Target Details
| UniProt AC | P78527 |
|---|---|
| Gene Symbol | PRKDC |
| Protein Name | DNA-dependent protein kinase catalytic subunit |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF20500 (DNA-PKcs_N) PF20502 (DNAPKcs_CC1-2) PF08163 (DNAPKcs_CC3) PF19704 (DNAPKcs_CC5) PF02259 (FAT) PF02260 (FATC) PF00454 (PI3_PI4_kinase) |
Summary
- Multi-target molecules 312
- Clinical molecules 140
- Avg pChEMBL 7.22
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (312)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GDWZFRMYHRRYAR
|
7.0 | IC50 | 2 | — | |
OVFIHIWNXSZYOH
|
7.0 | Ki | 3 | — | |
PQRFMBAACAPZPP
|
7.0 | IC50 | 12 | Yes | |
PSYXHVWBVRRNHD
|
7.0 | IC50 | 11 | Yes | |
UQTJNUFTALPBOP
|
7.0 | IC50 | 2 | — | |
UQTJNUFTALPBOP
|
7.0 | IC50 | 2 | — | |
IJEDYDGSAXSVPY
|
6.9 | IC50 | 4 | — | |
PGXQNHGXDFCMOJ
|
6.9 | IC50 | 10 | Yes | |
QDLHCMPXEPAAMD
|
6.9 | Ki | 13 | Yes | |
VRCXIJAYLCUSHC
|
6.9 | IC50 | 3 | — | |
VRCXIJAYLCUSHC
|
6.9 | IC50 | 3 | — | |
HYSFHTXNKQSESE
|
6.9 | IC50 | 2 | — | |
KAHMZYOZNYFPKN
|
6.9 | IC50 | 3 | — | |
AGEIBLLCZVGHLI
|
6.9 | IC50 | 9 | Yes | |
AOTRIQLYUAFVSC
|
6.8 | IC50 | 5 | — | |
MSJODEOZODDVGW
|
6.8 | IC50 | 10 | — | |
UFZMEAYSFGBIBJ
|
6.8 | IC50 | 4 | — | |
YJFMDYHDHYLLEX
|
6.8 | IC50 | 2 | — | |
DAXOOIRHYYCDDH
|
6.8 | IC50 | 10 | Yes | |
DINPOPQNCDTVPQ
|
6.8 | IC50 | 10 | Yes | |
HBTYJGOOZWMVOI
|
6.8 | IC50 | 2 | — | |
HJSSPYJVWLTYHG
|
6.8 | IC50 | 8 | — | |
LQRSFPTVTRTRMP
|
6.8 | IC50 | 3 | — | |
MRZVUZUMBCEAGI
|
6.8 | IC50 | 11 | Yes | |
RUQMPILTACLXOK
|
6.8 | IC50 | 6 | Yes | |
SYVQAQHCFMTBNA
|
6.8 | IC50 | 3 | — | |
WRNCIFYXNUAFIH
|
6.8 | IC50 | 2 | — | |
RHFWTFDTRBFIHU
|
6.8 | IC50 | 13 | Yes | |
FNNGURVIOIZXRF
|
6.8 | Ki | 3 | — | |
HWVZGRVXWDKHFX
|
6.8 | IC50 | 2 | — | |
NGMBEJKZRRVAGQ
|
6.8 | IC50 | 2 | — | |
YJNVZAXZUDOAAI
|
6.8 | IC50 | 10 | Yes | |
GRWJFKQBVQNWQW
|
6.8 | IC50 | 10 | Yes | |
NVHKWMBHTXQWRP
|
6.8 | IC50 | 9 | Yes | |
TXZDVQGUIJKUMP
|
6.8 | IC50 | 6 | Yes | |
FZLLSBHPQYLGLH
|
6.7 | Ki | 3 | — | |
JFJRIADKVAOEDG
|
6.7 | IC50 | 4 | Yes | |
JNRPKMKRMUTLDI
|
6.7 | IC50 | 2 | — | |
UAZUSSYGOQZXRK
|
6.7 | IC50 | 2 | — | |
XRKYMMUGXMWDAO
|
6.7 | IC50 | 5 | Yes | |
CHPHDLQQSCKHOK
|
6.7 | IC50 | 8 | Yes | |
DUQGHTXMYYQABR
|
6.7 | IC50 | 4 | Yes | |
FAWGCSGOLCHXBH
|
6.7 | IC50 | 11 | Yes | |
MWYBBCLGEHZSCP
|
6.7 | IC50 | 11 | Yes | |
RFWCIJWQGHFULK
|
6.7 | IC50 | 2 | Yes | |
GZMCDKYNELBFSQ
|
6.7 | IC50 | 2 | — | |
XVTLRUAQTJKQLQ
|
6.7 | IC50 | 9 | Yes | |
CBWWAMHIIZVQTP
|
6.7 | IC50 | 6 | — | |
FPWSKINOJYCEJK
|
6.7 | IC50 | 3 | — | |
CORFNGYLXZFTMD
|
6.7 | IC50 | 3 | — |