Target Details
| UniProt AC | P57059 |
|---|---|
| Gene Symbol | SIK1 |
| Protein Name | Serine/threonine-protein kinase SIK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF23312 (UBA_SIK3) |
Summary
- Multi-target molecules 192
- Clinical molecules 11
- Avg pChEMBL 7.69
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (192)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KZVDQIXBUFBWLM
|
7.6 | IC50 | 3 | — | |
CNFUDCYXMQHQFO
|
7.6 | IC50 | 3 | — | |
UKXHMXAKNAXPBS
|
7.5 | IC50 | 3 | — | |
CRLZGLXSANQWFT
|
7.5 | IC50 | 6 | — | |
QAMUWRFOZKONDU
|
7.5 | IC50 | 7 | — | |
UBPYILGKFZZVDX
|
7.5 | Kd | 130 | Yes | |
RTRHXDLGBINMNM
|
7.5 | IC50 | 5 | — | |
WWTRFWLRGARRAD
|
7.5 | IC50 | 10 | — | |
HRKJFKJZUNJKNU
|
7.5 | IC50 | 10 | — | |
TZEWBPGVTYPITP
|
7.5 | IC50 | 5 | — | |
ZBCMHWUFWQFPLV
|
7.5 | IC50 | 9 | — | |
SGMHSWUFNYQVBA
|
7.5 | IC50 | 9 | — | |
GRPZYURNHYVZBO
|
7.4 | IC50 | 3 | — | |
SIICZZZVCXGXGX
|
7.4 | IC50 | 3 | — | |
JOOXLOJCABQBSG
|
7.4 | Kd | 139 | — | |
XPSCTAWDRZNUCF
|
7.4 | IC50 | 3 | — | |
BYKVUESQXQHBEP
|
7.4 | IC50 | 7 | — | |
NZJCXRPMZJGVCC
|
7.3 | Kd | 8 | — | |
SHMKAHZOTDZUIN
|
7.3 | IC50 | 3 | — | |
OHQUFRHYRLCLFC
|
7.3 | IC50 | 3 | — | |
KNOCCCXGASNIAF
|
7.3 | IC50 | 3 | — | |
NHHQJBCNYHBUSI
|
7.3 | Kd | 220 | — | |
AEYQVJYAPMGHSF
|
7.3 | IC50 | 3 | — | |
QKNBRNSGPNCARD
|
7.3 | IC50 | 9 | — | |
BHFWGYATBPONNI
|
7.2 | IC50 | 3 | — | |
JPVJPXAQFGYJDI
|
7.2 | IC50 | 3 | — | |
CBLISIIXOMPZFZ
|
7.2 | IC50 | 3 | — | |
ZZSBPGIGIUFJRA
|
7.2 | Kd | 46 | — | |
QTBWCSQGBMPECM
|
7.2 | IC50 | 21 | Yes | |
WCLYSPWUHSZWOR
|
7.2 | IC50 | 3 | — | |
VCZDFACOFNRTMG
|
7.1 | IC50 | 6 | — | |
IDHYGWPCQJKIOG
|
7.1 | IC50 | 3 | — | |
MGMOBQWMSWOTLL
|
7.1 | IC50 | 3 | — | |
PBQKEWXFKZOWAZ
|
7.1 | IC50 | 3 | — | |
UIARLYUEJFELEN
|
7.1 | Kd | 289 | Yes | |
ZXYITDGKYOBFAO
|
7.1 | IC50 | 3 | — | |
XOZORSAAPNHXFP
|
7.1 | IC50 | 3 | — | |
DSKYHEJWWIBREA
|
7.0 | IC50 | 8 | — | |
ZGIZZXHFELWYTH
|
7.0 | IC50 | 3 | — | |
MYYIXDJCLRMEBI
|
7.0 | IC50 | 3 | — | |
LZUYOYKXEXENTQ
|
7.0 | IC50 | 5 | — | |
OFIFLUFVENTCNZ
|
7.0 | IC50 | 11 | — | |
YPGZOVPNRGMYIT
|
7.0 | IC50 | 3 | — | |
JDNFAAUUFUBZKC
|
7.0 | IC50 | 3 | — | |
CKVPYFIWJCSSSQ
|
6.9 | IC50 | 3 | — | |
NEHHEDJQRHQOOW
|
6.9 | IC50 | 5 | — | |
YHKXOSIWOVIDSP
|
6.9 | IC50 | 3 | — | |
ANQJLVHORSBOEP
|
6.8 | IC50 | 3 | — | |
XPJFDYHVVLGXHY
|
6.8 | IC50 | 3 | — | |
BMGQWWVMWDBQGC
|
6.8 | Kd | 147 | Yes |