Target Details
| UniProt AC | P63000 |
|---|---|
| Gene Symbol | RAC1 |
| Protein Name | Ras-related C3 botulinum toxin substrate 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00071 (Ras) |
Summary
- Multi-target molecules 3
- Clinical molecules 0
- Avg pChEMBL 6.78
KEGG Pathways (56)
- AGE-RAGE signaling pathway in diabetic complications
- Adherens junction
- Amyotrophic lateral sclerosis
- Axon guidance
- B cell receptor signaling pathway
- Bacterial invasion of epithelial cells
- Cadherin signaling
- Chemical carcinogenesis - reactive oxygen species
- Chemokine signaling pathway
- Choline metabolism in cancer
- Colorectal cancer
- Diabetic cardiomyopathy
- Efferocytosis
- Epithelial cell signaling in Helicobacter pylori infection
- Epstein-Barr virus infection
- Fc epsilon RI signaling pathway
- Fc gamma R-mediated phagocytosis
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- IgSF CAM signaling
- Integrin signaling
- Kaposi sarcoma-associated herpesvirus infection
- Leukocyte transendothelial migration
- Lipid and atherosclerosis
- MAPK signaling pathway
- Natural killer cell mediated cytotoxicity
- Neurotrophin signaling pathway
- Neutrophil extracellular trap formation
- Non-alcoholic fatty liver disease
- Osteoclast differentiation
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pancreatic secretion
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Phagosome
- Prion disease
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Renal cell carcinoma
- Salmonella infection
- Shigellosis
- Sphingolipid signaling pathway
- Tight junction
- Toll-like receptor signaling pathway
- VEGF signaling pathway
- Viral carcinogenesis
- Viral myocarditis
- Wnt signaling pathway
- Yersinia infection
- cAMP signaling pathway
Associated Diseases (1)
Active Molecules (3)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MIDUFIRTIFUTQA
|
7.3 | Kd | 3 | — | |
LJCANTASZGYJLG
|
7.0 | IC50 | 4 | — | |
OZWKMVRBQXNZKK
|
6.0 | IC50 | 2 | — |