Target Details
| UniProt AC | P57078 |
|---|---|
| Gene Symbol | RIPK4 |
| Protein Name | Receptor-interacting serine/threonine-protein kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12796 (Ank_2) PF13637 (Ank_4) PF00069 (Pkinase) |
Summary
- Multi-target molecules 15
- Clinical molecules 5
- Avg pChEMBL 6.65
Active Molecules (15)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UIARLYUEJFELEN
|
7.9 | Kd | 289 | Yes | |
ASMLDRAEBPYENO
|
7.0 | IC50 | 10 | — | |
UJIAQDJKSXQLIT
|
7.0 | Kd | 38 | — | |
HKSZLNNOFSGOKW
|
7.0 | Kd | 408 | — | |
YYLKKYCXAOBSRM
|
6.9 | Kd | 191 | — | |
YRDHKIFCGOZTGD
|
6.8 | Kd | 21 | — | |
ODPGGGTTYSGTGO
|
6.7 | Kd | 153 | — | |
NHHQJBCNYHBUSI
|
6.7 | Kd | 220 | — | |
MFAQYJIYDMLAIM
|
6.5 | Kd | 130 | Yes | |
GCIKSSRWRFVXBI
|
6.5 | Kd | 109 | Yes | |
XZXHXSATPCNXJR
|
6.4 | Kd | 165 | Yes | |
UHTHHESEBZOYNR
|
6.2 | Kd | 66 | Yes | |
CXQHYVUVSFXTMY
|
6.0 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
6.0 | Kd | 149 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — |