Target Details
| UniProt AC | P78396 |
|---|---|
| Gene Symbol | CCNA1 |
| Protein Name | Cyclin-A1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02984 (Cyclin_C) PF00134 (Cyclin_N) PF16500 (Cyclin_N2) |
Summary
- Multi-target molecules 730
- Clinical molecules 121
- Avg pChEMBL 7.17
KEGG Pathways (12)
- AMPK signaling pathway
- Acute myeloid leukemia
- Cell cycle
- Cellular senescence
- Epstein-Barr virus infection
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human papillomavirus infection
- Pathways in cancer
- Progesterone-mediated oocyte maturation
- Transcriptional misregulation in cancer
- Viral carcinogenesis
Active Molecules (730)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AEIHOULIOWEFLO
|
9.7 | Ki | 5 | — | |
BHQZGGSZRHDQFZ
|
9.5 | IC50 | 13 | Yes | |
HGAKLLFPOGATII
|
9.5 | IC50 | 3 | — | |
KQWTXAWKBUUOMU
|
9.4 | IC50 | 20 | Yes | |
ARIOBGGRZJITQX
|
9.3 | IC50 | 24 | — | |
CXOQOETYRJXMGY
|
9.2 | IC50 | 3 | — | |
AJDJBEBKIUAWFT
|
9.0 | IC50 | 3 | — | |
BWONSNVPSAEXDY
|
9.0 | Ki | 9 | — | |
KTHBXZCLQRQLAW
|
9.0 | IC50 | 3 | — | |
LXPGTNVSVSANEJ
|
9.0 | IC50 | 3 | — | |
NRGPURJFHVVJFI
|
9.0 | IC50 | 3 | — | |
OKCKMDCMHXPONP
|
9.0 | IC50 | 3 | — | |
OOKAYBMMWNSBPA
|
9.0 | Ki | 9 | — | |
RRFFYQAIEDMMQD
|
9.0 | IC50 | 3 | — | |
VBQONCXEWJGAOC
|
9.0 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
8.8 | IC50 | 408 | — | |
FPHITTVVVWKENE
|
8.8 | Ki | 9 | — | |
FLFGOZHEFLZZRQ
|
8.8 | IC50 | 3 | — | |
UOYOWVPLBRMQFZ
|
8.8 | IC50 | 3 | — | |
JXJHPQHLHQTQQI
|
8.7 | IC50 | 15 | — | |
CXWKPXGAGKBITA
|
8.7 | IC50 | 3 | — | |
FJXHHPBKCWCXDJ
|
8.7 | IC50 | 3 | — | |
ASUFRYKYWHJUIO
|
8.7 | Ki | 9 | — | |
BJDCORPGTMJYTL
|
8.7 | IC50 | 3 | — | |
BXMBIVXDTXURDF
|
8.7 | Ki | 9 | — | |
CQWBHMMWZICZRH
|
8.7 | IC50 | 10 | — | |
KDKUVYLMPJIGKA
|
8.7 | IC50 | 91 | Yes | |
KFFAVLFSAMSPDH
|
8.7 | IC50 | 3 | — | |
KIVYVNLAIOQLEN
|
8.7 | IC50 | 3 | — | |
KOLSEKSFVMGHDV
|
8.7 | IC50 | 12 | — | |
KUCYABDDCHEOBN
|
8.7 | IC50 | 3 | — | |
NTHSDAJAHNMPGF
|
8.7 | IC50 | 3 | — | |
OMOOZNJIAYMBSP
|
8.7 | IC50 | 5 | Yes | |
OUFGAEIXDBKNPC
|
8.7 | IC50 | 3 | — | |
PBJNPQMXAFFDSZ
|
8.7 | IC50 | 3 | — | |
UTHWBIPHRYUJSU
|
8.7 | IC50 | 11 | Yes | |
VIUFPQPXJYQVSE
|
8.7 | IC50 | 3 | — | |
XWQNZYCWLMEIBB
|
8.7 | IC50 | 5 | Yes | |
YUJZDAUCYWRKAP
|
8.7 | IC50 | 3 | — | |
ZYQXOZKYXADECC
|
8.7 | IC50 | 5 | Yes | |
NMWURSLYBLOJKP
|
8.7 | IC50 | 3 | — | |
JGWMRHPAGIJSBO
|
8.7 | IC50 | 3 | — | |
VXLAKHWYGRKCGI
|
8.6 | IC50 | 9 | — | |
AFMWZFUPVUGJPF
|
8.5 | IC50 | 3 | — | |
AXAQVNRYNMCZCK
|
8.5 | Ki | 10 | Yes | |
DIASEXMEBNQQHZ
|
8.5 | IC50 | 13 | — | |
GAIOPWBQKZMUNO
|
8.5 | Ki | 13 | — | |
HJKBVLZABNNRFO
|
8.5 | IC50 | 5 | Yes | |
KZKOIZXRAQJRPY
|
8.5 | Ki | 5 | — | |
LQBKAYJFACGUCC
|
8.5 | IC50 | 3 | — |