Target Details
| UniProt AC | P78396 |
|---|---|
| Gene Symbol | CCNA1 |
| Protein Name | Cyclin-A1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02984 (Cyclin_C) PF00134 (Cyclin_N) PF16500 (Cyclin_N2) |
Summary
- Multi-target molecules 730
- Clinical molecules 121
- Avg pChEMBL 7.17
KEGG Pathways (12)
- AMPK signaling pathway
- Acute myeloid leukemia
- Cell cycle
- Cellular senescence
- Epstein-Barr virus infection
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human papillomavirus infection
- Pathways in cancer
- Progesterone-mediated oocyte maturation
- Transcriptional misregulation in cancer
- Viral carcinogenesis
Active Molecules (730)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OXPLZKSKLWBEIM
|
8.5 | IC50 | 8 | Yes | |
PIMQWRZWLQKKBJ
|
8.5 | IC50 | 36 | — | |
WEHOMMKULWQPKY
|
8.5 | IC50 | 3 | — | |
YVRLFXOPNVVCQT
|
8.5 | Ki | 5 | — | |
ZHMRPXZRUZLCNL
|
8.5 | IC50 | 8 | Yes | |
ZOBRPBVIEUWYJR
|
8.5 | IC50 | 5 | Yes | |
VUVZPZAXDNURQR
|
8.5 | IC50 | 3 | — | |
WTKYHVUVQSLNBW
|
8.5 | IC50 | 6 | — | |
QQWUCWPOJLZHJB
|
8.4 | IC50 | 3 | — | |
ABEYZUJMIYFBTH
|
8.4 | IC50 | 3 | — | |
HHYDLEDJMDNGIO
|
8.4 | IC50 | 3 | — | |
KMVQBPWEFOSEIR
|
8.4 | IC50 | 3 | — | |
LDTOTGIFPXIEOT
|
8.4 | IC50 | 3 | — | |
MGCAXDANYPKQKY
|
8.4 | IC50 | 4 | — | |
OTPFZAVDWPCJLJ
|
8.4 | Ki | 9 | — | |
SGOFFNQMBSXTRU
|
8.4 | Ki | 9 | — | |
XCYGTFKOOGNUMR
|
8.4 | IC50 | 5 | Yes | |
ZODJDUZBNLTRCH
|
8.4 | IC50 | 3 | — | |
NEQUYNFKQDRNGP
|
8.3 | IC50 | 3 | — | |
NYFSAYXCSAIWGI
|
8.3 | IC50 | 3 | — | |
ALWICLGIEFINRR
|
8.3 | IC50 | 3 | — | |
CDKRFBBXZQUTDX
|
8.3 | Ki | 9 | — | |
DFBJIWSACMQONP
|
8.3 | IC50 | 4 | — | |
DLFAVSIXCMXECW
|
8.3 | IC50 | 3 | — | |
GVDMJOHUPKJFQU
|
8.3 | IC50 | 3 | — | |
HWASNOYCCGHVQF
|
8.3 | IC50 | 5 | Yes | |
KORLUXLXWXODAL
|
8.3 | IC50 | 3 | — | |
LNXFGXNXUQLHLF
|
8.3 | IC50 | 3 | — | |
PWURWOZBUAQZAZ
|
8.3 | IC50 | 3 | — | |
RMWMYMKOIOFLED
|
8.3 | IC50 | 3 | — | |
WPIFRGDKXSWKPX
|
8.3 | IC50 | 5 | Yes | |
YYOQLHOTDBEPGW
|
8.3 | IC50 | 3 | — | |
YRURITXEWXPMAI
|
8.3 | IC50 | 8 | Yes | |
QIILXVJHCJSXQI
|
8.3 | IC50 | 3 | — | |
OWXORKPNCHJYOF
|
8.3 | IC50 | 17 | Yes | |
DVPVWROTHYIYLX
|
8.2 | IC50 | 3 | — | |
UDVJBRYBBSVDDS
|
8.2 | IC50 | 14 | — | |
AHUQZOZSCWOMOS
|
8.2 | IC50 | 4 | — | |
DVXZIFWSUHATCY
|
8.2 | IC50 | 3 | — | |
ROSDVEJRVQTUEV
|
8.2 | IC50 | 3 | — | |
UGPIPEQLSUSUOZ
|
8.2 | IC50 | 3 | — | |
VJMCWOUEUKZFIB
|
8.2 | IC50 | 3 | — | |
XBIWTDZZJVRIIX
|
8.2 | IC50 | 3 | — | |
ZKDXRFMOHZVXSG
|
8.2 | IC50 | 13 | Yes | |
AAYPLLWGPJQWCC
|
8.2 | IC50 | 15 | Yes | |
CJJMNECGBUPMAV
|
8.2 | IC50 | 8 | Yes | |
DPROZSHCTFNYSW
|
8.2 | IC50 | 6 | Yes | |
JCRCSNBABSGPEN
|
8.2 | IC50 | 7 | Yes | |
LNYKHAPIJVILRZ
|
8.2 | IC50 | 7 | Yes | |
NOAACOSHLOXNIY
|
8.2 | IC50 | 3 | — |