Target Details
| UniProt AC | P78334 |
|---|---|
| Gene Symbol | GABRE |
| Protein Name | Gamma-aminobutyric acid receptor subunit epsilon |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 325
- Clinical molecules 0
- Avg pChEMBL 7.41
KEGG Pathways (7)
Active Molecules (325)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MZFKWSFOAVBLQM
|
9.8 | IC50 | 16 | — | |
WFPXOWCKXUEKCA
|
9.7 | IC50 | 16 | — | |
KVKWRJDNIJTMGN
|
9.6 | IC50 | 16 | — | |
QUUNMICPMYIHFS
|
9.4 | IC50 | 16 | — | |
VMDUABMKBUKKPG
|
9.4 | IC50 | 16 | — | |
XKENJWNGLCKOBP
|
9.3 | IC50 | 16 | — | |
NJUMMJUUDUYSKB
|
9.3 | IC50 | 16 | — | |
ALBKMJDFBZVHAK
|
9.3 | IC50 | 16 | — | |
BYMDBFGHCDTBMT
|
9.3 | IC50 | 16 | — | |
IUHKSTINHDUYRO
|
9.3 | IC50 | 16 | — | |
VJVAWKPXJCDEQG
|
9.3 | IC50 | 16 | — | |
WRXDVVALWQGPMW
|
9.3 | IC50 | 16 | — | |
BLJPKQXXDFIIFR
|
9.2 | IC50 | 16 | — | |
XJMIBNLJFYSGAR
|
9.2 | IC50 | 16 | — | |
JFGUJXZLJIUVPZ
|
9.1 | IC50 | 16 | — | |
LYFROTHEKIFZAU
|
9.1 | IC50 | 16 | — | |
RYIVVNHBYBYXHF
|
9.1 | IC50 | 16 | — | |
VZKRZUPJCVFVGR
|
9.1 | IC50 | 16 | — | |
DGBIGWXXNGSACT
|
9.1 | Ki | 16 | — | |
OFBIFZUFASYYRE
|
9.1 | Ki | 16 | — | |
YJZGQBGGTBIAOP
|
9.1 | IC50 | 16 | — | |
AQKFCEWRKDXGMK
|
9.0 | Ki | 16 | — | |
FVFFDKKTXYVCCW
|
9.0 | IC50 | 16 | — | |
IPHSQMSRIWZULE
|
9.0 | Ki | 16 | — | |
KDMMIKQMHNBKAV
|
9.0 | Ki | 17 | — | |
KOVRZNUMIKACTB
|
9.0 | IC50 | 17 | — | |
RLFKILXOLJVUNF
|
9.0 | IC50 | 16 | — | |
WGRVAGIQTHEEQW
|
9.0 | IC50 | 16 | — | |
BSBLYLUAUVTSMM
|
9.0 | IC50 | 16 | — | |
OJLYUGSSUKAWJC
|
8.8 | Ki | 16 | — | |
KVKYGVOAHGNAKZ
|
8.7 | IC50 | 16 | — | |
QTEUJQNPMLXVLL
|
8.7 | IC50 | 16 | — | |
UKHFPVCOXBJPIN
|
8.7 | IC50 | 17 | — | |
ZOCSXAVNDGMNBV
|
8.6 | IC50 | 16 | — | |
CHIFCDOIPRCHCF
|
8.6 | IC50 | 16 | — | |
CHQPOBHNDRMXFK
|
8.6 | Ki | 18 | — | |
KVKYGVOAHGNAKZ
|
8.5 | IC50 | 17 | — | |
LENHHZQGSWCZJW
|
8.5 | Ki | 16 | — | |
LPAODQAWVMEXKR
|
8.5 | IC50 | 16 | — | |
NEOUOHDNZDRDNJ
|
8.5 | IC50 | 16 | — | |
QIZPCEVRKTWHIE
|
8.5 | IC50 | 16 | — | |
RYLDZJANGRBUGW
|
8.5 | IC50 | 16 | — | |
MVBVNOZDVRVMNH
|
8.4 | IC50 | 16 | — | |
ACUNYYFYYWOKOD
|
8.4 | IC50 | 16 | — | |
AXPGZURVLRWNBR
|
8.4 | Ki | 16 | — | |
BZVWONIGXAYZIT
|
8.4 | IC50 | 16 | — | |
CDWXZILKRXSANI
|
8.4 | IC50 | 16 | — | |
DYSDYZCGZCYPCT
|
8.4 | IC50 | 16 | — | |
JTYYMOMTGZSRFM
|
8.4 | IC50 | 16 | — | |
LMXUGQJMQSMLIQ
|
8.4 | Ki | 17 | — |