Target Details
| UniProt AC | P68366 |
|---|---|
| Gene Symbol | TUBA4A |
| Protein Name | Tubulin alpha-4A chain |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00091 (Tubulin) PF03953 (Tubulin_C) |
Summary
- Multi-target molecules 268
- Clinical molecules 0
- Avg pChEMBL 6.46
KEGG Pathways (14)
Associated Diseases (4)
Active Molecules (268)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WYRFZTFZPZDGIF
|
10.3 | IC50 | 16 | — | |
ICROQBNUKGSVGS
|
9.8 | IC50 | 16 | — | |
DFWBYSXAPDBNKH
|
8.9 | IC50 | 15 | — | |
OFDNQWIFNXBECV
|
8.9 | IC50 | 15 | — | |
BANKOOHMAFMTES
|
8.8 | IC50 | 15 | — | |
YRMXYQDFDXFFPU
|
8.6 | IC50 | 15 | — | |
HPKIQGFGVRGFRW
|
8.5 | Kd | 15 | — | |
QXRSDHAAWVKZLJ
|
8.5 | IC50 | 15 | — | |
MAYJVBBZJLABTA
|
8.4 | IC50 | 15 | — | |
CNGKIRSNRQSORA
|
8.2 | IC50 | 15 | — | |
YOJHPSLHBFFDDL
|
8.0 | IC50 | 19 | — | |
MJQIGYITZDMOHL
|
8.0 | IC50 | 15 | — | |
NUYWEXUUHJLAPJ
|
8.0 | Ki | 15 | — | |
MQYZCKOGTWYJAZ
|
8.0 | Kd | 15 | — | |
ZCCPLJOKGAACRT
|
7.9 | Kd | 599 | — | |
WKPWGQKGSOKKOO
|
7.8 | Kd | 15 | — | |
GBABOYUKABKIAF
|
7.8 | IC50 | 17 | — | |
DFHHLNDKKOTNGJ
|
7.7 | IC50 | 15 | — | |
FKVVWNAJLKZIHY
|
7.7 | Kd | 15 | — | |
KTZONPJUXCHDGO
|
7.7 | Ki | 15 | — | |
QHXOKFICRLZQNX
|
7.7 | IC50 | 17 | — | |
XIHGDBYGUWEHCV
|
7.6 | IC50 | 8 | — | |
ZGHAKJYOYPNCDO
|
7.5 | IC50 | 15 | — | |
LSXOBYNBRKOTIQ
|
7.3 | Kd | 15 | — | |
NKNUEBKXJIQFBJ
|
7.3 | Ki | 15 | — | |
OOYWFPLKWZVWFR
|
7.3 | Kd | 15 | — | |
JBZVXYXXVXMBHM
|
7.2 | Ki | 15 | — | |
GTNIINDRYIDZEJ
|
7.2 | IC50 | 15 | — | |
ZVVCUVYHNAOYCY
|
7.1 | IC50 | 15 | — | |
HUNUMKDNWUBRDX
|
7.1 | IC50 | 15 | — | |
HUNUMKDNWUBRDX
|
7.0 | IC50 | 15 | — | |
ISALLVOZADSZHM
|
7.0 | Ki | 15 | — | |
QATWEQGSTKHUFM
|
7.0 | IC50 | 15 | — | |
QATWEQGSTKHUFM
|
7.0 | IC50 | 15 | — | |
KEEGEWFDKNKLJX
|
7.0 | IC50 | 15 | — | |
ACOOGNWCLUIBMF
|
7.0 | IC50 | 16 | — | |
WURUPVNQTCOGJC
|
7.0 | IC50 | 15 | — | |
FFTSFVUSBPOJKD
|
7.0 | IC50 | 16 | — | |
AYSXURJZVXBSRV
|
6.9 | IC50 | 16 | — | |
JXLYSJRDGCGARV
|
6.9 | IC50 | 17 | — | |
HGVNKQONHGKNOE
|
6.9 | Kd | 15 | — | |
XINWQRHEYTZCMW
|
6.8 | IC50 | 15 | — | |
JXLYSJRDGCGARV
|
6.8 | IC50 | 15 | — | |
YWUJMYGISLHKRO
|
6.8 | Ki | 15 | — | |
AAAQFGUYHFJNHI
|
6.8 | IC50 | 252 | — | |
UIIQTKRZMOZGAC
|
6.8 | IC50 | 15 | — | |
NNMNQNZESDQXQW
|
6.8 | IC50 | 15 | — | |
AWUKPUYMLOLFIE
|
6.7 | IC50 | 15 | — | |
IAKHMKGGTNLKSZ
|
6.7 | IC50 | 16 | — | |
HUNUMKDNWUBRDX
|
6.7 | IC50 | 15 | — |