Target Details
| UniProt AC | P62593 |
|---|---|
| Gene Symbol | bla |
| Protein Name | Beta-lactamase TEM |
| Organism | Escherichia coli |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF13354 (Beta-lactamase2) |
Summary
- Multi-target molecules 106
- Clinical molecules 0
- Avg pChEMBL 7.66
Top Co-occurrence Targets
- ampC 51 shared
- ampC 44 shared
- OXA-48 34 shared
- ccrA 34 shared
- nmcA 12 shared
- blaZ 9 shared
- imiA 4 shared
- OXA-1 2 shared
- blaCTX-M-9a 1 shared
- blaCTX-M-14 1 shared
Active Molecules (106)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AVPVJZPIBNHZQN
|
6.2 | IC50 | 2 | — | |
UAILHDKDBBFHDN
|
6.1 | IC50 | 3 | — | |
XSJFKEVFSPGNJZ
|
6.1 | IC50 | 3 | — | |
ITFVZKLBKASFHP
|
6.1 | IC50 | 3 | — | |
SUKFPPMYJISQEB
|
6.1 | IC50 | 2 | — | |
NHCGBXGSGNHZFN
|
6.0 | IC50 | 2 | — |