Target Details
| UniProt AC | P78396 |
|---|---|
| Gene Symbol | CCNA1 |
| Protein Name | Cyclin-A1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02984 (Cyclin_C) PF00134 (Cyclin_N) PF16500 (Cyclin_N2) |
Summary
- Multi-target molecules 730
- Clinical molecules 121
- Avg pChEMBL 7.17
KEGG Pathways (12)
- AMPK signaling pathway
- Acute myeloid leukemia
- Cell cycle
- Cellular senescence
- Epstein-Barr virus infection
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human papillomavirus infection
- Pathways in cancer
- Progesterone-mediated oocyte maturation
- Transcriptional misregulation in cancer
- Viral carcinogenesis
Active Molecules (730)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DUZMNSPOOJGCPL
|
7.6 | IC50 | 3 | — | |
HCLVUOIGTCCQQB
|
7.6 | IC50 | 3 | — | |
IRQVBNQXTXFQTM
|
7.6 | IC50 | 3 | — | |
ZPKXDHHDZZKMKI
|
7.6 | IC50 | 6 | — | |
IUVOVXQLMSRQDH
|
7.6 | IC50 | 3 | — | |
LBVIZFWUIQSZHP
|
7.6 | IC50 | 10 | — | |
ORKGHNGKNDEWIV
|
7.6 | IC50 | 3 | — | |
PWMQUOFEZWCTAE
|
7.6 | IC50 | 3 | — | |
VQNXOAVFMIVTAT
|
7.6 | IC50 | 7 | Yes | |
YOPGDOJJGFKDRC
|
7.6 | IC50 | 3 | — | |
KSDTZAWGXZOFIW
|
7.6 | IC50 | 4 | — | |
GQDHKYZSKSDSNQ
|
7.6 | IC50 | 3 | — | |
TZBRTWANJDQXNF
|
7.6 | IC50 | 3 | — | |
VLBVJPDXCSRGGN
|
7.6 | IC50 | 3 | — | |
XNKBKFNLOYVTSF
|
7.6 | IC50 | 3 | — | |
HFTMAKGAOQSXPI
|
7.6 | IC50 | 3 | — | |
NUXMDKWZVUQHTP
|
7.6 | IC50 | 3 | — | |
AGRGOPGRMMWYAC
|
7.6 | IC50 | 3 | — | |
AGRGOPGRMMWYAC
|
7.6 | IC50 | 3 | — | |
ITRNHZPVFGOWGQ
|
7.6 | IC50 | 3 | — | |
CDNCNMWWSCRJGY
|
7.5 | IC50 | 3 | — | |
HFEVNTGRPXCJIM
|
7.5 | IC50 | 6 | — | |
LEDNSKJDSVXHBN
|
7.5 | IC50 | 3 | — | |
OYBUHXCVUFCTQD
|
7.5 | IC50 | 3 | — | |
NTUSSPZSLWLBQF
|
7.5 | IC50 | 3 | — | |
PUXCYCHNNDMPTI
|
7.5 | IC50 | 3 | — | |
SBNNOXYSSSCMJX
|
7.5 | IC50 | 6 | — | |
XRHXLPUHGOTIJG
|
7.5 | IC50 | 3 | — | |
YPRFZGADERCJFT
|
7.5 | IC50 | 3 | — | |
ZRKZVQWEOWMPPZ
|
7.5 | IC50 | 3 | — | |
UGZGQNGZCRYGKF
|
7.5 | IC50 | 3 | — | |
ABDGGOBNHQMXIJ
|
7.5 | IC50 | 3 | Yes | |
AMPGTDPLFIQJLI
|
7.5 | IC50 | 3 | — | |
BDRDBXXWQDFXEC
|
7.5 | IC50 | 5 | Yes | |
BOLOCLITWRGHFA
|
7.5 | IC50 | 6 | — | |
CDEIEGNYDSWLCD
|
7.5 | IC50 | 3 | — | |
CHSPOGGCOKIJJT
|
7.5 | IC50 | 3 | — | |
LRKDOQPVSVUIPK
|
7.5 | IC50 | 3 | — | |
NSLNFDFRWNVNFZ
|
7.5 | IC50 | 3 | — | |
BGFIVDZJUZNYNB
|
7.5 | IC50 | 3 | — | |
LMEANLPGOCWAMD
|
7.5 | IC50 | 3 | — | |
MRLPFDAKEJSGRI
|
7.5 | IC50 | 3 | — | |
AOJLBKYLAVRMQT
|
7.5 | IC50 | 3 | — | |
NQQUFCAHMNCUIZ
|
7.5 | IC50 | 3 | — | |
HSOAJSRVFMRIRY
|
7.5 | IC50 | 3 | — | |
JKLNMYJBWWAZSO
|
7.5 | IC50 | 3 | — | |
FLXKJXLZBWOYGN
|
7.5 | IC50 | 3 | — | |
LVJZZDNNQXAXPX
|
7.5 | Ki | 7 | — | |
NUDSGDYZHKNNPW
|
7.5 | IC50 | 3 | — | |
MXLJQTVDWFSRDC
|
7.5 | IC50 | 3 | — |