Target Details
| UniProt AC | P78396 |
|---|---|
| Gene Symbol | CCNA1 |
| Protein Name | Cyclin-A1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02984 (Cyclin_C) PF00134 (Cyclin_N) PF16500 (Cyclin_N2) |
Summary
- Multi-target molecules 730
- Clinical molecules 121
- Avg pChEMBL 7.17
KEGG Pathways (12)
- AMPK signaling pathway
- Acute myeloid leukemia
- Cell cycle
- Cellular senescence
- Epstein-Barr virus infection
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human papillomavirus infection
- Pathways in cancer
- Progesterone-mediated oocyte maturation
- Transcriptional misregulation in cancer
- Viral carcinogenesis
Active Molecules (730)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OYDGHJTZNAFKAQ
|
8.2 | IC50 | 6 | Yes | |
UBJOERFPSFZJGL
|
8.2 | IC50 | 3 | — | |
UUINGAOFFFDPBY
|
8.2 | IC50 | 5 | Yes | |
GFXJPWQHPZNCGC
|
8.1 | IC50 | 3 | — | |
VXGBFWNTVZKGOT
|
8.1 | IC50 | 3 | — | |
DRYXVGHAKVVZFL
|
8.1 | IC50 | 3 | — | |
HUXYBQXJVXOMKX
|
8.1 | IC50 | 28 | — | |
HZRJYORBAMJSIQ
|
8.1 | IC50 | 7 | Yes | |
ILYYGWWTDBOGTR
|
8.1 | IC50 | 3 | — | |
MYMHNTVTLZQVKZ
|
8.1 | IC50 | 7 | Yes | |
QWTLNMRLRGDLQY
|
8.1 | IC50 | 3 | — | |
XZDHZYQSEWOJPD
|
8.1 | IC50 | 3 | — | |
XCBJCPRTHXKIAE
|
8.1 | IC50 | 3 | — | |
WSRSUSKJBOADHJ
|
8.1 | IC50 | 3 | — | |
MDPQZSCXKLJMQD
|
8.1 | IC50 | 7 | Yes | |
QKWMIPQJODDALR
|
8.1 | IC50 | 3 | — | |
WDHVWMXOJHHBQJ
|
8.1 | IC50 | 3 | — | |
WTJYXNCBJUYEKS
|
8.1 | IC50 | 3 | — | |
YUZFQJVRZIQCGL
|
8.1 | IC50 | 3 | — | |
NPLHHQHEODJUBY
|
8.0 | IC50 | 6 | — | |
KJVSTAAHJQPRFJ
|
8.0 | IC50 | 3 | — | |
GCYXEGSPUDSZJY
|
8.0 | IC50 | 17 | Yes | |
JPAVVQWCECWANY
|
8.0 | IC50 | 3 | — | |
KTERAHWGWLFDLN
|
8.0 | IC50 | 3 | — | |
MANZCDIQWXSESD
|
8.0 | IC50 | 3 | — | |
PYFVXOCGURDMHR
|
8.0 | IC50 | 3 | — | |
QVMLLKMJKQGGDX
|
8.0 | IC50 | 3 | — | |
ZOLPUEOXQAILTM
|
8.0 | Ki | 9 | — | |
WAFHXBBZJZYUIJ
|
8.0 | IC50 | 7 | — | |
GGEWEQJWGGJUHO
|
8.0 | IC50 | 8 | Yes | |
HTFBNTYFTGIOEK
|
8.0 | IC50 | 7 | — | |
IOOBSCBCJCFBKU
|
8.0 | IC50 | 3 | — | |
JNMFNQYJOKDMNT
|
8.0 | IC50 | 3 | — | |
SMHOLGURUXBSTC
|
8.0 | IC50 | 3 | — | |
MQQJPZHXGJGMDE
|
7.9 | IC50 | 3 | — | |
BJDCORPGTMJYTL
|
7.9 | IC50 | 3 | — | |
CUZZHCAJGYQFDT
|
7.9 | IC50 | 3 | — | |
NYRVLHGVDPPWJS
|
7.9 | Ki | 5 | — | |
VIHUAIODGTUZLN
|
7.9 | IC50 | 3 | — | |
XUGUDFCFRSMZSF
|
7.9 | IC50 | 3 | — | |
FOIWJMGHUDACNX
|
7.9 | IC50 | 3 | — | |
GAFYDJGFHJBXQQ
|
7.9 | Ki | 9 | — | |
KRKQVGZXTNLQSV
|
7.9 | IC50 | 9 | Yes | |
NOQYGKAHNPQBEW
|
7.9 | IC50 | 3 | — | |
OUFGAEIXDBKNPC
|
7.9 | IC50 | 3 | — | |
RLTFKHPSPUGIRA
|
7.9 | IC50 | 3 | — | |
VXBAJLGYBMTJCY
|
7.9 | IC50 | 34 | Yes | |
WAJZMHFJIYMYOJ
|
7.9 | IC50 | 3 | — | |
ZUSSYTUFZXQWGO
|
7.9 | IC50 | 4 | — | |
OEHHKRVHXQAAQT
|
7.9 | IC50 | 3 | — |