Target Details
| UniProt AC | P78396 |
|---|---|
| Gene Symbol | CCNA1 |
| Protein Name | Cyclin-A1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02984 (Cyclin_C) PF00134 (Cyclin_N) PF16500 (Cyclin_N2) |
Summary
- Multi-target molecules 730
- Clinical molecules 121
- Avg pChEMBL 7.17
KEGG Pathways (12)
- AMPK signaling pathway
- Acute myeloid leukemia
- Cell cycle
- Cellular senescence
- Epstein-Barr virus infection
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human papillomavirus infection
- Pathways in cancer
- Progesterone-mediated oocyte maturation
- Transcriptional misregulation in cancer
- Viral carcinogenesis
Active Molecules (730)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YKJLUQWCJRSTKA
|
7.0 | IC50 | 5 | — | |
HOJYIPVBRINFGF
|
7.0 | IC50 | 3 | — | |
XZAWRWLSBCORLH
|
7.0 | IC50 | 3 | — | |
ZDEIBVDDZHUQLD
|
7.0 | IC50 | 3 | — | |
FPRGSAMEQUWSEZ
|
7.0 | IC50 | 3 | — | |
FTJPZMIPDWESGB
|
7.0 | IC50 | 3 | — | |
FQFGDUPFMGYOMB
|
7.0 | IC50 | 6 | — | |
IRMQPTLEJRNDAI
|
7.0 | IC50 | 3 | — | |
KWLUBUXQTWBTEJ
|
7.0 | IC50 | 3 | — | |
NMOPSVILFGBLLC
|
7.0 | IC50 | 6 | — | |
PHIBUDNSTRRWNP
|
7.0 | IC50 | 7 | Yes | |
RBUHYDCTYUXFLT
|
7.0 | IC50 | 3 | — | |
ZSSHCAVAAPDLII
|
7.0 | IC50 | 5 | — | |
BIIVYFLTOXDAOV
|
6.9 | IC50 | 82 | Yes | |
JPMKZYFDSNDPCM
|
6.9 | IC50 | 3 | — | |
ASRWRMWLFZMROI
|
6.9 | IC50 | 6 | — | |
CMLCAVWKWRNWPH
|
6.9 | IC50 | 3 | — | |
COGUZYALRYMQTD
|
6.9 | IC50 | 9 | — | |
HFEVNTGRPXCJIM
|
6.9 | IC50 | 6 | — | |
IQQAPAMUKYXXIQ
|
6.9 | IC50 | 4 | Yes | |
PRIGRJPRGZCFAS
|
6.9 | IC50 | 13 | Yes | |
SSEDQERECATUBR
|
6.9 | Ki | 5 | — | |
XFFCUJYCBFPUOA
|
6.9 | IC50 | 3 | — | |
KPMPMEOEHDFLEG
|
6.9 | IC50 | 3 | — | |
NCBDOQFSGNRAHL
|
6.9 | IC50 | 6 | — | |
WSZLNFZLFQJSAJ
|
6.9 | IC50 | 10 | Yes | |
XPEBENJJZXOJBA
|
6.9 | IC50 | 7 | Yes | |
DZHBFQMOLIUZMP
|
6.9 | Ki | 9 | — | |
UBKCVLVAEFXGTJ
|
6.9 | Ki | 5 | — | |
NSKDXALGDBAGSA
|
6.9 | IC50 | 4 | — | |
RBXFOVQKVXUOEG
|
6.9 | IC50 | 3 | — | |
CXBHMSHVCKEEGW
|
6.8 | IC50 | 5 | Yes | |
QWFWQJOFUNDIAZ
|
6.8 | IC50 | 7 | — | |
SCNMJGFMXAIFOK
|
6.8 | IC50 | 4 | — | |
SJCAIGIQEIAUQR
|
6.8 | IC50 | 3 | — | |
UNZVQIJLQQYQLN
|
6.8 | IC50 | 6 | — | |
VRFCKEOJPDSCNC
|
6.8 | IC50 | 5 | — | |
XAKCLNJQGRBKPQ
|
6.8 | IC50 | 5 | — | |
XOIQTGKKNJREKY
|
6.8 | IC50 | 3 | — | |
RLOPENNMNPVKFM
|
6.8 | IC50 | 3 | — | |
UFUGKBGESCNADR
|
6.8 | Ki | 7 | — | |
YNYBKXDJIMUFAQ
|
6.8 | IC50 | 3 | — | |
AONVCSVCAYXLEL
|
6.8 | IC50 | 3 | — | |
LCBAPHXEAOBWKR
|
6.8 | IC50 | 5 | — | |
MGCHCKUUSGHSES
|
6.8 | IC50 | 4 | — | |
RFPKDRLIUJAMFY
|
6.8 | IC50 | 3 | — | |
RPAYUDDKBDJILL
|
6.8 | IC50 | 7 | Yes | |
RUOIDLYFQJFGQQ
|
6.8 | IC50 | 3 | — | |
USIDNFXDNPBRBR
|
6.8 | IC50 | 5 | Yes | |
GMIZZEXBPRLVIV
|
6.8 | IC50 | 4 | — |