Target Details
UniProt ACP78334
Gene SymbolGABRE
Protein NameGamma-aminobutyric acid receptor subunit epsilon
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 325
  • Clinical molecules 0
  • Avg pChEMBL 7.41
Top Co-occurrence Targets
Active Molecules (325)
InChIKey pChEMBL Type Targets Clinical
QJCQEAQHBMKTCT 7.5 IC50 16
DOKJHXYCSUQRQV 7.4 Ki 16
JGVCISSLGASTTA 7.4 Ki 18
GCSRDJACUSRHBX 7.4 Ki 16
CMVZUGQWJUPOJA 7.4 IC50 16
QMHTYKLXSOQULX 7.4 Ki 16
DUZTVXKYJROMJJ 7.4 IC50 16
BMIKDIWICOAHJN 7.4 Ki 16
MSFAMEBSEKIVDI 7.4 Ki 16
VUZAUNZSDCMUTH 7.4 Ki 16
LDBHRENGPXWKOD 7.3 IC50 16
GWCQPEHFUKZODL 7.3 Ki 16
QYEIQYJLVREYBI 7.3 IC50 16
SIBRGSBVGDWJAF 7.3 IC50 16
WHGIBMIKSVYLCR 7.3 IC50 16
AURFZBICLPNKBZ 7.3 IC50 16
DGZYPGWWTKGBQP 7.3 Ki 16
NTZNKZHCQIJCPO 7.3 IC50 16
SNEWVMXJSABDSK 7.3 Ki 16
VWCCHJFFYCGXFL 7.3 Ki 16
JBDRNSFDKSBSFE 7.3 Ki 16
NNHRCSJWUBQYQV 7.3 IC50 16
PISRVNOAPOPQHJ 7.3 Ki 18
KRVDMABBKYMBHG 7.3 Ki 16
VOZOMZWSLGQRKP 7.3 IC50 16
XEJHLKHWRSNEOC 7.3 IC50 16
UEWSJGMYAPQKKT 7.2 Ki 16
URMNROOZTOLUHQ 7.2 Ki 16
PWOQCZLPANHRRJ 7.2 Ki 16
NKSQLOHZBFUKLF 7.2 IC50 16
PRUQRKPURHYKRP 7.2 Ki 16
VAVBWHIBLOPOEM 7.2 Ki 16
IOOGUHXPDYRXFJ 7.2 IC50 16
WCYJVRQPVHPWLQ 7.2 Ki 16
WHEUGJHMVJCNEP 7.2 IC50 16
SINAJPKUKOSXOT 7.2 IC50 16
LPOZDKMXSPAATL 7.2 Ki 16
VOZOMZWSLGQRKP 7.1 IC50 16
YBRXFNLNMSTVNQ 7.1 IC50 16
HRTSOMLTEJFUCO 7.1 IC50 16
PGTVWKLGGCQMBR 7.1 IC50 16
OMQHFPMEAPEGTA 7.1 Ki 16
AEYRTFCCYIWUJJ 7.1 Ki 16
NFXAWQDTYKJJTD 7.1 IC50 16
JSRKYARWMIOKOB 7.0 Ki 16
LWLYOXPDYPYNHH 7.0 IC50 16
SZSNAHWJFCIUBV 7.0 IC50 17
WUNJCJOCGLXHNU 7.0 IC50 16
GSNCQRDETZIWAE 7.0 Ki 16
KWHWSXISOMCUPZ 7.0 IC50 16
2D structure