Target Details
| UniProt AC | P62343 |
|---|---|
| Gene Symbol | CDPK1 |
| Protein Name | Calcium-dependent protein kinase 1 |
| Organism | Plasmodium falciparum (isolate K1 / Thailand) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF13499 (EF-hand_7) PF00069 (Pkinase) |
Summary
- Multi-target molecules 15
- Clinical molecules 10
- Avg pChEMBL 6.84
Active Molecules (15)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YZDJQTHVDDOVHR
|
8.8 | Kd | 23 | — | |
UIARLYUEJFELEN
|
8.2 | Kd | 289 | Yes | |
ODPGGGTTYSGTGO
|
8.1 | Kd | 153 | — | |
BBRVCZSXNXYZKS
|
7.4 | Ki | 2 | — | |
ZDESNDWWUUVJLG
|
7.3 | Kd | 6 | — | |
MLDQJTXFUGDVEO
|
6.7 | Kd | 85 | Yes | |
SEJGTFPOEJWEGG
|
6.6 | Kd | 149 | — | |
CUIHSIWYWATEQL
|
6.4 | Kd | 61 | Yes | |
MFAQYJIYDMLAIM
|
6.3 | Kd | 130 | Yes | |
PIQCTGMSNWUMAF
|
6.2 | Kd | 137 | Yes | |
ZBNZXTGUTAYRHI
|
6.2 | Kd | 102 | Yes | |
QQWUGDVOUVUTOY
|
6.2 | Kd | 231 | Yes | |
HHZIURLSWUIHRB
|
6.1 | Kd | 57 | Yes | |
CDMGBJANTYXAIV
|
6.1 | Kd | 34 | Yes | |
BMGQWWVMWDBQGC
|
6.0 | Kd | 147 | Yes |