Target Details
| UniProt AC | P78527 |
|---|---|
| Gene Symbol | PRKDC |
| Protein Name | DNA-dependent protein kinase catalytic subunit |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF20500 (DNA-PKcs_N) PF20502 (DNAPKcs_CC1-2) PF08163 (DNAPKcs_CC3) PF19704 (DNAPKcs_CC5) PF02259 (FAT) PF02260 (FATC) PF00454 (PI3_PI4_kinase) |
Summary
- Multi-target molecules 312
- Clinical molecules 140
- Avg pChEMBL 7.22
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (312)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OHERNBRGXOVCSR
|
8.3 | IC50 | 4 | — | |
QXILYQTXHFZFST
|
8.3 | IC50 | 3 | — | |
TXGXVGZVOFHZBI
|
8.3 | IC50 | 4 | — | |
UUAWGVGBYJWRND
|
8.3 | IC50 | 2 | — | |
VFJHEBMKBXLCDG
|
8.3 | IC50 | 2 | — | |
VTNYVWSVPWEXFE
|
8.3 | IC50 | 4 | — | |
XMSRADCMDDJZDM
|
8.3 | IC50 | 3 | — | |
XNQLBCLHQMLKIC
|
8.3 | IC50 | 3 | — | |
YVQDIBOPRZOYGI
|
8.3 | IC50 | 3 | — | |
ZQXXURIZTYXFML
|
8.3 | IC50 | 2 | — | |
XYGUWWJXZYCPEF
|
8.2 | IC50 | 2 | — | |
GHUICRRPTSLMIY
|
8.2 | IC50 | 6 | Yes | |
GNEFGLFGNKFHAR
|
8.2 | Ki | 2 | — | |
GCKKBGHFJIZIAB
|
8.2 | Ki | 3 | — | |
JFZBEJKCLYCEPN
|
8.2 | IC50 | 2 | — | |
XXTQNUUFXVHHHD
|
8.2 | IC50 | 2 | — | |
NXVVYRYBOAFGHA
|
8.1 | IC50 | 2 | — | |
HHAPAAFKKUAWAI
|
8.1 | IC50 | 5 | — | |
SZJQPMPJULBZRG
|
8.1 | IC50 | 2 | — | |
GEZALMMCQYDFML
|
8.1 | IC50 | 15 | Yes | |
YUZWKYFHKYQPMO
|
8.1 | IC50 | 2 | — | |
BYTKNUOMWLJVNQ
|
8.1 | IC50 | 10 | — | |
DHYADLCEAXMYPS
|
8.1 | IC50 | 9 | Yes | |
QBPMDFDPUIVKQA
|
8.0 | IC50 | 11 | Yes | |
HXIMOOZRCPTJDQ
|
8.0 | IC50 | 5 | — | |
LHTOPXIXDAUXST
|
8.0 | IC50 | 3 | — | |
LPJIZDSOUGHTNB
|
8.0 | IC50 | 3 | — | |
YJZNDQMSXXSTQC
|
8.0 | IC50 | 2 | — | |
MFRGGAROFRXKRT
|
7.9 | IC50 | 10 | Yes | |
UDUPSRWUDACGIS
|
7.9 | IC50 | 13 | Yes | |
ZJAVHOMVDCMAMF
|
7.9 | IC50 | 9 | — | |
GMYLVKUGJMYTFB
|
7.9 | IC50 | 7 | — | |
TUVCWJQQGGETHL
|
7.8 | IC50 | 22 | — | |
ZGBQFYGLPMXTSZ
|
7.8 | IC50 | 7 | Yes | |
FUCGVOYZRSDCPC
|
7.8 | IC50 | 4 | — | |
ZBTLTVIYBHYEHL
|
7.8 | IC50 | 13 | Yes | |
ZLMVXCGWUJXFNP
|
7.8 | IC50 | 15 | Yes | |
HRRMXIICSWVXIS
|
7.7 | IC50 | 13 | Yes | |
QRJVSLZNMWIKRS
|
7.7 | IC50 | 7 | Yes | |
JAMULYFATHSZJM
|
7.7 | IC50 | 7 | Yes | |
SERJTVXHERVFCQ
|
7.6 | IC50 | 2 | — | |
DUIHHZKTCSNTGM
|
7.6 | IC50 | 2 | — | |
ISIOGRVXKGDUFP
|
7.6 | IC50 | 5 | — | |
PQEIMHBVHXTVNA
|
7.6 | IC50 | 5 | — | |
GCHBEJBYMQHZEM
|
7.6 | IC50 | 5 | — | |
COAQRADEUYYCDG
|
7.5 | IC50 | 12 | Yes | |
UOKGZPYGRJDACN
|
7.5 | IC50 | 7 | Yes | |
LVUGPVDXTSJQQD
|
7.5 | IC50 | 13 | Yes | |
COAQRADEUYYCDG
|
7.5 | IC50 | 12 | Yes | |
DPLMXAYKJZOTKO
|
7.4 | IC50 | 5 | — |