Target Details
| UniProt AC | P78368 |
|---|---|
| Gene Symbol | CSNK1G2 |
| Protein Name | Casein kinase I isoform gamma-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12605 (CK1gamma_C) PF00069 (Pkinase) |
Summary
- Multi-target molecules 121
- Clinical molecules 6
- Avg pChEMBL 6.7
KEGG Pathways (1)
Active Molecules (121)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MUOKSQABCJCOPU
|
8.4 | IC50 | 36 | — | |
RJZDECGDCKOHBV
|
8.4 | Ki | 70 | — | |
SBFPHSVZEXSHTL
|
8.4 | Ki | 62 | — | |
XFWUTMHVDGPWLH
|
8.2 | Ki | 75 | — | |
ZGZVRPRSFXRGCF
|
8.2 | Ki | 76 | — | |
KEEOFKPCOCGLAA
|
8.1 | IC50 | 4 | — | |
UDFDIIVNIYWXDM
|
8.1 | Ki | 74 | — | |
PRPGMEHVPYNUSF
|
7.8 | IC50 | 3 | — | |
RVSKJUNTDGBSSS
|
7.7 | Ki | 25 | — | |
VGNSQEJXQARLLC
|
7.6 | IC50 | 3 | — | |
KOHNRDPXFDZZJF
|
7.6 | Ki | 31 | — | |
RKUKAACYUCUJEE
|
7.6 | Ki | 58 | — | |
FLHJZUQGFPJXRD
|
7.5 | Ki | 12 | — | |
UTFXYGYVDDLJER
|
7.5 | Ki | 36 | — | |
VUVUREKZWANTPW
|
7.5 | IC50 | 4 | — | |
ATBAETXFFCOZOY
|
7.5 | IC50 | 39 | — | |
BIDPCEXNMCKHCG
|
7.5 | IC50 | 3 | — | |
CLEGDJQQHUTCOW
|
7.4 | Ki | 43 | — | |
LXVBELDBJGYFEM
|
7.4 | Ki | 20 | — | |
QAJPIJHWTGPUNZ
|
7.4 | Ki | 37 | — | |
WYOFSHLAFWJJAZ
|
7.4 | IC50 | 3 | — | |
FVNNTRZFDXTUGO
|
7.4 | IC50 | 3 | — | |
DKZYXHCYPUVGAF
|
7.3 | Kd | 112 | — | |
GCBJDOWIQHMCMR
|
7.3 | Ki | 84 | — | |
PVVJMBBQASQRAX
|
7.3 | IC50 | 3 | — | |
SYLTYCLPHHSEIJ
|
7.3 | Ki | 27 | — | |
CIUATZJWGJGLPW
|
7.3 | IC50 | 4 | — | |
KPGMXAQTPURKMK
|
7.3 | IC50 | 3 | — | |
CKVWQORGCCEYHS
|
7.2 | Ki | 50 | — | |
DKXHSOUZPMHNIZ
|
7.2 | Ki | 51 | Yes | |
JJJSCYSPSKBQAX
|
7.2 | Ki | 34 | — | |
NLUPJKQOKWBWFC
|
7.2 | Ki | 69 | — | |
AECVPUDXLSQNOL
|
7.1 | IC50 | 3 | — | |
LYNBNVBMAGDJRW
|
7.1 | Ki | 81 | — | |
NJPWCTYVEJIQBM
|
7.1 | Ki | 72 | — | |
ZCCPLJOKGAACRT
|
7.1 | Kd | 599 | — | |
BGVLELSCIHASRV
|
7.0 | Kd | 11 | — | |
ISEDKXOMRIKZPK
|
7.0 | Ki | 13 | — | |
YMIJUBCSOKSFRU
|
7.0 | Ki | 87 | — | |
XDJCLCLBSGGNKS
|
7.0 | Kd | 21 | — | |
WINHZLLDWRZWRT
|
7.0 | Kd | 201 | Yes | |
AOBLBPWPSKBHSI
|
6.9 | Ki | 55 | — | |
CHTMRWQLNNRRFJ
|
6.9 | Ki | 70 | — | |
KNGBZHZRBXFQLV
|
6.8 | IC50 | 3 | — | |
ADMFLILDQJSEIK
|
6.8 | Ki | 72 | — | |
UMTWTCVTRDYHQQ
|
6.8 | Ki | 56 | — | |
XCHWBXBDZRJVDP
|
6.8 | Ki | 51 | — | |
XJJYJNMNYDNXNO
|
6.8 | Ki | 23 | — | |
GMIKNOQZLHKCFH
|
6.7 | IC50 | 3 | — | |
IMHKMKWSWHFKTM
|
6.7 | Ki | 13 | — |