Target Details
| UniProt AC | P78527 |
|---|---|
| Gene Symbol | PRKDC |
| Protein Name | DNA-dependent protein kinase catalytic subunit |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF20500 (DNA-PKcs_N) PF20502 (DNAPKcs_CC1-2) PF08163 (DNAPKcs_CC3) PF19704 (DNAPKcs_CC5) PF02259 (FAT) PF02260 (FATC) PF00454 (PI3_PI4_kinase) |
Summary
- Multi-target molecules 312
- Clinical molecules 140
- Avg pChEMBL 7.22
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (312)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WLGXNSHVQAUMAT
|
10.2 | IC50 | 4 | — | |
WMVFYJNFGFTSCQ
|
10.0 | IC50 | 2 | — | |
LOQIJPHCNFJJTO
|
9.9 | IC50 | 2 | — | |
PCTWMWBDQSWVBE
|
9.8 | IC50 | 2 | — | |
WGZHCNCLATVGMN
|
9.8 | IC50 | 2 | — | |
XGWVDWGXBYRXIX
|
9.8 | IC50 | 2 | — | |
ATTXFDBPVDTNAP
|
9.7 | IC50 | 2 | — | |
JHYPYJLPMJWBRK
|
9.7 | IC50 | 2 | — | |
MUSBPXCQBAUPOW
|
9.7 | IC50 | 2 | — | |
SKLZRGKNDWBPBV
|
9.7 | IC50 | 2 | — | |
CGBJSGAELGCMKE
|
9.6 | IC50 | 11 | — | |
MOWXJLUYGFNTAL
|
9.4 | IC50 | 5 | — | |
FAPBUMXELNHUHE
|
9.4 | IC50 | 2 | — | |
GUXXEUUYCAYESJ
|
9.3 | IC50 | 11 | — | |
QVFCDPRQRUAFKS
|
9.3 | IC50 | 10 | Yes | |
BAIBLIJJASBKKL
|
9.2 | IC50 | 3 | — | |
JEKDMEAMHWNRLL
|
9.2 | IC50 | 4 | — | |
DFPIFDHNNWOIDD
|
9.1 | IC50 | 3 | — | |
MZQKKBHRPQCGSA
|
9.1 | IC50 | 5 | — | |
OICCEQGFJHNAPZ
|
9.1 | IC50 | 3 | — | |
UNETUVMFOUXHNZ
|
9.0 | IC50 | 2 | — | |
WEEIJHAKEWVFES
|
9.0 | IC50 | 2 | — | |
XISVSTPEXYIKJL
|
9.0 | IC50 | 5 | — | |
YDMGJNNVRFAERS
|
9.0 | IC50 | 2 | — | |
MGKLYPORYDLRLO
|
9.0 | IC50 | 4 | — | |
JOGKUKXHTYWRGZ
|
8.9 | IC50 | 28 | — | |
CRZTZRWPHCWXOK
|
8.7 | IC50 | 5 | — | |
OJFQDQYUIAHKRJ
|
8.7 | IC50 | 2 | — | |
RTARVPHTCQRSDW
|
8.6 | IC50 | 7 | Yes | |
GUFVTKTWKYLOQP
|
8.5 | IC50 | 7 | — | |
YGBMCLDVRUGXOV
|
8.5 | IC50 | 8 | Yes | |
MFVOIPKDSOFMQO
|
8.5 | IC50 | 3 | — | |
MFVOIPKDSOFMQO
|
8.5 | IC50 | 3 | — | |
YKIWXNATSYCOKT
|
8.5 | IC50 | 7 | Yes | |
PMBCEMXDAJTEQO
|
8.4 | IC50 | 2 | — | |
AATCBLYHOUOCTO
|
8.3 | IC50 | 4 | — | |
KGAAOKXUCALAPY
|
8.3 | IC50 | 8 | — | |
KZJLHYQNEJSYNN
|
8.3 | IC50 | 6 | — | |
YSOQBYOYIBXQGO
|
8.3 | IC50 | 6 | — | |
BSGBCKRSUJYENI
|
8.3 | IC50 | 2 | — | |
DFUFAVMVCOEDLG
|
8.3 | IC50 | 2 | — | |
FLODHIIWXLIRRR
|
8.3 | IC50 | 4 | — | |
FPHLASQTEAWKKW
|
8.3 | IC50 | 2 | — | |
GQUJOOVYNSNQLU
|
8.3 | IC50 | 3 | — | |
GYWPMKOUCJEYNO
|
8.3 | IC50 | 3 | — | |
IJDLDJGJYHPWSI
|
8.3 | IC50 | 3 | — | |
JVKKETWPNJSWSC
|
8.3 | IC50 | 2 | — | |
KASNAMAOPPOPNR
|
8.3 | IC50 | 2 | — | |
LCWHFJMGEPVAGK
|
8.3 | IC50 | 3 | — | |
LUGPTJMETIONMP
|
8.3 | IC50 | 3 | — |