Target Details
| UniProt AC | P61073 |
|---|---|
| Gene Symbol | CXCR4 |
| Protein Name | C-X-C chemokine receptor type 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) PF12109 (CXCR4_N) |
Summary
- Multi-target molecules 57
- Clinical molecules 0
- Avg pChEMBL 7.21
KEGG Pathways (14)
- Axon guidance
- Calcium signaling pathway
- Chemokine signaling pathway
- Cytokine-cytokine receptor interaction
- Endocytosis
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Intestinal immune network for IgA production
- Leukocyte transendothelial migration
- Pathways in cancer
- Regulation of actin cytoskeleton
- Viral life cycle - HIV-1
- Viral protein interaction with cytokine and cytokine receptor
- Virion - Human immunodeficiency virus
Associated Diseases (1)
Active Molecules (57)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LGEIHKKMICVKAE
|
8.7 | IC50 | 2 | — | |
QUDMHFVRKBVGBY
|
8.6 | IC50 | 3 | — | |
KVZDMWMWTDNKDM
|
8.4 | IC50 | 2 | — | |
ZKWKKAVOVBLNQA
|
8.2 | IC50 | 2 | — | |
BASXCEHVMKEGCB
|
8.1 | IC50 | 2 | — | |
VUXQRANDPGSPRS
|
8.0 | IC50 | 3 | — | |
ZWRNWGSOEVSTSJ
|
7.8 | IC50 | 2 | — | |
YPLCBNLGVGQEFT
|
7.8 | IC50 | 2 | — | |
HAKFGEFAVSVPJO
|
7.7 | IC50 | 2 | — | |
MWUZFFWTKOGEKF
|
7.7 | IC50 | 2 | — | |
ALNLTEGQXKHFSE
|
7.6 | IC50 | 2 | — | |
OWWQLCCEAAGOJW
|
7.6 | IC50 | 2 | — | |
MYCKNKHATQGHEV
|
7.6 | IC50 | 2 | — | |
KDSKMOVNVSMORM
|
7.5 | IC50 | 2 | — | |
VUKMAAVKUIIBCS
|
7.5 | IC50 | 3 | — | |
RKAMQPGAELEERO
|
7.5 | IC50 | 2 | — | |
SBWDNXAOTCMVAA
|
7.5 | IC50 | 7 | — | |
HSCURGZCDKRUEI
|
7.4 | IC50 | 3 | — | |
OOSUDWRRWZVFEB
|
7.4 | IC50 | 2 | — | |
VUKMAAVKUIIBCS
|
7.4 | IC50 | 2 | — | |
RLDXRZALYBNDPT
|
7.3 | IC50 | 2 | — | |
WDRULORDXYZPQS
|
7.3 | IC50 | 2 | — | |
KCTNGNPVURILGU
|
7.3 | Ki | 2 | — | |
ISYILQOWKQBKJP
|
7.3 | IC50 | 2 | — | |
KKUZNBPYLQBJGJ
|
7.2 | IC50 | 2 | — | |
LMTVSDLVMVDXEP
|
7.2 | IC50 | 3 | — | |
DZNHRLXBJDORJM
|
7.2 | IC50 | 3 | — | |
VMUZNUDUOJPDTC
|
7.2 | IC50 | 2 | — | |
YPWOVOYHSYFRRC
|
7.2 | IC50 | 2 | — | |
AEOPBRLVLXDVLL
|
7.1 | IC50 | 2 | — | |
ONNXLKVJJQMNHD
|
7.1 | IC50 | 2 | — | |
MLQQKXMYXPIYTH
|
7.1 | IC50 | 2 | — | |
UOJYAHYPXYXUMQ
|
7.1 | IC50 | 2 | — | |
PZYIAIVLQMGYOR
|
7.1 | IC50 | 3 | — | |
DBUIDMKLHBXFJG
|
7.0 | IC50 | 2 | — | |
REMRQQHCGVYVPH
|
7.0 | IC50 | 3 | — | |
SKGLJORAKHJXMQ
|
7.0 | IC50 | 2 | — | |
UOJYAHYPXYXUMQ
|
7.0 | IC50 | 2 | — | |
DDHIANMDFDBMJW
|
7.0 | IC50 | 2 | — | |
MCTNGARCDMPDNT
|
6.9 | IC50 | 2 | — | |
VUXQRANDPGSPRS
|
6.9 | IC50 | 2 | — | |
ZVAPDTKXMZXVSP
|
6.9 | IC50 | 3 | — | |
VXFZOKLPMVMVEZ
|
6.8 | IC50 | 3 | — | |
LGZXNSNDFUQXOX
|
6.8 | IC50 | 2 | — | |
YPLCBNLGVGQEFT
|
6.8 | IC50 | 2 | — | |
AWKOHKZMMSJRFV
|
6.8 | IC50 | 2 | — | |
SGYSZCMQJNBMFO
|
6.7 | IC50 | 3 | — | |
YIQPUIGJQJDJOS
|
6.7 | IC50 | 5 | — | |
ZEUBXUYIRFFOOY
|
6.7 | IC50 | 2 | — | |
HCZHUJUTBCLSTK
|
6.6 | IC50 | 2 | — |