Target Details
| UniProt AC | P62508 |
|---|---|
| Gene Symbol | ESRRG |
| Protein Name | Estrogen-related receptor gamma |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 45
- Clinical molecules 2
- Avg pChEMBL 7.1
Active Molecules (45)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IISBACLAFKSPIT
|
8.3 | IC50 | 3 | — | |
ZTAZBLSYCOAIDZ
|
8.0 | IC50 | 2 | — | |
TXUZVZSFRXZGTL
|
7.9 | IC50 | 6 | — | |
OIUCUUXSMIJSEB
|
7.9 | IC50 | 2 | — | |
TXUZVZSFRXZGTL
|
7.9 | IC50 | 7 | Yes | |
ZUSXRJKXJTTXKD
|
7.6 | IC50 | 2 | — | |
ZUSXRJKXJTTXKD
|
7.6 | IC50 | 2 | — | |
ZUSXRJKXJTTXKD
|
7.5 | IC50 | 2 | — | |
BGMSYZADXHOOKI
|
7.5 | IC50 | 3 | — | |
BGMSYZADXHOOKI
|
7.5 | IC50 | 3 | — | |
ZUSXRJKXJTTXKD
|
7.5 | IC50 | 2 | — | |
ZUSXRJKXJTTXKD
|
7.5 | IC50 | 2 | — | |
SYZJGNRKRGPMOF
|
7.3 | IC50 | 2 | — | |
FACDVWBDBZWZTA
|
7.3 | IC50 | 2 | — | |
QVQADUPEEMYSFQ
|
7.2 | IC50 | 2 | — | |
NKANXQFJJICGDU
|
7.2 | IC50 | 35 | Yes | |
QLISPFNKBMBCQJ
|
7.2 | IC50 | 2 | — | |
QLISPFNKBMBCQJ
|
7.2 | IC50 | 2 | — | |
SDVZGUZPOXADLQ
|
7.2 | IC50 | 2 | — | |
BAVCXZJGGIUPCK
|
7.1 | IC50 | 2 | — | |
BAVCXZJGGIUPCK
|
7.1 | IC50 | 2 | — | |
YAZOPMJURQIDRH
|
7.1 | IC50 | 2 | — | |
SYZJGNRKRGPMOF
|
7.1 | IC50 | 2 | — | |
UTNLGSPOQMFYKD
|
7.1 | IC50 | 2 | — | |
UTNLGSPOQMFYKD
|
7.1 | IC50 | 2 | — | |
UTNLGSPOQMFYKD
|
7.1 | IC50 | 2 | — | |
QMJDQQMIKSBOSP
|
7.0 | IC50 | 2 | — | |
UFPFMVPHDSUBQY
|
7.0 | IC50 | 2 | — | |
ZVSFNBNLNLXEFQ
|
7.0 | IC50 | 2 | — | |
ZJWVUIDDICJVDQ
|
6.9 | IC50 | 2 | — | |
ZJWVUIDDICJVDQ
|
6.9 | IC50 | 2 | — | |
NJYHQVPRPYSYGP
|
6.9 | IC50 | 2 | — | |
BYOHHOLODBNIMD
|
6.8 | IC50 | 2 | — | |
BYOHHOLODBNIMD
|
6.8 | IC50 | 2 | — | |
LSXNUCOYUCKQNA
|
6.8 | IC50 | 2 | — | |
LSXNUCOYUCKQNA
|
6.8 | IC50 | 2 | — | |
HZWPCGJKFLEGFZ
|
6.7 | IC50 | 2 | — | |
MZLLOCKOYWOFPI
|
6.6 | IC50 | 2 | — | |
RDGFLUWTBBDQBO
|
6.6 | IC50 | 2 | — | |
RDGFLUWTBBDQBO
|
6.6 | IC50 | 2 | — | |
QJKDTGBJOBJWGU
|
6.5 | IC50 | 2 | — | |
YXZWFFNGLDURRL
|
6.5 | IC50 | 2 | — | |
KRPGZUBOFAMQPA
|
6.1 | IC50 | 2 | — | |
KOKFDHHICYICJW
|
6.0 | IC50 | 2 | — | |
UCXOFWMSZIFPGX
|
6.0 | IC50 | 2 | — |