Target Details
| UniProt AC | P78396 |
|---|---|
| Gene Symbol | CCNA1 |
| Protein Name | Cyclin-A1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02984 (Cyclin_C) PF00134 (Cyclin_N) PF16500 (Cyclin_N2) |
Summary
- Multi-target molecules 730
- Clinical molecules 121
- Avg pChEMBL 7.17
KEGG Pathways (12)
- AMPK signaling pathway
- Acute myeloid leukemia
- Cell cycle
- Cellular senescence
- Epstein-Barr virus infection
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human papillomavirus infection
- Pathways in cancer
- Progesterone-mediated oocyte maturation
- Transcriptional misregulation in cancer
- Viral carcinogenesis
Active Molecules (730)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AVMGEAZKDWAZIC
|
7.9 | IC50 | 3 | — | |
NCKHSDFHCYCSFF
|
7.8 | IC50 | 3 | — | |
NCSLRHGXEKHUGV
|
7.8 | IC50 | 3 | — | |
RNNCVRNBQXSBEN
|
7.8 | IC50 | 3 | — | |
UOSAKCKTUUCAQF
|
7.8 | IC50 | 3 | — | |
VMSMVRDDPGJMQF
|
7.8 | IC50 | 5 | — | |
YRWDEKPEPUVMIZ
|
7.8 | IC50 | 3 | — | |
DZFYFXAPZWMNAS
|
7.8 | IC50 | 3 | — | |
KGLRLXMTNCPNET
|
7.8 | IC50 | 3 | Yes | |
OLUKILHGKRVDCT
|
7.8 | IC50 | 44 | Yes | |
RVGFQABNRSQREF
|
7.8 | IC50 | 3 | — | |
SYCCUDVKTARJAW
|
7.8 | IC50 | 3 | — | |
GRJMSFULANHLPW
|
7.8 | IC50 | 3 | — | |
KHUWOOWXQFGVBZ
|
7.8 | IC50 | 7 | — | |
MUPFEKGTMRGPLJ
|
7.8 | IC50 | 3 | — | |
RSCVJZXCKTYHOT
|
7.8 | IC50 | 3 | — | |
OVSVIUOGHPWXNH
|
7.8 | IC50 | 6 | — | |
QXAKKDDDYAESLJ
|
7.8 | IC50 | 6 | Yes | |
WVVCBUMOFSHDAJ
|
7.8 | IC50 | 3 | — | |
YOWFAJOGDAREKF
|
7.8 | IC50 | 3 | — | |
YPRFZGADERCJFT
|
7.8 | IC50 | 3 | — | |
ASRWRMWLFZMROI
|
7.8 | IC50 | 6 | — | |
JYGNOLIKBUTZNC
|
7.8 | IC50 | 8 | Yes | |
ZPKXDHHDZZKMKI
|
7.8 | IC50 | 6 | — | |
AGULHSVYEDTEEI
|
7.7 | IC50 | 3 | — | |
BTYJREGEVYGXIK
|
7.7 | IC50 | 3 | — | |
JKEKTNKQNJPFHO
|
7.7 | IC50 | 3 | — | |
UOZGSFYRTXKQQR
|
7.7 | IC50 | 6 | Yes | |
ZLKKDZBQWFTZAN
|
7.7 | IC50 | 3 | — | |
AJFMJEKRFWUUMF
|
7.7 | IC50 | 3 | — | |
BCTKIAROAQVJQI
|
7.7 | IC50 | 3 | — | |
BNBOPMICSCGSGW
|
7.7 | IC50 | 3 | — | |
CKIFWVSQRJHDKI
|
7.7 | Ki | 9 | — | |
FQFGDUPFMGYOMB
|
7.7 | IC50 | 6 | — | |
HXZXJLLRGFULES
|
7.7 | Ki | 9 | — | |
NCBDOQFSGNRAHL
|
7.7 | IC50 | 6 | — | |
PQTPLILJDUSKCC
|
7.7 | IC50 | 3 | — | |
QDKYQDQBFZUQHE
|
7.7 | IC50 | 3 | — | |
UUPHPKKIPSWLBT
|
7.7 | IC50 | 3 | — | |
XNKBKFNLOYVTSF
|
7.7 | IC50 | 11 | — | |
BKQWSKYSXQIREO
|
7.7 | IC50 | 3 | — | |
JEMMIJOETMAKME
|
7.7 | IC50 | 7 | Yes | |
OAXIWAHMCPRCIQ
|
7.7 | IC50 | 3 | — | |
OPCCGXSXPYCKGR
|
7.7 | IC50 | 3 | — | |
OUSFTKFNBAZUKL
|
7.7 | IC50 | 58 | Yes | |
SYBNWJLVMPEJGJ
|
7.7 | IC50 | 3 | — | |
UOLGGWWZSJIIHY
|
7.7 | IC50 | 3 | — | |
ZCUPTZASSFWMPJ
|
7.7 | IC50 | 3 | — | |
BUVPYHQHZUQYBS
|
7.7 | IC50 | 7 | Yes | |
AUTIVJGNZXILJJ
|
7.6 | IC50 | 3 | — |