL 7.22
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (312)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PCPZDHWQPMHSIG
|
6.7 | IC50 | 2 | — | |
BTIKYUUNPGWLNG
|
6.7 | IC50 | 12 | Yes | |
CMUZPNXYCOKJJJ
|
6.7 | IC50 | 7 | Yes | |
FVPBLAKABVRLRX
|
6.7 | IC50 | 9 | Yes | |
KUUKOPMICNKRGE
|
6.7 | IC50 | 12 | Yes | |
QOYOSSAKTDDRJV
|
6.7 | IC50 | 11 | Yes | |
IVPZQVJSLCFTTO
|
6.7 | IC50 | 10 | Yes | |
JSGRAJRLMWHOTJ
|
6.7 | IC50 | 7 | Yes | |
PBWTXSSLHGGJBR
|
6.7 | IC50 | 2 | Yes | |
KKTZALUTXUZPSN
|
6.6 | IC50 | 2 | Yes | |
AAHKGRWRYBCWDL
|
6.6 | IC50 | 11 | Yes | |
VPSLBUMYCILBRD
|
6.6 | IC50 | 8 | Yes | |
LQIVXZFCXIBJSU
|
6.6 | IC50 | 10 | Yes | |
RXNGGTYNZUEFOM
|
6.6 | IC50 | 8 | Yes | |
ALVMITILHVYXEU
|
6.6 | IC50 | 3 | — | |
AXQKJTHCYRYSLF
|
6.6 | IC50 | 3 | Yes | |
DREWJJJKWOJZQM
|
6.6 | Ki | 2 | — | |
YRJGEWAWXXEJNX
|
6.6 | IC50 | 3 | Yes | |
MRZVUZUMBCEAGI
|
6.6 | IC50 | 12 | Yes | |
YWWWQQYKTOUASO
|
6.6 | IC50 | 3 | — | |
BVRDQVRQVGRNHG
|
6.5 | IC50 | 2 | Yes | |
RMKWCFQVLOKCHU
|
6.5 | IC50 | 2 | — | |
ROBUSLZBFPYNBA
|
6.5 | IC50 | 4 | — | |
CIZOSCVUGRBXEZ
|
6.5 | IC50 | 4 | — | |
JDRPVJJOYKLLFH
|
6.5 | IC50 | 2 | Yes | |
OWQIHYNKDOPWGC
|
6.5 | IC50 | 2 | — | |
ZCCPLJOKGAACRT
|
6.5 | Kd | 599 | — | |
AULCRCVNIWNUTH
|
6.5 | IC50 | 10 | Yes | |
CZQHHVNHHHRRDU
|
6.5 | IC50 | 12 | Yes | |
SQYGYXGOJYZQEI
|
6.5 | IC50 | 2 | — | |
UCEVYDVOUKTNMU
|
6.5 | IC50 | 2 | — | |
QYPSALIXKCRYNZ
|
6.5 | IC50 | 12 | Yes | |
HGALDAPNHYJZAJ
|
6.5 | IC50 | 11 | Yes | |
NRZFXYCLDSAYDI
|
6.5 | IC50 | 7 | Yes | |
PSICWGWNIOOULV
|
6.5 | IC50 | 3 | — | |
BHXYWMKHQZDQLR
|
6.5 | IC50 | 2 | — | |
DUPSNQFPAJUAKA
|
6.5 | IC50 | 9 | Yes | |
YBXRSCXGRPSTMW
|
6.5 | IC50 | 6 | — | |
KUMLEJXITHSWSP
|
6.5 | IC50 | 9 | Yes | |
WGYPOAXANMFHMT
|
6.5 | IC50 | 10 | Yes | |
YKDLGDBIORZVLP
|
6.5 | IC50 | 10 | Yes | |
SPUWUOGLPPVXCW
|
6.5 | IC50 | 15 | Yes | |
KFBBXKBRSICFJT
|
6.5 | IC50 | 8 | Yes | |
SVNJBEMPMKWDCO
|
6.5 | IC50 | 3 | — | |
SSVLAVRFVKSIND
|
6.4 | IC50 | 4 | Yes | |
IBSCAHNKEHRFKF
|
6.4 | IC50 | 4 | Yes | |
XHNKFGYYGPLYPT
|
6.4 | IC50 | 3 | — | |
XNODQMMIMXSTMX
|
6.4 | IC50 | 12 | Yes | |
HVUAYFFHDRNLOX
|
6.4 | IC50 | 11 | Yes | |
MFAQYJIYDMLAIM
|
6.4 | IC50 | 130 | Yes |