Target Details
| UniProt AC | P78396 |
|---|---|
| Gene Symbol | CCNA1 |
| Protein Name | Cyclin-A1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02984 (Cyclin_C) PF00134 (Cyclin_N) PF16500 (Cyclin_N2) |
Summary
- Multi-target molecules 730
- Clinical molecules 121
- Avg pChEMBL 7.17
KEGG Pathways (12)
- AMPK signaling pathway
- Acute myeloid leukemia
- Cell cycle
- Cellular senescence
- Epstein-Barr virus infection
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human papillomavirus infection
- Pathways in cancer
- Progesterone-mediated oocyte maturation
- Transcriptional misregulation in cancer
- Viral carcinogenesis
Active Molecules (730)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PHLVHKVYPBUWOL
|
6.8 | IC50 | 7 | — | |
PUIIOZKFJGRCIW
|
6.8 | IC50 | 3 | — | |
RYVKHHFVVPELDV
|
6.8 | IC50 | 3 | — | |
WYZJNWDUVFKVRN
|
6.8 | IC50 | 3 | — | |
ZWHTWAOLEGXRTP
|
6.8 | IC50 | 5 | — | |
XOKMDOXIMWIBTG
|
6.8 | IC50 | 3 | — | |
BUKNIOLWHFXEIG
|
6.8 | IC50 | 6 | — | |
KFBWYQJUHSEIDI
|
6.8 | IC50 | 7 | Yes | |
OUFGAEIXDBKNPC
|
6.8 | IC50 | 3 | — | |
SRYUEFQETIIMNO
|
6.8 | IC50 | 4 | — | |
UAOIPNOTWOYAMU
|
6.8 | IC50 | 3 | — | |
WAORXCNOCDHNFB
|
6.8 | IC50 | 4 | — | |
XXLVWAXFJXMBMJ
|
6.8 | IC50 | 3 | — | |
ZCQQEWOROAMZJH
|
6.8 | IC50 | 3 | — | |
GMMJFFFHKSLXFV
|
6.8 | IC50 | 3 | — | |
YQMXFJYNHFPIRQ
|
6.8 | IC50 | 3 | — | |
BSVWYBFSOQGZFD
|
6.8 | IC50 | 3 | — | |
CGHADMRBCNGDHX
|
6.8 | IC50 | 8 | Yes | |
FWFMLCFXVACEPD
|
6.8 | IC50 | 3 | — | |
IOPNYIOXLBPQAF
|
6.8 | IC50 | 3 | — | |
RAXSAOMTCOKDBJ
|
6.7 | IC50 | 3 | — | |
RKCBSCHBRMVAOI
|
6.7 | IC50 | 3 | — | |
BPFHXLYKZFEZRE
|
6.7 | IC50 | 5 | — | |
FHDFIUFWMGMGTR
|
6.7 | IC50 | 5 | — | |
GPQIBYPHUDMSPA
|
6.7 | IC50 | 3 | — | |
GSTGMOJCZPXYBR
|
6.7 | IC50 | 3 | — | |
LQYHWFFRRIMAPW
|
6.7 | IC50 | 5 | — | |
LSEHLBIXAOGNBF
|
6.7 | IC50 | 5 | — | |
MUPFBXXZGZFXEZ
|
6.7 | IC50 | 6 | Yes | |
NUXNHYJNSHRNAN
|
6.7 | IC50 | 3 | — | |
POYXCJPTKLIEPQ
|
6.7 | IC50 | 5 | — | |
PVKVVNSXCCOROL
|
6.7 | IC50 | 7 | Yes | |
QKQHOBLWOPPYDH
|
6.7 | IC50 | 5 | — | |
UHWJFOMTKXVUFY
|
6.7 | IC50 | 4 | — | |
WATZRHFPUUTHEW
|
6.7 | IC50 | 3 | — | |
WLFYGMMLYPUPNR
|
6.7 | IC50 | 3 | — | |
YAVWDSSODXPSHQ
|
6.7 | IC50 | 7 | Yes | |
ZUPLIVGNVOWXJE
|
6.7 | IC50 | 3 | — | |
APFZUNBSYNZMFG
|
6.7 | IC50 | 4 | — | |
BKDUVKJYBJDZQW
|
6.7 | IC50 | 7 | Yes | |
GXNUDSNBBQOPIA
|
6.7 | IC50 | 4 | — | |
IGNFICQZFLTMED
|
6.7 | IC50 | 3 | — | |
PBWZYCBGLAEXQD
|
6.7 | IC50 | 3 | — | |
RGCTVKIRPPNPGC
|
6.7 | IC50 | 3 | — | |
TVRWSLUHAPQTGR
|
6.7 | IC50 | 3 | — | |
UVANEUUATLLBKA
|
6.7 | IC50 | 7 | — | |
VGAXWFQZQONAPZ
|
6.7 | IC50 | 6 | — | |
VMUOSMBOEBOHFE
|
6.7 | IC50 | 3 | — | |
VRMCCAPNDOJKRZ
|
6.7 | IC50 | 3 | — | |
DHJHGYYBWIWMJK
|
6.7 | IC50 | 3 | — |