Target Details
| UniProt AC | P78396 |
|---|---|
| Gene Symbol | CCNA1 |
| Protein Name | Cyclin-A1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02984 (Cyclin_C) PF00134 (Cyclin_N) PF16500 (Cyclin_N2) |
Summary
- Multi-target molecules 730
- Clinical molecules 121
- Avg pChEMBL 7.17
KEGG Pathways (12)
- AMPK signaling pathway
- Acute myeloid leukemia
- Cell cycle
- Cellular senescence
- Epstein-Barr virus infection
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human papillomavirus infection
- Pathways in cancer
- Progesterone-mediated oocyte maturation
- Transcriptional misregulation in cancer
- Viral carcinogenesis
Active Molecules (730)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DIKZCYKVEDCJAC
|
7.4 | IC50 | 3 | — | |
GZKUIKKDBXPCIY
|
7.4 | IC50 | 13 | Yes | |
HQTXGTXCDFXDLO
|
7.4 | IC50 | 3 | — | |
TXYKUCFACDXMFT
|
7.4 | IC50 | 7 | Yes | |
PUNSFHAWASZDFO
|
7.4 | IC50 | 3 | — | |
RIGZCVNCFXYBEG
|
7.4 | IC50 | 11 | Yes | |
UAOIPNOTWOYAMU
|
7.4 | IC50 | 11 | Yes | |
ZEHXSPZMRLUPSR
|
7.4 | IC50 | 7 | Yes | |
ATTMEZRDDPAMBY
|
7.4 | IC50 | 3 | — | |
HTRPJPBYPJZVLQ
|
7.4 | IC50 | 3 | — | |
RBAODIAUJYQMMC
|
7.4 | IC50 | 4 | — | |
SVBJNUDKKXGVHI
|
7.4 | IC50 | 5 | — | |
LOYSCNBYDPTSAA
|
7.4 | IC50 | 10 | — | |
QAWBPBLABQUSRL
|
7.4 | IC50 | 9 | — | |
QZEZKSMIUTYGRU
|
7.4 | IC50 | 9 | — | |
SZVPDWROAQYJHW
|
7.4 | IC50 | 3 | — | |
VWBUFGGJMMUSBL
|
7.4 | IC50 | 4 | — | |
GHBWBLLGGANTFE
|
7.4 | IC50 | 3 | — | |
MTIKFQKFTRIHCE
|
7.4 | IC50 | 3 | — | |
UGLMDRPTTBWXIB
|
7.4 | IC50 | 3 | — | |
BCKLVLDQAAHMQR
|
7.4 | Ki | 9 | — | |
MCFCYLCLAYXQIZ
|
7.4 | Ki | 9 | — | |
BGPUFSMDGGQOIE
|
7.4 | Ki | 9 | — | |
DQKJGZAOXUAOIO
|
7.3 | IC50 | 3 | — | |
GRIBJJIZUIEJFG
|
7.3 | IC50 | 3 | — | |
IRXXTCIJUUOCGV
|
7.3 | IC50 | 3 | — | |
YZRRSIPTHDIILM
|
7.3 | Ki | 9 | — | |
HMAFXPLOLABOEY
|
7.3 | IC50 | 3 | — | |
JSJVSQMHVJPNON
|
7.3 | IC50 | 5 | — | |
OQCYIOKKFGCDSR
|
7.3 | IC50 | 4 | Yes | |
ORRMXVSTILKSNY
|
7.3 | IC50 | 3 | — | |
PMXCMJLOPOFPBT
|
7.3 | IC50 | 17 | Yes | |
MTCJIHKSTBDECF
|
7.3 | IC50 | 3 | — | |
OVPNQJVDAFNBDN
|
7.3 | IC50 | 44 | Yes | |
WPBZYJGEMAIFMZ
|
7.3 | IC50 | 3 | — | |
YVYVDXXWQANVCI
|
7.3 | IC50 | 4 | — | |
MYIYDTISJDJCKB
|
7.3 | IC50 | 3 | — | |
UDYXTWRJETXAKK
|
7.3 | IC50 | 4 | — | |
AHWMQFPWQLNDNV
|
7.3 | IC50 | 3 | — | |
DMTKMRCNVGYHOZ
|
7.3 | IC50 | 9 | — | |
ITHULDOZQFKWFX
|
7.3 | IC50 | 3 | — | |
WYMXGRUKKZVBIY
|
7.3 | IC50 | 3 | — | |
KTIAVDWJHSVFJO
|
7.3 | IC50 | 3 | — | |
OOYUOUNLWCMZHC
|
7.3 | IC50 | 3 | — | |
SVBJNUDKKXGVHI
|
7.3 | IC50 | 6 | — | |
VMSMVRDDPGJMQF
|
7.3 | IC50 | 6 | — | |
ZEJXJYCOUVOWGJ
|
7.3 | IC50 | 13 | Yes | |
ACXFBDRQBQFLGH
|
7.3 | IC50 | 3 | — | |
AMTPXYFBGSXPMD
|
7.3 | IC50 | 3 | — | |
GNTSKAUZBDGNGK
|
7.3 | IC50 | 6 | — |