Target Details
| UniProt AC | P78396 |
|---|---|
| Gene Symbol | CCNA1 |
| Protein Name | Cyclin-A1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02984 (Cyclin_C) PF00134 (Cyclin_N) PF16500 (Cyclin_N2) |
Summary
- Multi-target molecules 730
- Clinical molecules 121
- Avg pChEMBL 7.17
KEGG Pathways (12)
- AMPK signaling pathway
- Acute myeloid leukemia
- Cell cycle
- Cellular senescence
- Epstein-Barr virus infection
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human papillomavirus infection
- Pathways in cancer
- Progesterone-mediated oocyte maturation
- Transcriptional misregulation in cancer
- Viral carcinogenesis
Active Molecules (730)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KLVYMYQTRZCMLE
|
7.1 | IC50 | 11 | Yes | |
KWKWTBFZIUSWFJ
|
7.1 | IC50 | 3 | — | |
MOSIOPGNCROISC
|
7.1 | IC50 | 3 | — | |
ZCNCKHAAOYENHC
|
7.1 | IC50 | 3 | — | |
INYWDKXOTYZOJX
|
7.1 | IC50 | 3 | — | |
IWXIAMLCFOOOMV
|
7.1 | IC50 | 8 | Yes | |
MHDFKOBMOQJFBJ
|
7.1 | IC50 | 3 | — | |
MHSDRURPTIXMJZ
|
7.1 | IC50 | 5 | — | |
WUTFIZGMCPBYJH
|
7.1 | Ki | 5 | — | |
DXZFQTAPRSQZBA
|
7.1 | IC50 | 4 | Yes | |
JETXRGKNZYUPEF
|
7.1 | IC50 | 6 | — | |
JPKKSVJWAFKQPI
|
7.1 | IC50 | 3 | — | |
KGFWOPNBCVKALC
|
7.1 | IC50 | 3 | — | |
TVSSLJHFDCVIRP
|
7.1 | IC50 | 3 | — | |
BWDFXIOBWGOKGE
|
7.1 | IC50 | 3 | — | |
CSEWCIIPSWNSJT
|
7.1 | IC50 | 3 | — | |
HGRMYMRCAGWXEQ
|
7.1 | IC50 | 6 | — | |
VMZGYYCCAWUCHJ
|
7.1 | IC50 | 4 | — | |
XXLVWAXFJXMBMJ
|
7.1 | IC50 | 3 | — | |
CXQJGJMKSNFPQC
|
7.1 | IC50 | 3 | — | |
IWYINOFYXWFKAR
|
7.1 | IC50 | 3 | — | |
NQIYAEQYNSJUOZ
|
7.1 | IC50 | 3 | — | |
ZHXQLMCSTVATST
|
7.1 | Ki | 9 | — | |
IUMARYQWTKVJMI
|
7.1 | IC50 | 3 | — | |
JSLLPPFWLQWPKD
|
7.1 | IC50 | 3 | — | |
NNLIBDONTYMYIU
|
7.1 | IC50 | 7 | Yes | |
ODEUXLJOADOSHS
|
7.1 | IC50 | 3 | — | |
RLYJZQKMTLQQIR
|
7.1 | IC50 | 3 | — | |
UJVJXKMEZMFCNM
|
7.1 | IC50 | 6 | — | |
WFZLOYYQIHKJAI
|
7.1 | IC50 | 3 | — | |
HQHSJJZIICGOIX
|
7.0 | IC50 | 8 | Yes | |
IFWRXHDSVNMZIT
|
7.0 | IC50 | 3 | — | |
MZMAYWNWHCZWNL
|
7.0 | IC50 | 3 | — | |
WRKQTFCCJAMNGR
|
7.0 | IC50 | 5 | — | |
KPQFNABLUHMRMB
|
7.0 | IC50 | 3 | — | |
OJPZPHHRLPRKHR
|
7.0 | IC50 | 6 | Yes | |
QNWXRLPZIFMTBK
|
7.0 | IC50 | 12 | — | |
RBPFQBARVLHLER
|
7.0 | IC50 | 3 | — | |
BHIZLKHDUFXUSQ
|
7.0 | IC50 | 3 | — | |
HDNVPRNOUJXPEZ
|
7.0 | IC50 | 3 | — | |
BBNBFSYCPUPPCC
|
7.0 | IC50 | 5 | — | |
DMMKWSKGQPTHGZ
|
7.0 | IC50 | 6 | — | |
HWIHAMKZTYYAKI
|
7.0 | IC50 | 7 | Yes | |
KTMGWYXHOHWEPU
|
7.0 | IC50 | 3 | — | |
NGDQZHZQUZQYHB
|
7.0 | IC50 | 5 | — | |
QFPGZNFSVUUBNZ
|
7.0 | IC50 | 3 | — | |
SWRFZQFPQPZUEQ
|
7.0 | IC50 | 3 | — | |
UTGQWJIIGZIEDP
|
7.0 | IC50 | 7 | Yes | |
UUXLORHYMYNKFC
|
7.0 | IC50 | 4 | — | |
VNUICWVLRHUNJF
|
7.0 | IC50 | 7 | Yes |