Target Details
| UniProt AC | P78396 |
|---|---|
| Gene Symbol | CCNA1 |
| Protein Name | Cyclin-A1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02984 (Cyclin_C) PF00134 (Cyclin_N) PF16500 (Cyclin_N2) |
Summary
- Multi-target molecules 730
- Clinical molecules 121
- Avg pChEMBL 7.17
KEGG Pathways (12)
- AMPK signaling pathway
- Acute myeloid leukemia
- Cell cycle
- Cellular senescence
- Epstein-Barr virus infection
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human papillomavirus infection
- Pathways in cancer
- Progesterone-mediated oocyte maturation
- Transcriptional misregulation in cancer
- Viral carcinogenesis
Active Molecules (730)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JRLCFYYHBUWFDK
|
7.3 | IC50 | 3 | — | |
XZZOVHIAPZXMHM
|
7.3 | IC50 | 4 | — | |
GYMVEDSUJRTLGP
|
7.3 | IC50 | 3 | — | |
KKCXFNXPIIHRJW
|
7.3 | IC50 | 3 | — | |
RGRWBAXPKCSYSG
|
7.3 | IC50 | 3 | — | |
FQJFTSMSJXOYME
|
7.2 | IC50 | 3 | — | |
HAVTUEFHYMRXDG
|
7.2 | IC50 | 7 | Yes | |
HMCJMBDXHYZRRL
|
7.2 | Ki | 9 | — | |
BTKRPPLRYLYGOR
|
7.2 | IC50 | 3 | — | |
DZQHZAAIBBSMPD
|
7.2 | IC50 | 3 | — | |
HWFOUEQKCWVCBH
|
7.2 | IC50 | 3 | — | |
KPEWGEQNXTXESG
|
7.2 | IC50 | 7 | Yes | |
RWZLXWPAWBIAIB
|
7.2 | IC50 | 3 | — | |
SCWFKTCRDHIMRO
|
7.2 | IC50 | 3 | — | |
VKQRQRVHRJQAAP
|
7.2 | IC50 | 2 | — | |
YUBJEBHGGUAVPW
|
7.2 | IC50 | 3 | — | |
HMAJGFYNRRZUJX
|
7.2 | IC50 | 4 | — | |
ISCPEDZQFVQCAM
|
7.2 | IC50 | 3 | — | |
NVLFLJAFSQNISZ
|
7.2 | IC50 | 3 | — | |
RANSINIOMGOPCF
|
7.2 | IC50 | 3 | — | |
XOLAFGHOWMROGX
|
7.2 | IC50 | 3 | — | |
BOYUIYWAXWEOCT
|
7.2 | IC50 | 3 | — | |
DTBMYSHZPNXMDE
|
7.2 | IC50 | 8 | Yes | |
QXBKFUBBGBWPCJ
|
7.2 | IC50 | 8 | — | |
XEMJTISGDXHELX
|
7.2 | IC50 | 8 | Yes | |
DHZFLITTYGDMNK
|
7.2 | IC50 | 3 | — | |
DMXIHKQKBYZIHM
|
7.2 | IC50 | 5 | Yes | |
ZZRNITRBTLLTQE
|
7.2 | IC50 | 3 | — | |
JWZMXYSZZSYDGV
|
7.2 | IC50 | 4 | — | |
ZKMCBDJTPIOLBR
|
7.2 | IC50 | 3 | — | |
GCEJQMWZAFXILZ
|
7.2 | IC50 | 3 | — | |
OSWILUKXEWYOHP
|
7.2 | IC50 | 3 | — | |
HGEJNHUGVPFHIF
|
7.2 | IC50 | 3 | — | |
MJSXSLBYCSPRHR
|
7.2 | IC50 | 10 | Yes | |
VBWXQPUACHCVRW
|
7.2 | IC50 | 3 | — | |
YFXWYMXXKFMSOB
|
7.2 | IC50 | 3 | — | |
ATBAETXFFCOZOY
|
7.2 | IC50 | 39 | — | |
GHLNHRXCRGGCPK
|
7.2 | IC50 | 3 | — | |
VVXLHYKOWIXRSV
|
7.2 | IC50 | 5 | — | |
WYJJUIPBAVISMJ
|
7.2 | IC50 | 7 | Yes | |
DUXWDMGSXRPDFV
|
7.1 | IC50 | 3 | — | |
SBNNOXYSSSCMJX
|
7.1 | IC50 | 6 | — | |
VAGPVIGSUDIGHA
|
7.1 | IC50 | 3 | — | |
FPBKUBUKBWJEMH
|
7.1 | IC50 | 7 | — | |
IEMIQIMEMFFPEZ
|
7.1 | IC50 | 3 | — | |
NTHMDBBWWNTVAZ
|
7.1 | IC50 | 5 | — | |
RJESYXNLLLQOLH
|
7.1 | IC50 | 3 | — | |
YHVVVHLDNQXTEZ
|
7.1 | IC50 | 3 | — | |
BHBIHSQEXUFLCT
|
7.1 | IC50 | 3 | — | |
BTJHWCJCRJUEGO
|
7.1 | IC50 | 7 | Yes |