Target Details
| UniProt AC | P78368 |
|---|---|
| Gene Symbol | CSNK1G2 |
| Protein Name | Casein kinase I isoform gamma-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12605 (CK1gamma_C) PF00069 (Pkinase) |
Summary
- Multi-target molecules 121
- Clinical molecules 6
- Avg pChEMBL 6.7
KEGG Pathways (1)
Active Molecules (121)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HWGZXYUOXGVACR
|
6.6 | Ki | 6 | — | |
NEWAULHLLUCDPD
|
6.6 | Ki | 27 | — | |
SPOBBSBKXJKGBG
|
6.6 | Ki | 16 | — | |
VBIYDORVDCFKHM
|
6.6 | Ki | 13 | — | |
VXYDJXMHISGSDA
|
6.6 | Ki | 59 | — | |
XUZMWHLSFXCVMG
|
6.6 | Kd | 24 | — | |
BGVLELSCIHASRV
|
6.6 | Kd | 12 | — | |
BGVLELSCIHASRV
|
6.6 | Kd | 12 | — | |
DPDZHVCKYBCJHW
|
6.5 | IC50 | 11 | — | |
BPNUQXPIQBZCMR
|
6.5 | Ki | 60 | — | |
CLRFYTGANQZOBS
|
6.5 | Ki | 41 | — | |
KXPWWMPXNUOYOH
|
6.5 | Ki | 24 | — | |
MVJMMLFMPWITEJ
|
6.5 | Ki | 110 | — | |
OWFLADWRSCINST
|
6.5 | Ki | 30 | — | |
XBAIEEJJCJHBDL
|
6.5 | Ki | 17 | — | |
BPNUQXPIQBZCMR
|
6.4 | Kd | 83 | Yes | |
GEGCXGMFUYJULA
|
6.4 | Ki | 30 | Yes | |
KYACBMRLQMEIAI
|
6.4 | Ki | 30 | — | |
QXRJBJVCBQSLTA
|
6.4 | Ki | 29 | — | |
SQXSMLLCDWJNAC
|
6.4 | Ki | 20 | — | |
XPHWIERLJBFPFV
|
6.4 | Ki | 69 | — | |
YEHCNYAQEBQCCS
|
6.4 | Ki | 74 | — | |
CALAEFSQWBJMDU
|
6.3 | Ki | 21 | — | |
HEUSUIRCBWROMH
|
6.3 | Ki | 64 | — | |
HHSVICUMCOBRPT
|
6.3 | Ki | 33 | — | |
JZTOUVBEZONDKA
|
6.3 | Ki | 80 | — | |
LCKDESRGCHSHHO
|
6.3 | Ki | 18 | — | |
LRESELHEXSUQGE
|
6.3 | Ki | 10 | — | |
PEXKNSGOEOREKM
|
6.3 | Ki | 13 | — | |
SVUIYNKSDCANAY
|
6.3 | Ki | 16 | — | |
KDGFLJKFZUIJMX
|
6.3 | Kd | 10 | — | |
KQWTXAWKBUUOMU
|
6.2 | IC50 | 20 | Yes | |
YYLKKYCXAOBSRM
|
6.2 | Kd | 191 | — | |
FGWOKLCRQJXPPQ
|
6.2 | Ki | 14 | — | |
FLEAYYMORDPWAJ
|
6.2 | Ki | 90 | — | |
FUMCKNCUEAQHCV
|
6.2 | Ki | 103 | — | |
JOIUJUJSHIHBDT
|
6.2 | Ki | 18 | — | |
WINHZLLDWRZWRT
|
6.2 | Ki | 66 | — | |
XYZNKCSDQRKAFR
|
6.2 | Ki | 53 | — | |
YEPNVBNYCRGZRX
|
6.2 | Ki | 26 | — | |
YWTBGJGMTBHQTM
|
6.2 | Ki | 65 | — | |
JKDGKIBAOAFRPJ
|
6.2 | IC50 | 3 | — | |
KDKUVYLMPJIGKA
|
6.1 | Kd | 91 | Yes | |
HKSZLNNOFSGOKW
|
6.1 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
6.1 | Kd | 213 | — | |
BIKYDWLMTPRSQL
|
6.1 | Ki | 50 | — | |
BSFNGHCTZDCQBF
|
6.1 | Ki | 93 | — | |
CTNPALGJUAXMMC
|
6.1 | Kd | 151 | — | |
IHGUHCPMDSTTIW
|
6.1 | Ki | 5 | — | |
MFMXAWQGPQXDRJ
|
6.1 | Ki | 27 | — |