Target Details
| UniProt AC | P68400 |
|---|---|
| Gene Symbol | CSNK2A1 |
| Protein Name | Casein kinase II subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 639
- Clinical molecules 14
- Avg pChEMBL 7.48
KEGG Pathways (10)
Associated Diseases (1)
Active Molecules (639)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HNIDDGUBRPIXPG
|
6.3 | IC50 | 7 | — | |
AEBNGBBFOVOYDE
|
6.3 | IC50 | 2 | — | |
LEZMJYDNPSKPIL
|
6.3 | IC50 | 2 | — | |
RNIUZVHLSOCFGG
|
6.3 | IC50 | 2 | — | |
XHMVESPALKGSNL
|
6.3 | IC50 | 2 | — | |
CUBDXJALAMZYLD
|
6.2 | Kd | 4 | — | |
JLSRVJYBKQUFNV
|
6.2 | IC50 | 2 | — | |
KSEBMYQBYZTDHS
|
6.2 | IC50 | 7 | Yes | |
NDJDFASWUZEZMI
|
6.2 | IC50 | 4 | — | |
AIJJYTXSVJFNGP
|
6.2 | IC50 | 2 | — | |
HUECFCSRZKSRJF
|
6.2 | IC50 | 3 | — | |
QXMXIHBLICGPMG
|
6.2 | IC50 | 9 | — | |
AXZCENIZJLHNSM
|
6.2 | IC50 | 4 | — | |
OARXLGLBMAHALM
|
6.2 | IC50 | 12 | Yes | |
UUXDJIVNVOOKFQ
|
6.2 | IC50 | 9 | — | |
ZQVAOVVVPPUILG
|
6.2 | Ki | 4 | — | |
BNLPAUPVSCPTDM
|
6.2 | Ki | 15 | — | |
CPGKMMMSMJKHDL
|
6.2 | Ki | 16 | — | |
ILHPOUBFADFYIT
|
6.2 | Ki | 2 | — | |
OWFLADWRSCINST
|
6.2 | Ki | 30 | — | |
WHVFDYQCAMPLMS
|
6.2 | Ki | 20 | Yes | |
ZVWRFVCNQOECJS
|
6.2 | Ki | 71 | — | |
ACPOUJIDANTYHO
|
6.2 | IC50 | 17 | Yes | |
LOSMIMWNQPCHQW
|
6.2 | IC50 | 3 | — | |
SABLEOBBNNRHAD
|
6.2 | IC50 | 6 | — | |
XJONKSWKTASLQP
|
6.2 | IC50 | 3 | — | |
DTBFDAJNODVUMF
|
6.2 | IC50 | 4 | — | |
UBLIGMBRLOJZPG
|
6.2 | IC50 | 4 | — | |
WNDNHVKGAOSTKP
|
6.2 | IC50 | 3 | — | |
LZJRNLRASBVRRX
|
6.2 | IC50 | 6 | — | |
QHPKKGUGRGRSGA
|
6.1 | IC50 | 7 | Yes | |
WIMPWBKZHKEQQS
|
6.1 | Ki | 2 | — | |
FZIXDSBXXBDCIU
|
6.1 | IC50 | 4 | — | |
TZVUFJMGSMRSMC
|
6.1 | IC50 | 4 | — | |
ULYNWOFGCTVEMP
|
6.1 | IC50 | 2 | — | |
XVDZCNRRNDWVCH
|
6.1 | IC50 | 3 | — | |
AHJRHEGDXFFMBM
|
6.1 | Kd | 28 | — | |
KZNIFHPLKGYRTM
|
6.1 | IC50 | 21 | Yes | |
LGRJHSGKEBRDHI
|
6.1 | IC50 | 4 | — | |
MEKFXUFACKZUCV
|
6.1 | IC50 | 9 | — | |
ONHQPZWMSNCSPQ
|
6.1 | IC50 | 4 | — | |
YKDZIFFKQUNVHH
|
6.1 | IC50 | 3 | — | |
FJZXDUKUMALHNP
|
6.1 | Ki | 10 | — | |
HVXHDYSWCHQWBD
|
6.1 | IC50 | 3 | — | |
IRDNLBJYBJGZKE
|
6.1 | IC50 | 3 | — | |
IUEBPIPDFMCSTP
|
6.1 | Ki | 29 | — | |
JJJSCYSPSKBQAX
|
6.1 | Ki | 34 | — | |
KRXQWLCJHMDEDM
|
6.1 | IC50 | 8 | — | |
KTFLFGFPJQSPNR
|
6.1 | IC50 | 3 | — | |
OADRBDVURCEKRP
|
6.1 | Ki | 44 | — |