Target Details
| UniProt AC | P62593 |
|---|---|
| Gene Symbol | bla |
| Protein Name | Beta-lactamase TEM |
| Organism | Escherichia coli |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF13354 (Beta-lactamase2) |
Summary
- Multi-target molecules 106
- Clinical molecules 0
- Avg pChEMBL 7.66
Top Co-occurrence Targets
- ampC 51 shared
- ampC 44 shared
- OXA-48 34 shared
- ccrA 34 shared
- nmcA 12 shared
- blaZ 9 shared
- imiA 4 shared
- OXA-1 2 shared
- blaCTX-M-9a 1 shared
- blaCTX-M-14 1 shared
Active Molecules (106)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QEYQIONWPOMBON
|
7.7 | IC50 | 2 | — | |
YHANUKIZKPOWPW
|
7.6 | IC50 | 3 | — | |
ZEICLMMMMGQHIK
|
7.6 | IC50 | 3 | — | |
CZCMDCKIUIXEQC
|
7.6 | IC50 | 3 | — | |
OPBQWQXRAFJUEL
|
7.6 | IC50 | 3 | — | |
YNCYPMUJDDXIRH
|
7.6 | Ki | 3 | — | |
ZZWPJCNMJSBJDZ
|
7.5 | IC50 | 2 | — | |
FCBUHCWXTMAQGJ
|
7.5 | IC50 | 3 | — | |
BVKNUAKQEQUMSY
|
7.5 | IC50 | 3 | — | |
HTXPDRHSGPNWKA
|
7.5 | IC50 | 2 | — | |
WOFAABWEQYFPBT
|
7.4 | IC50 | 3 | — | |
VDZDNZXKYYQECM
|
7.4 | IC50 | 2 | — | |
SIVNUZUWNGEGKW
|
7.4 | IC50 | 3 | — | |
BLOSWWBHNLGJRP
|
7.3 | IC50 | 3 | — | |
WVZOCYGRXONJLX
|
7.3 | IC50 | 3 | — | |
FXRXKUVQNAIPQC
|
7.3 | IC50 | 3 | — | |
ACQFJWSLWQLLIA
|
7.3 | IC50 | 2 | — | |
KYVATCVZAZHVGK
|
7.2 | IC50 | 2 | — | |
YFHXDSIOXRFREU
|
7.2 | IC50 | 3 | — | |
HZZVJAQRINQKSD
|
7.2 | IC50 | 2 | — | |
LPQZKKCYTLCDGQ
|
7.2 | IC50 | 4 | — | |
RFMIKMMOLPNEDG
|
7.2 | IC50 | 3 | — | |
FQSPFOVCHGZCIK
|
7.2 | IC50 | 2 | — | |
HLBYYYVPQDVZIQ
|
7.2 | IC50 | 2 | — | |
HLBYYYVPQDVZIQ
|
7.2 | IC50 | 2 | — | |
VRAFEQHIWHNGLC
|
7.2 | IC50 | 3 | — | |
XSDSQTYLBBGLJR
|
7.1 | IC50 | 2 | — | |
XSDSQTYLBBGLJR
|
7.1 | IC50 | 2 | — | |
NZNHTQCXWOAKDT
|
7.1 | IC50 | 2 | — | |
FCBPOMQVJRBNEN
|
7.1 | IC50 | 3 | — | |
SFPTWFMBZJRMKD
|
7.1 | IC50 | 3 | — | |
ABPLMHATNQPHNC
|
7.1 | IC50 | 3 | — | |
OOBLDYJFUBJOPF
|
7.1 | IC50 | 3 | — | |
STUCJEURXSAYOH
|
7.0 | IC50 | 2 | — | |
WYRIPYFYOUAORN
|
7.0 | IC50 | 3 | — | |
QEEMJZXDEIFDDR
|
7.0 | IC50 | 3 | — | |
WCRPDOYIEXPPSD
|
7.0 | IC50 | 3 | — | |
BFVDGHQWCMHZCR
|
6.9 | IC50 | 2 | — | |
JYGFUXUBGZBBAC
|
6.9 | IC50 | 5 | — | |
DIRLPWJRIWGPCS
|
6.8 | IC50 | 3 | — | |
TYGMQYXAGAWAHU
|
6.8 | IC50 | 2 | — | |
SFPTWFMBZJRMKD
|
6.7 | IC50 | 3 | — | |
SWIHLLNXGOJYRM
|
6.7 | IC50 | 3 | — | |
SOQURWNDDXDSTI
|
6.6 | IC50 | 2 | — | |
XUUNBOUAUWVPDD
|
6.6 | IC50 | 2 | — | |
KMIMTPSCZSJCPM
|
6.5 | IC50 | 3 | — | |
CBBUHGXUJWGHRX
|
6.5 | IC50 | 3 | — | |
LTSHHIPSCFMNJJ
|
6.5 | IC50 | 2 | — | |
RUDGJWAKUPBPKU
|
6.4 | IC50 | 2 | — | |
XXDOEORVWMNHIY
|
6.2 | IC50 | 3 | — |