Target Details
| UniProt AC | P78368 |
|---|---|
| Gene Symbol | CSNK1G2 |
| Protein Name | Casein kinase I isoform gamma-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12605 (CK1gamma_C) PF00069 (Pkinase) |
Summary
- Multi-target molecules 121
- Clinical molecules 6
- Avg pChEMBL 6.7
KEGG Pathways (1)
Active Molecules (121)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OMKZJNFKGWJFNX
|
6.1 | Ki | 8 | — | |
RYAVJHIPOWNWDE
|
6.1 | Ki | 38 | — | |
UTMRCMCLMBDPNW
|
6.1 | Ki | 10 | — | |
ODPGGGTTYSGTGO
|
6.0 | Kd | 153 | — | |
QDITZBLZQQZVEE
|
6.0 | Kd | 19 | — | |
CPGKMMMSMJKHDL
|
6.0 | Ki | 16 | — | |
CQBBMNXXVMOFCA
|
6.0 | Ki | 39 | — | |
FQEODTMNWMDUMD
|
6.0 | Ki | 25 | — | |
GQLWKGVBOIYMTN
|
6.0 | Ki | 35 | — | |
IQNOGQGSOHNMCL
|
6.0 | Ki | 14 | — | |
ISVHLTLEHRZKJC
|
6.0 | Ki | 19 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
LVECPYVAIBNSRV
|
6.0 | Ki | 33 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
MGNQNQOSSLCUFP
|
6.0 | Ki | 12 | — | |
PYDWRLNPMMKKCI
|
6.0 | Ki | 7 | — | |
PYQFQGXOARMGAQ
|
6.0 | IC50 | 11 | — | |
TZSJMSZEKQGCBI
|
6.0 | Ki | 15 | — | |
XSDJOIOVIMPMHD
|
6.0 | Ki | 44 | — | |
ZPVLRSVLOWVDJC
|
6.0 | Ki | 14 | — |