Target Details
| UniProt AC | P78334 |
|---|---|
| Gene Symbol | GABRE |
| Protein Name | Gamma-aminobutyric acid receptor subunit epsilon |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 325
- Clinical molecules 0
- Avg pChEMBL 7.41
KEGG Pathways (7)
Active Molecules (325)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WQIWYEISPHMPOA
|
6.2 | IC50 | 16 | — | |
ARCJBXYEOMXBSZ
|
6.2 | IC50 | 16 | — | |
CTPREUOHTKHCHT
|
6.2 | IC50 | 16 | — | |
XFUAEWGHLXLENC
|
6.2 | IC50 | 16 | — | |
BSEVRQDRIQMBCV
|
6.2 | IC50 | 16 | — | |
DHEXTYZLLGWEFS
|
6.2 | Ki | 16 | — | |
HBOSSQBJUBOEJN
|
6.1 | Ki | 16 | — | |
XVFJUDUNNHPHLN
|
6.1 | IC50 | 16 | — | |
HYJUIJYNZHZBOK
|
6.1 | IC50 | 16 | — | |
WJEPRNMCEBRSDB
|
6.1 | IC50 | 16 | — | |
YLZBNNDOEUIHFB
|
6.1 | IC50 | 16 | — | |
LKUSWPRPRBXYPH
|
6.1 | IC50 | 16 | — | |
VKMJGKFQKLVODR
|
6.1 | IC50 | 16 | — | |
VAEZVMCCCWEXEH
|
6.1 | Ki | 16 | — | |
ZXYMHGABHZSFOI
|
6.1 | Ki | 16 | — | |
DOOGDICMBOTQOZ
|
6.1 | IC50 | 16 | — | |
SLNCMJYPLFSUGO
|
6.0 | Ki | 16 | — | |
SZHSENNQOQSFEA
|
6.0 | IC50 | 16 | — | |
DHLJRIFIBJGWBS
|
6.0 | IC50 | 16 | — | |
DQDLJDCSJFQOHI
|
6.0 | IC50 | 16 | — | |
FUULVCWWUPGUMY
|
6.0 | IC50 | 16 | — | |
GCTOZKWOFVUEAW
|
6.0 | IC50 | 16 | — | |
IHFBPDAQLQOCBX
|
6.0 | Ki | 18 | — | |
KVZVPZYFPDOIMI
|
6.0 | IC50 | 16 | — | |
RYFIWEJRWHTFBM
|
6.0 | IC50 | 16 | — |