Target Details
| UniProt AC | P57059 |
|---|---|
| Gene Symbol | SIK1 |
| Protein Name | Serine/threonine-protein kinase SIK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF23312 (UBA_SIK3) |
Summary
- Multi-target molecules 192
- Clinical molecules 11
- Avg pChEMBL 7.69
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (192)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZBNZXTGUTAYRHI
|
8.4 | Kd | 102 | Yes | |
UNBNKYSPLOMIOY
|
8.4 | IC50 | 7 | — | |
VCQQIZTUIHARTH
|
8.4 | IC50 | 3 | — | |
DEJPFOVGKKDPLD
|
8.3 | IC50 | 3 | — | |
KAUKMJZXRPFGAB
|
8.3 | IC50 | 3 | — | |
IVKGWWZSELOWKX
|
8.3 | IC50 | 3 | — | |
RGEJEFYGSBMYRS
|
8.3 | IC50 | 3 | — | |
PZFORNOVSGDEAS
|
8.3 | IC50 | 3 | — | |
IIRJOBJKMBEOMH
|
8.3 | IC50 | 3 | — | |
FZBVNCFBCNXULH
|
8.3 | IC50 | 18 | — | |
VNWAWEZKWMFEJY
|
8.2 | IC50 | 6 | — | |
NELFAFAXIZFQJB
|
8.2 | IC50 | 3 | — | |
FPNPNYBQZUNHGQ
|
8.2 | IC50 | 3 | — | |
HJHOVADSVUHROW
|
8.2 | IC50 | 3 | — | |
UKMGZRUGIXWOJQ
|
8.2 | IC50 | 3 | — | |
VAARYSWULJUGST
|
8.2 | Kd | 119 | Yes | |
VOYZWDQJVPQGCO
|
8.2 | IC50 | 9 | — | |
ARXQRVVEKOEUEV
|
8.2 | IC50 | 3 | — | |
OYDTWNVVTPPDDO
|
8.1 | IC50 | 3 | — | |
XIAKIYQZBHRETP
|
8.1 | IC50 | 3 | — | |
ZMAJVXKEVISHMQ
|
8.1 | IC50 | 9 | — | |
RXHXLESLBWUVQS
|
8.1 | IC50 | 3 | — | |
XCGUGTWHQADPNS
|
8.1 | IC50 | 3 | — | |
UGMDEPACJFWQTK
|
8.0 | IC50 | 3 | — | |
VQINULODWGEVBB
|
8.0 | IC50 | 4 | — | |
XGEBOBAOVSOQCV
|
8.0 | IC50 | 10 | — | |
DFZKXFCZKLBBRG
|
7.9 | IC50 | 3 | — | |
JKDJAOQUTMBBQB
|
7.9 | IC50 | 5 | — | |
SXMRTOWWEVQQSC
|
7.8 | IC50 | 3 | — | |
CAWABSRZIMATJO
|
7.8 | IC50 | 9 | — | |
DCDKXVMMAAIMRA
|
7.8 | IC50 | 3 | — | |
QQWUGDVOUVUTOY
|
7.8 | Kd | 231 | Yes | |
KCUIXXONNLBRFH
|
7.8 | IC50 | 3 | — | |
OLULSQINUASNMI
|
7.8 | IC50 | 3 | — | |
MMGVIQXQPXLHQK
|
7.8 | IC50 | 3 | — | |
QYFGVVMJUHWKNB
|
7.8 | IC50 | 3 | — | |
AZCVMDQKOWCQAG
|
7.8 | IC50 | 3 | — | |
XVNZURGXHLXJIR
|
7.8 | IC50 | 3 | — | |
JWADUJSXPDSTOX
|
7.7 | IC50 | 3 | — | |
DVQJNPZTPKFTFL
|
7.7 | IC50 | 3 | — | |
SVJBHQPXESBDEQ
|
7.7 | IC50 | 9 | — | |
UARVSLPFGRKWQN
|
7.7 | IC50 | 11 | — | |
FCJGMZMSVIAAJU
|
7.7 | IC50 | 9 | — | |
LZCGMQZFMKDCSR
|
7.7 | IC50 | 2 | — | |
WEHOIIGXTMKVRG
|
7.7 | IC50 | 3 | — | |
NQANXDMJOUTFBB
|
7.7 | IC50 | 3 | — | |
RIJYZTZQMRSSEU
|
7.7 | IC50 | 3 | — | |
MXJMJNRCJKHFPP
|
7.6 | IC50 | 10 | — | |
HJSKVVATRBELDD
|
7.6 | IC50 | 3 | — | |
CSZAJEXPQFERTK
|
7.6 | IC50 | 10 | — |