Target Details
| UniProt AC | P78325 |
|---|---|
| Gene Symbol | ADAM8 |
| Protein Name | Disintegrin and metalloproteinase domain-containing protein 8 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08516 (ADAM_CR) PF00200 (Disintegrin) PF01562 (Pep_M12B_propep) PF01421 (Reprolysin) |
Summary
- Multi-target molecules 5
- Clinical molecules 1
- Avg pChEMBL 6.76
Active Molecules (5)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QTXVPJOTKLUYMQ
|
7.4 | IC50 | 5 | — | |
JQLHAXGMYALIFJ
|
7.4 | IC50 | 3 | — | |
LJOOWNHZCTUDSG
|
6.8 | IC50 | 3 | — | |
JSVQSOCCWRHOES
|
6.2 | IC50 | 3 | — | |
CKZHFOKQZRZCPF
|
6.0 | IC50 | 9 | Yes |