Target Details
| UniProt AC | P57059 |
|---|---|
| Gene Symbol | SIK1 |
| Protein Name | Serine/threonine-protein kinase SIK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF23312 (UBA_SIK3) |
Summary
- Multi-target molecules 192
- Clinical molecules 11
- Avg pChEMBL 7.69
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (192)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BMGQWWVMWDBQGC
|
6.8 | Kd | 91 | Yes | |
CXQHYVUVSFXTMY
|
6.8 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
6.8 | Kd | 149 | — | |
HWSYLCVSNZMWCP
|
6.8 | IC50 | 3 | — | |
LXRITECWUGVGTD
|
6.8 | IC50 | 6 | — | |
HYMHVNNHIASECU
|
6.8 | IC50 | 5 | — | |
UWLKLAVEUJFHNV
|
6.7 | IC50 | 3 | — | |
XSGDOSCYEQRDBE
|
6.7 | IC50 | 3 | — | |
QHXBWJSQXSYAGG
|
6.7 | IC50 | 16 | — | |
XLSPYLMTRXPYKY
|
6.7 | IC50 | 13 | — | |
JWNPDZNEKVCWMY
|
6.7 | Kd | 57 | Yes | |
LHZJHTRTELKUDE
|
6.6 | IC50 | 2 | — | |
WRPKJPATUZRQFL
|
6.6 | IC50 | 3 | — | |
CHPOIFDTUJGSBW
|
6.6 | IC50 | 2 | — | |
JXJARIRMZQINMV
|
6.6 | IC50 | 3 | — | |
UKBGBACORPRCGG
|
6.6 | IC50 | 17 | — | |
LWHNEYJBIRCBSR
|
6.6 | IC50 | 3 | — | |
FNEDDGRJWXWDNZ
|
6.5 | IC50 | 5 | — | |
INSVCYRFDCTMIA
|
6.5 | IC50 | 5 | — | |
INDWAJWLSOYKGH
|
6.5 | IC50 | 3 | — | |
MFAQYJIYDMLAIM
|
6.5 | Kd | 130 | Yes | |
GMTZLHADUFDDDN
|
6.5 | IC50 | 5 | — | |
XELNNUJRQXCODY
|
6.4 | IC50 | 3 | — | |
MBBASLHNWYZIRZ
|
6.4 | IC50 | 3 | — | |
RGUMENUIWKKDQS
|
6.4 | IC50 | 3 | — | |
XASOHFCUIQARJT
|
6.4 | IC50 | 4 | — | |
CJGYTKZVACPSNS
|
6.4 | IC50 | 3 | — | |
RJLWSBWYWAAETQ
|
6.3 | IC50 | 3 | — | |
YZDJQTHVDDOVHR
|
6.3 | Kd | 23 | — | |
KSCBSHLEWGZVON
|
6.2 | IC50 | 4 | — | |
XUOIDCGCIMNQCG
|
6.2 | IC50 | 3 | — | |
ULGBXNOOIDGVSQ
|
6.2 | IC50 | 3 | — | |
XZXHXSATPCNXJR
|
6.2 | Kd | 165 | Yes | |
YYLKKYCXAOBSRM
|
6.2 | Kd | 191 | — | |
PJFVPKCPIJSWQT
|
6.2 | IC50 | 3 | — | |
NJMKEYLTIHAWEP
|
6.1 | IC50 | 3 | — | |
PMXGPFCKENCVOL
|
6.1 | IC50 | 3 | — | |
GTSDNTZRPRBMTP
|
6.1 | IC50 | 3 | — | |
ZMNVPNNTSQXNLO
|
6.1 | IC50 | 3 | — | |
SZGFJHKSBCTFLK
|
6.0 | IC50 | 3 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |