Target Details
| UniProt AC | P78527 |
|---|---|
| Gene Symbol | PRKDC |
| Protein Name | DNA-dependent protein kinase catalytic subunit |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF20500 (DNA-PKcs_N) PF20502 (DNAPKcs_CC1-2) PF08163 (DNAPKcs_CC3) PF19704 (DNAPKcs_CC5) PF02259 (FAT) PF02260 (FATC) PF00454 (PI3_PI4_kinase) |
Summary
- Multi-target molecules 312
- Clinical molecules 140
- Avg pChEMBL 7.22
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (312)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UGUJFPIEAZXKAK
|
7.4 | IC50 | 5 | Yes | |
VBUMOGXFBGYXDV
|
7.4 | IC50 | 11 | Yes | |
QKBGNVCABCTNCY
|
7.4 | IC50 | 3 | — | |
MQXVMMLHAWPDPI
|
7.4 | IC50 | 4 | — | |
VEORWCZDRQSGJH
|
7.4 | IC50 | 10 | Yes | |
WIYTYGLDKRTSHX
|
7.4 | IC50 | 2 | — | |
BSYIKIPUNRLIEZ
|
7.4 | IC50 | 4 | — | |
JPOWZUHXAXNZNE
|
7.3 | IC50 | 4 | — | |
HFBMCRRHMRLGSA
|
7.3 | IC50 | 7 | Yes | |
DBZCDBKTCUKQPQ
|
7.3 | IC50 | 8 | Yes | |
ITOYZJGFTNTKKR
|
7.3 | IC50 | 11 | Yes | |
DYEJYFAQYRMVFS
|
7.3 | IC50 | 9 | Yes | |
NIIYHUNRXQLMBG
|
7.3 | IC50 | 6 | — | |
IYVUNPAVFASLSV
|
7.3 | IC50 | 6 | Yes | |
MONJJHLZSIEMDE
|
7.3 | IC50 | 6 | Yes | |
DTUMIKLOEHJGJT
|
7.3 | IC50 | 3 | Yes | |
ZSAJPWOGVMFXHN
|
7.3 | IC50 | 10 | Yes | |
JPOWZUHXAXNZNE
|
7.3 | IC50 | 2 | — | |
PEKHSWOOLJTLAP
|
7.3 | IC50 | 3 | — | |
PQQPUILDPHGQHI
|
7.3 | IC50 | 2 | — | |
XQSYLEMSNXLJBZ
|
7.3 | IC50 | 2 | — | |
ZITCKJQNZLGXNI
|
7.3 | IC50 | 2 | — | |
YZGKSARXIQYKAW
|
7.2 | IC50 | 2 | — | |
NVRXTLZYXZNATH
|
7.2 | IC50 | 47 | Yes | |
UXLMBWJITRRKHJ
|
7.2 | IC50 | 2 | — | |
KIZCESWOQMCQAK
|
7.2 | IC50 | 2 | — | |
JFVNFXCESCXMBC
|
7.2 | IC50 | 8 | — | |
NVHKWMBHTXQWRP
|
7.2 | IC50 | 9 | Yes | |
KTTGLAHMSDMRLJ
|
7.2 | IC50 | 12 | Yes | |
LQCFRUUPBAMHIY
|
7.2 | IC50 | 6 | — | |
OKNNPZZFEHDVHC
|
7.1 | IC50 | 2 | — | |
ATKHYZXUMVNCIO
|
7.1 | IC50 | 4 | — | |
SCELLOWTHJGVIC
|
7.1 | IC50 | 4 | — | |
UBJGLXSFXKIIFY
|
7.1 | IC50 | 12 | Yes | |
ULPBTMCLMXCXEB
|
7.1 | IC50 | 11 | Yes | |
MRCFTWAYZAHAFA
|
7.1 | IC50 | 12 | Yes | |
QFUHCUNJMQVKME
|
7.1 | IC50 | 8 | Yes | |
UAFBQETUXPWPCQ
|
7.1 | IC50 | 2 | — | |
HRZBUHAVTBTHTM
|
7.1 | IC50 | 3 | — | |
XOKCNIACFBBJGV
|
7.1 | IC50 | 11 | Yes | |
CJMMCIXRPVLDBH
|
7.1 | IC50 | 12 | Yes | |
UVFCDQJUKYMBAZ
|
7.1 | IC50 | 10 | Yes | |
PNEGWAQERPTPDN
|
7.0 | IC50 | 12 | Yes | |
DPKWEPQBVKHUQT
|
7.0 | IC50 | 4 | — | |
JCMWWPAJCOQLAF
|
7.0 | IC50 | 11 | Yes | |
ZNUODSNRAGKDRE
|
7.0 | IC50 | 6 | Yes | |
SNHKARUQVBJTQS
|
7.0 | IC50 | 11 | Yes | |
MBPKPSDAPFPECJ
|
7.0 | IC50 | 12 | Yes | |
CEUPOOINALBZRR
|
7.0 | IC50 | 6 | — | |
FRKWMLCUONAHJH
|
7.0 | IC50 | 13 | Yes |